|
靶点/功能
|
产品名
|
编号
|
|
Cell Proliferation
|
CCK-8试剂盒
|
M4839
|
|
Inhibitor Cocktails
|
蛋白酶抑制剂Cocktail
|
M5293
|
|
Inhibitor Cocktails
|
磷酸酶抑制剂Cocktail
|
M7528
|
|
ACE
|
Enalapril maleate
|
M3543
|
|
AChR/AChE
|
Aclidinium bromide
|
M2368
|
|
AChR/AChE
|
Bethanechol chloride
|
M3309
|
|
AChR/AChE
|
Carbachol
|
M2489
|
|
AChR/AChE
|
Donepezil HCl
|
M3601
|
|
AChR/AChE
|
Hyoscyamine
|
M2762
|
|
AChR/AChE
|
Methscopolamine bromide
|
M3589
|
|
AChR/AChE
|
Oxybutynin chloride
|
M2909
|
|
AChR/AChE
|
PNU-282987
|
M3190
|
|
AChR/AChE
|
Rocuronium bromide
|
M2268
|
|
AChR/AChE
|
Solifenacin succinate
|
M3025
|
|
AChR/AChE
|
Tropicamide
|
M6040
|
|
ACL
|
BMS-303141
|
M3762
|
|
Adenosine Receptor
|
CGS 21680 HCl
|
M2282
|
|
AdipoR
|
AdipoRon
|
M2369
|
|
Adrenergic Receptor
|
Bambuterol HCl
|
M3662
|
|
Adrenergic Receptor
|
Esmolol HCl
|
M2682
|
|
Adrenergic Receptor
|
Formoterol hemifumarate
|
M5116
|
|
Adrenergic Receptor
|
Guanabenz acetate
|
M2738
|
|
Adrenergic Receptor
|
Isoprenaline HCl
|
M3186
|
|
Adrenergic Receptor
|
Methoxamine HCl
|
M2842
|
|
Adrenergic Receptor
|
Mirabegron
|
M2069
|
|
Adrenergic Receptor
|
Norepinephrine
|
M9264
|
|
Adrenergic Receptor
|
Propranolol HCl
|
M2964
|
|
AhR
|
CH-223191
|
M7727
|
|
Akt
|
GDC-0068
|
M1862
|
|
Akt
|
GSK690693
|
M1789
|
|
Akt
|
MK-2206 2HCl
|
M1837
|
|
Akt
|
Paeoniflorin
|
M3941
|
|
Akt
|
Perifosine
|
M1823
|
|
Akt
|
SC79
|
M5153
|
|
Akt
|
Triciribine
|
M1884
|
|
ALDH
|
Alda-1
|
M6423
|
|
ALDH
|
Disulfiram
|
M3390
|
|
ALK
|
ALK5 Inhibitor II
|
M1859
|
|
ALK
|
ASP3026
|
M1950
|
|
ALK
|
AZD3463
|
M2109
|
|
ALK
|
CH5424802
|
M1942
|
|
ALK
|
LDK378
|
M2075
|
|
ALK
|
LDN-193189
|
M1873
|
|
ALK
|
SB431542
|
M1794
|
|
RNA
|
N6-Methyladenosine
|
M5151
|
|
AMPK
|
A-769662
|
M3444
|
|
AMPK
|
AICAR
|
M4897
|
|
AMPK
|
Dorsomorphin 2HCl
|
M2238
|
|
AMPK
|
Metformin
|
M3244
|
|
Androgen Receptor
|
ARN-509
|
M2270
|
|
Androgen Receptor
|
Bicalutamide
|
M1960
|
|
Androgen Receptor
|
Dexmedetomidine HCl
|
M5565
|
|
Androgen Receptor
|
Dihydrotestosterone
|
M6033
|
|
Androgen Receptor
|
Galeterone
|
M2717
|
|
Androgen Receptor
|
Mesterolone
|
M3685
|
|
Androgen Receptor
|
Ostarine
|
M1973
|
|
Androgen Receptor
|
R1881
|
M8128
|
|
Androgen Receptor
