M2206
|
TH-302 (Evofosfamide) |
TH-302是一种选择性低氧激活的前体药物，靶向作用于实体瘤的hypoxic区域，IC50为19 nM，在缺氧条件下比在有氧条件下细胞毒性增强270倍，细胞色素P450代谢稳定。 |
| M6098
|
Baicalein |
Baicalein（5,6,7-Trihydroxyflavone，Noroxylin，黄芩素）是一种存在于黄芩，木蝴蝶，百里香等植物中的天然黄酮类化合物，具有抗炎和抗癌活性。Baicalein可明显抑制PI3K/Akt/NF-κB途径，同时也可通过上调GPX4，抑制黑素细胞的铁死亡（ferroptosis），用于白癜风和肿瘤的相关研究。 |
| M9325
|
EGTA |
EGTA是一种特殊的钙离子螯合剂，在生理 pH 值 (7.4) 下，Kd 为 60.5 nM，对 Ca2+ 比对 Mg2+ 有很高的特异性。EGTA 显著抑制炎性巨噬细胞的底物粘附能力。 |
| M9330
|
Brij-35 |
Brij-35（月桂醇聚氧乙烯醚）是一种无毒的非离子表面活性剂，可降低非特定蛋白质的吸附，应用于红曲霉深层发酵时，能显著提高红曲色素产量。 |
| M6154
|
2-PMPA tetrasodium |
2-PMPA（PMPA tetrasodium salt）是高效选择性的谷氨酸羧肽酶II (GCPII)抑制剂，IC50值为300 pM。 |
| M2250
|
Pamidronate disodium |
Pamidronate Disodium（帕米膦酸二钠）是一种含氮的双磷酸盐类化合物，具有抑制骨吸收的作用，可用于癌症相关的溶骨性病变等研究。 |
| M9916
|
DPPH |
DPPH (2,2-Diphenyl-1-picrylhydrazyl，2,2-联苯基-1-苦基肼基) 是一种稳定的自由基，可用于测量抗氧化剂的自由基清除活性。 |
| M9194
|
Insulin (human) |
Insulin (human) 是一种多肽激素，其调节血液中的糖（葡萄糖）水平并且由胰岛的β细胞产生。 |
| M3409
|
Formestane |
Formestane（4-hydroxyandrostenedione，福美司坦）是第二代选择性芳香酶抑制剂，IC50为80 nM。 |
| M9665
|
N-(2-amino-2-oxoethyl)acrylamide |
N-(2-Amino-2-oxoethyl)acrylamide（N-acryloyl-glycinamide，丙烯酰基甘氨酰胺）是一种单体，其聚合物能制备水凝胶，并用于酶的固定化。 |
| M7036
|
Nonactin |
Nonactin is a monovalent cation ionophore. |
| M7033
|
NNC 05-2090 hydrochloride |
NNC 05-2090 hydrochloride is a gABA uptake inhibitor; moderately BGT-1 selective. |
| M7032
|
N-MPPP Hydrochloride |
N-MPPP Hydrochloride is a selective κ agonist. |
| M7028
|
Nicergoline |
Nicergoline is a α antagonist. |
| M7027
|
NI 42 |
NI 42 is a high affinity BRPF inhibitor. |
| M7026
|
NGB 2904 |
NGB 2904 is a potent and selective D
3 antagonist. |
| M7025
|
NFPS |
NFPS is a selective non-transportable GlyT1 inhibitor. |
| M7023
|
NDT 9513727 |
NDT 9513727 is a potent, selective human C5a receptor antagonist. |
| M7022
|
NCX 466 |
NCX 466 is a cyclooxygenase-inhibiting nitric oxide donor. |
| M7019
|
NBD 556 |
NBD 556 is a cD4 mimetic; blocks HIV-1 cell entry. |
| M7018
|
NAV 26 |
NAV 26 is a selective Na
v1.7 channel blocker. |
| M7017
|
NAS-181 |
NAS-181 is a selective r5-HT
1B antagonist. Active
in vivo. |
| M7014
|
Naltrindole hydrochloride |
Naltrindole hydrochloride is a selective non-peptide δ antagonist. |
| M7013
|
Naltriben mesylate |
Naltriben mesylate is a standard δ
2 selective antagonist. |
| M7011
|
NADA |
NADA is a endogenous CB
1 agonist. Also vanilloid agonist and inhibitor of FAAH and AMT. |
| M7010
|
N20C hydrochloride |
N20C hydrochloride is a non-competitive NMDA receptor open-channel blocker. |
| M7009
|
Muristerone A |
Muristerone A is a stimulates Bcl-XL mRNA transcription; antiapoptotic. |
| M7006
|
MSOP |
MSOP is a specific group III mGlu antagonist. |
| M7005
|
MS 245 oxalate |
MS 245 oxalate is a high affinity 5-HT
6 antagonist. |
| M7004
|
MS 21570 |
MS 21570 is a gPR171 antagonist. |