|
RU 58841
|
M2344
|
|
Androgen Receptor
|
Spironolactone
|
M3028
|
|
Androgen Receptor
|
Testosterone
|
M6105
|
|
Angiotensin Receptor
|
Losartan potassium
|
M2258
|
|
Angiotensin Receptor
|
Tranilast
|
M6025
|
|
Antibiotics
|
Ampicillin sodium
|
M2390
|
|
Antibiotics
|
Carbenicillin disodium
|
M2491
|
|
Antibiotics
|
Ceftriaxone
|
M4916
|
|
Antibiotics
|
Chloramphenicol
|
M4901
|
|
Antibiotics
|
Clarithromycin
|
M3235
|
|
Antibiotics
|
Fidaxomicin
|
M2701
|
|
Antibiotics
|
G-418 disulfate
|
M2719
|
|
Antibiotics
|
Gentamycin sulfate
|
M3595
|
|
Antibiotics
|
Hygromycin B
|
M2761
|
|
Antibiotics
|
Kanamycin sulfate
|
M6229
|
|
Antibiotics
|
Lomefloxacin
|
M4941
|
|
Antibiotics
|
Methacycline HCl
|
M5777
|
|
Antibiotics
|
Metronidazole
|
M3311
|
|
Antibiotics
|
Minocycline HCl
|
M2854
|
|
Antibiotics
|
Monensin sodium salt
|
M6991
|
|
Antibiotics
|
Natamycin
|
M1958
|
|
Antibiotics
|
Penicillin G sodium
|
M5868
|
|
Antibiotics
|
Streptomycin sulfate
|
M4947
|
|
Antibiotics
|
Teicoplanin
|
M2009
|
|
Antibiotics
|
Tetracycline HCl
|
M3207
|
|
Antibiotics
|
Vancomycin HCl
|
M4862
|
|
Antifolate
|
Abitrexate
|
M2228
|
|
Antifolate
|
Pemetrexed
|
M7108
|
|
Anti-infection
|
Atovaquone
|
M2409
|
|
Anti-infection
|
Caspofungin acetate
|
M3726
|
|
Anti-infection
|
Cidofovir
|
M1695
|
|
Anti-infection
|
Clofazimine
|
M2528
|
|
Anti-infection
|
Entecavir monohydrate
|
M1707
|
|
Anti-infection
|
Ganciclovir
|
M5058
|
|
Anti-infection
|
Micafungin sodium
|
M3669
|
|
Anti-infection
|
Olsalazine disodium
|
M2898
|
|
Anti-infection
|
Ornidazole
|
M2900
|
|
Anti-infection
|
Oseltamivir
|
M1959
|
|
Anti-infection
|
PA-824
|
M2163
|
|
Anti-infection
|
Peramivir trihydrate
|
M3222
|
|
Anti-infection
|
Remdesivir
|
M3864
|
|
Anti-infection
|
Ribavirin
|
M3334
|
|
Anti-infection
|
Sulfadimethoxine
|
M1939
|
|
Anti-infection
|
Telbivudine
|
M3357
|
|
Antimetabolite
|
Thioguanine
|
M3258
|
|
Aromatase
|
Formestane
|
M3409
|
|
ATM/ATR
|
Candesartan Cilexetil
|
M3570
|
|
ATM/ATR
|
KU-55933
|
M1801
|
|
ATM/ATR
|
Mirin
|
M5138
|
|
ATM/ATR
|
VE-821
|
M2047
|
|
ATM/ATR
|
VE-822
|
M3115
|
|
ATPase
|
Sodium orthovanadate
|
M5161
|
|
Aurora Kinase
|
AZD1152-HQPA
|
M1663
|
|
Aurora Kinase
|
Hesperadin
|
M2127
|
|
Aurora Kinase
|
MLN8237
|
M1752
|
|
Aurora Kinase
|
PHA-739358
|
M1769
|
|
Aurora Kinase
|
TAK-901
|
M2154
|
|
Aurora Kinase
|
Tozasertib
|
M1881
|
|
Aurora Kinase
|
ZM447439
|
M1877
|
|
Autophagy
|
AS1842856
|
M9069
|
|
Autophagy
|
Bergapten
|
M2450
|
|
Autophagy
|
Bromocriptine mesylate
|
M2472
|
|
Autophagy
|
Capsaicin
|
M3422
|
|
Autophagy
|
Chloroquine
|
M9559
|
|
Autophagy
|
Curcumin
|
M2198
|
|
Autophagy
|
Dexamethasone
|
M2176
|
|
Autophagy
|
FK-506
|
M1934
|
|
Autophagy
|
Hydroxychloroquine sulfate
|
M5159
|
|
Autophagy
|
Hydroxyurea
|
M3291
|
|
Autophagy
|
Ivermectin
|
M2256
|
|
Autophagy
|
Letrozole
|
M3699
|
|
Autophagy
|
Melatonin
|
M2226
|
|
Autophagy
|
Mifepristone
|
M3510
|
|
Autophagy
|
Pemetrexed disodium
|
M2034
|
|
Autophagy
|
Rosuvastatin calcium
|
M2283
|
|
Autophagy
|
SBI-0206965
|
M6086
|
|
Autophagy
|
Silibinin
|
M5961
|
|
Autophagy
|
Simvastatin
|
M3497
|
|
Autophagy
|
SR9009
|
M5143
|
|
Autophagy
|
TBHQ
|
M9059
|
|
Autophagy
|
Vinorelbine tartrate
|
M3120
|
|
Axl
|
SGI-7079
|
M2180
|
|
Bcl-2
|
ABT-263
|
M1637
|
|
Bcl-2
|
ABT-737
|
M1638
|
|
Bcl-2
|
ABT-199
|
M2017
|
|
BET bromodomain
|
(+)-JQ1
|
M2167
|
|
BET bromodomain
|
CPI-203
|
M3526
|
|
BET bromodomain
|
OTX015
|
M2903
|
|
BET bromodomain
|
PFI-1
|
M2932
|
|
Calcium chelator
|
BAPTA-AM
|
M4973
|
|
Calcium chelator
|
EGTA
|
M9325
|
|
Calcium Channel
|
Acetylcholine chloride
|
M3317
|
|
Calcium Channel
|
Amlodipine
|
M5139
|
|
Calcium Channel
|
Cilnidipine
|
M2248
|
|
Calcium Channel
|
Felodipine
|
M3959
|
|
Calcium Channel
|
KB-R7943 mesylate
|
M1927
|
|
Calcium Channel
|
Levetiracetam
|
M2257
|
|
Calcium Channel
|
Lomerizine HCl
|
M2820
|
|
Calcium Channel
|
Manidipine 2HCl
|
M3296
|
|
Calcium Channel
|
Nifedipine
|
M3424
|
|
Calcium Channel
|
Verapamil HCl
|
M3118
|
|
Cannabinoid
|
Rimonabant
|
M2981
|
|
Cannabinoid
|
WIN 55212-2 mesylate
|
M3266
|
|
Caspase
|
Apoptosis Activator 2
|
M2403
|
|
Caspase
|
LY573636
|
M2551
|
|
Caspase
|
PAC-1
|
M1867
|
|
Caspase
|
VX-765
|
M3532
|
|
Cathepsin
|
Odanacatib
|
M1985
|
|
CCR
|
SB297006
|
M8254
|
|
CDK
|
AT7519 HCl
|
M3687
|
|
CDK
|
Flavopiridol
|
M1710
|
|
CDK
|
LEE011
|
M2218
|
|
CDK
|
LY2835219
|
M2112
|
|
CDK
|
Palbociclib
|
M6167
|
|
CDK
|
PD 0332991 HCL
|
M1806
|
|
CDK
|
PF-477736
|
M1764
|
|
CDK
|
R547
|
M1740
|
|
CDK
|
Roscovitine
|
M1974
|
|
CDK
|
SCH727965
|
M1807
|
|
CETP
|
Evacetrapib
|
M2330
|
|
CFTR
|
CFTRinh-172
|
M2504
|
|
CFTR
|
Lonidamine
|
M1923
|
|
CFTR
|
PTC124
|
M1771
|
|
CFTR
|
VX-770
|
M1854
|
|
CFTR
|
VX-809
|
M2102
|
|
Chk
|
AZD7762
|
M1665
|
|
c-Kit
|
Imatinib
|
M3241
|
|
c-Kit
|
Pexidartinib
|
M4867
|
|
c-Met
|
AMG-208
|
M1647
|
|
c-Met
|
AMG-458
|
M1745
|
|
c-Met
|
ARQ-197
|
M1811
|
|
c-Met
|
BMS-777607
|
M1682
|
|
c-Met
|
Foretinib
|
M1758
|
|
c-Met
|
INCB28060
|
M2080
|
|
c-Met
|
JNJ-38877605
|
M1793
|
|
c-Met
|
PF-04217903
|
M1766
|
|
c-Met
|
PF-2341066
|
M1765
|
|
c-Met
|
PHA-665752
|
M1899
|
|
c-Met
|
SGX523
|
M1777
|
|
c-Met
|
XL-184
|
M1757
|
|
c-Myc
|
10058-F4
|
M2352
|
|
COX
|
Acetaminophen
|
M3301
|
|
COX
|
Aspirin
|
M5426
|
|
COX
|
Celecoxib
|
M1965
|
|
COX
|
Firocoxib
|
M1830
|
|
COX
|
Indomethacin
|
M3466
|
|
CRM1
|
KPT-330
|
M3152
|
|
CSF-1R
|
BLZ945
|
M5316
|
|
CSF-1R
|
GW2580
|
M2743
|
|
CSF-1R
|
PLX5622
|
M9512
|
|
CXCR
|
Plerixafor
|
M1898
|
|
CXCR
|
SB225002
|
M3887
|
|
CXCR
|
WZ 811
|
M2041
|
|
CYP450
|
Abiraterone
|
M1636
|
|
CYP450
|
Anastrozole
|
M3708
|
|
CYP450
|
Apigenin
|
M6451
|
|
CYP450
|
MDV3100
|
M1839
|
|
CYP450
|
Memantine HCl
|
M3326
|
|
Dehydrogenase
|
AGI-5198
|
M2067
|
|
Dehydrogenase
|
Ammonium Glycyrrhizinate
|
M3571
|
|
Dehydrogenase
|
Daidzin
|
M4152
|
|
Dehydrogenase
|
SW033291
|
M4930
|
|
Deubiquitinase
|
b-AP15
|
M2431
|
|
DHPI
|
Cilastatin
|
M6090
|
|
DNA Methyltransferase
|
Decitabine
|
M2052
|
|
DNA Methyltransferase
|
RG108
|
M2182
|
|
DNA Methyltransferase
|
SGI-1027
|
M3008
|
|
DNA/RNA Synthesis
|
5-Fluorouracil
|
M2289
|
|
DNA/RNA Synthesis
|
Azacitidine
|
M2291
|
|
DNA/RNA Synthesis
|
Bleomycin sulfate
|
M2100
|
|
DNA/RNA Synthesis
|
Carboplatin
|
M2288
|
|
DNA/RNA Synthesis
|
Cisplatin
|
M2223
|
|
DNA/RNA Synthesis
|
CX-5461
|
M2293
|
|
DNA/RNA Synthesis
|
Cycloheximide
|
M4879
|
|
DNA/RNA Synthesis
|
Cyclophosphamide monohydrate
|
M3671
|
|
DNA/RNA Synthesis
|
Cytarabine
|
M2292
|
|
DNA/RNA Synthesis
|
Dacarbazine
|
M2216
|
|
DNA/RNA Synthesis
|
Gemcitabine
|
M5680
|
|
DNA/RNA Synthesis
|
Ifosfamide
|
M3742
|
|
DNA/RNA Synthesis
|
Mizoribine
|
M1921
|
|
DNA/RNA Synthesis
|
Nelarabine
|
M1916
|
|
DNA/RNA Synthesis
|
Oxaliplatin
|
M2290
|
|
DNA/RNA Synthesis
|
Psoralen
|
M4478
|
|
DNA/RNA Synthesis
|
Streptozotocin
|
M2082
|
|
DNA/RNA Synthesis
|
Temozolomide
|
M2129
|
|
Dopamine Receptor
|
Dopamine HCl
|
M5590
|
|
Dopamine Receptor
|
Fluphenazine 2HCl
|
M5198
|
|
DPP-4
|
Linagliptin
|
M2814
|
|
DPP-4
|
Sitagliptin phosphate monohydrate
|
M1967
|
|
Dynamin
|
Dynasore
|
M2569
|
|
E1/E2/E3 Enzyme
|
PYR-41
|
M2969
|
|
EGFR/HER2
|
AG-1478
|
M2312
|
|
EGFR/HER2
|
AZD8931
|
M1667
|
|
EGFR/HER2
|
AZD9291
|
M2424
|
|
EGFR/HER2
|
BIBW2992
|
M1677
|
|
EGFR/HER2
|
Canertinib
|
M1943
|
|
EGFR/HER2
|
CO-1686
|
M2212
|
|
EGFR/HER2
|
Dacomitinib
|
M1869
|
|
EGFR/HER2
|
Erlotinib
|
M5621
|
|
EGFR/HER2
|
Gefitinib
|
M1749
|
|
EGFR/HER2
|
Genistein
|
M2255
|
|
EGFR/HER2
|
Lapatinib
|
M3517
|
|
EGFR/HER2
|
Neratinib
|
M1913
|
|
EGFR/HER2
|
PD153035 HCl
|
M3689
|
|
EGFR/HER2
|
Taxifolin
|
M4585
|
|
EGFR/HER2
|
WZ4002
|
M1850
|
|
EGFR/HER2
|
WZ8040
|
M1851
|
|
Endothelin Receptor
|
Bosentan
|
M2467
|
|
Endothelin Receptor
|
Zibotentan
|
M1816
|
|
ERK
|
SCH772984
|
M2084
|
|
ERK
|
XMD17-109
|
M4819
|
|
ERK
|
XMD8-92
|
M6089
|
|
Estrogen Receptor
|
Chlorotrianisene
|
M3692
|
|
Estrogen Receptor
|
Cholesterol
|
M2516
|
|
Estrogen Receptor
|
Estradiol
|
M5625
|
|
Estrogen Receptor
|
Estrone
|
M3945
|
|
Estrogen Receptor
|
Fulvestrant
|
M1966
|
|
Estrogen Receptor
|
G15
|
M7871
|
|
Estrogen Receptor
|
Kaempferol
|
M4368
|
|
Estrogen Receptor
|
Tamoxifen
|
M7353
|
|
EZH2
|
EPZ-6438
|
M2677
|
|
EZH2
|
GSK126
|
M2114
|
|
FAAH
|
PF-3845
|
M3525
|
|
FAAH
|
URB597
|
M3404
|
|
Factor Xa
|
Apixaban
|
M1649
|
|
Factor Xa
|
Rivaroxaban
|
M1776
|
|
FAK
|
PF-562271
|
M2302
|
|
Farnesoid X Receptor
|
GW4064
|
M2018
|
|
Farnesoid X Receptor
|
INT-747
|
M3775
|
|
FAS
|
Orlistat
|
M3549
|
|
Ferroptosis
|
Deferoxamine mesylate
|
M5558
|
|
Ferroptosis
|
Erastin
|
M2679
|
|
Ferroptosis
|
Ferrostatin-1
|
M2698
|
|
Ferroptosis
|
Liproxstatin-1
|
M8531
|
|
FGFR
|
AZD4547
|
M1721
|
|
FGFR
|
BGJ398
|
M1840
|
|
FGFR
|
PD173074
|
M1875
|
|
FLT3
|
Gilteritinib
|
M7527
|
|
FLT3
|
KW-2449
|
M1815
|
|
Fluorescent Dye
|
D-Luciferin potassium salt
|
M8873
|
|
FTase
|
Tipifarnib
|
M1885
|
|
GABA Receptor
|
Nefiracetam
|
M3344
|
|
GCR
|
Budesonide
|
M2245
|
|
GCR
|
Hydrocortisone
|
M3451
|
|
GCR
|
Mometasone furoate
|
M3212
|
|
GLI
|
GANT58
|
M1812
|
|
GLI
|
GANT61
|
M2448
|
|
Glucosylceramide synthase
|
Eliglustat tartrate
|
M9733
|
|
GluR
|
Dizocilpine
|
M2646
|
|
GluR
|
(-)-Huperzine A
|
M3253
|
|
GluR
|
Ifenprodil tartrate
|
M2767
|
|
GluR
|
Perampanel
|
M5157
|
|
GluR
|
Topiramate
|
M4950
|
|
GPR
|
GSK1292263
|
M3321
|
|
GPR
|
GW9508
|
M2020
|
|
GPR
|
MBX-2982
|
M3632
|
|
GPR
|
TAK-875
|
M2054
|
|
GSK-3
|
AR-A014418
|
M2405
|
|
GSK-3
|
AZD1080
|
M2417
|
|
GSK-3
|
AZD2858
|
M2178
|
|
GSK-3
|
Bikinin
|
M8228
|
|
GSK-3
|
CHIR-99021
|
M1692
|
|
GTPase
|
NSC23766 3HCl
|
M2889
|
|
HCV Protease
|
ABT-333
|
M2333
|
|
HCV Protease
|
Boceprevir
|
M3624
|
|
HCV Protease
|
PSI-7977
|
M3666
|
|
HDAC
|
Belinostat
|
M1670
|
|
HDAC
|
CUDC-101
|
M1693
|
|
HDAC
|
CUDC-907
|
M2111
|
|
HDAC
|
EX 527
|
M1708
|
|
HDAC
|
ITF2357
|
M1730
|
|
HDAC
|
LBH589
|
M1748
|
|
HDAC
|
MGCD0103
|
M1790
|
|
HDAC
|
MS-275
|
M1791
|
|
HDAC
|
PCI-24781
|
M1813
|
|
HDAC
|
4-Phenylbutyric acid
|
M9638
|
|
HDAC
|
RGFP966
|
M2977
|
|
HDAC
|
Sodium butyrate
|
M5152
|
|
HDAC
|
Sodium Phenylbutyrate
|
M3022
|
|
HDAC
|
Trichostatin A
|
M1753
|
|
HDAC
|
Valproic acid sodium salt
|
M1876
|
|
HDAC
|
Vorinostat
|
M1780
|
|
Hedgehog
|
GDC-0449
|
M1713
|
|
Hepatocyte
|
FH1
|
M2700
|
|
HIF
|
BAY 87-2243
|
M4869
|
|
HIF
|
DMOG
|
M2558
|
|
HIF
|
FG-4592
|
M1726
|
|
HIF
|
IOX2
|
M2573
|
|
HIF
|
LW6
|
M9279
|
|
HIF
|
2-Methoxyestradiol
|
M1992
|
|
HIF
|
YC-1
|
M3991
|
|
Histamine Receptor
|
Cimetidine
|
M3385
|
|
Histamine Receptor
|
Ciproxifan maleate
|
M2088
|
|
Histamine Receptor
|
Lidocaine
|
M5741
|
|
Histamine Receptor
|
Pheniramine maleate
|
M2935
|
|
Histone demethylases
|
GSK J4 HCl
|
M2731
|
|
Histone demethylases
|
SP2509
|
M6143
|
|
HIV Protease
|
Atazanavir sulfate
|
M1657
|
|
HIV Protease
|
Darunavir ethanolate
|
M3568
|
|
HIV Protease
|
Dolutegravir sodium
|
M4824
|
|
HIV Protease
|
Lopinavir
|
M2158
|
|
HIV Protease
|
Raltegravir potassium
|
M5084
|
|
HIV Protease
|
Ritonavir
|
M2159
|
|
HMG-CoA Reductase
|
Atorvastatin calcium
|
M5430
|