M2206
|
TH-302 (Evofosfamide) |
TH-302是一种选择性低氧激活的前体药物，靶向作用于实体瘤的hypoxic区域，IC50为19 nM，在缺氧条件下比在有氧条件下细胞毒性增强270倍，细胞色素P450代谢稳定。 |
| M6098
|
Baicalein |
Baicalein（5,6,7-Trihydroxyflavone，Noroxylin，黄芩素）是一种存在于黄芩，木蝴蝶，百里香等植物中的天然黄酮类化合物，具有抗炎和抗癌活性。Baicalein可明显抑制PI3K/Akt/NF-κB途径，同时也可通过上调GPX4，抑制黑素细胞的铁死亡（ferroptosis），用于白癜风和肿瘤的相关研究。 |
| M9325
|
EGTA |
EGTA是一种特殊的钙离子螯合剂，在生理 pH 值 (7.4) 下，Kd 为 60.5 nM，对 Ca2+ 比对 Mg2+ 有很高的特异性。EGTA 显著抑制炎性巨噬细胞的底物粘附能力。 |
| M9330
|
Brij-35 |
Brij-35（月桂醇聚氧乙烯醚）是一种无毒的非离子表面活性剂，可降低非特定蛋白质的吸附，应用于红曲霉深层发酵时，能显著提高红曲色素产量。 |
| M6154
|
2-PMPA tetrasodium |
2-PMPA（PMPA tetrasodium salt）是高效选择性的谷氨酸羧肽酶II (GCPII)抑制剂，IC50值为300 pM。 |
| M2250
|
Pamidronate disodium |
Pamidronate Disodium（帕米膦酸二钠）是一种含氮的双磷酸盐类化合物，具有抑制骨吸收的作用，可用于癌症相关的溶骨性病变等研究。 |
| M9916
|
DPPH |
DPPH (2,2-Diphenyl-1-picrylhydrazyl，2,2-联苯基-1-苦基肼基) 是一种稳定的自由基，可用于测量抗氧化剂的自由基清除活性。 |
| M9194
|
Insulin (human) |
Insulin (human) 是一种多肽激素，其调节血液中的糖（葡萄糖）水平并且由胰岛的β细胞产生。 |
| M3409
|
Formestane |
Formestane（4-hydroxyandrostenedione，福美司坦）是第二代选择性芳香酶抑制剂，IC50为80 nM。 |
| M9665
|
N-(2-amino-2-oxoethyl)acrylamide |
N-(2-Amino-2-oxoethyl)acrylamide（N-acryloyl-glycinamide，丙烯酰基甘氨酰胺）是一种单体，其聚合物能制备水凝胶，并用于酶的固定化。 |
| M7176
|
Quin C1 |
Quin C1 is a potent and selective FPR2 agonist. |
| M7174
|
PTAC oxalate |
PTAC oxalate is a muscarinic receptor ligand; exhibits partial agonist and antagonist activity at different subtypes. |
| M7173
|
PT 1 |
PT 1 is a aMPK activator. |
| M7172
|
Psora 4 |
Psora 4 is a potent K
V1.3 channel blocker. |
| M7168
|
PSB 10 hydrochloride |
PSB 10 hydrochloride is a potent, highly selective hA
3 receptor antagonist/inverse agonist. |
| M7166
|
PSB 069 |
PSB 069 is a non-selective NTPDase inhibitor. |
| M7165
|
PS 1145 dihydrochloride |
PS 1145 dihydrochloride is a selective IKK inhibitor; orally active. |
| M7164
|
Proxyfan oxalate |
Proxyfan oxalate is a high affinity H
3 ligand. |
| M7162
|
Propranolol glycol |
Propranolol glycol is a Propranolol metabolite. |
| M7161
|
Proglumide sodium salt |
Proglumide sodium salt is a non-selective CCK antagonist; orally active. |
| M7159
|
Pregnenolone sulfate sodium salt |
Pregnenolone sulfate sodium salt is a nMDA Potentiator. |
| M7158
|
Pregnanolone |
Pregnanolone is a gABA
A receptor positive allosteric modulator. |
| M7157
|
PQ 69 |
PQ 69 is a potent and selective A
1 inverse agonist. |
| M7156
|
PPY A |
PPY A is a potent inhibitor of Abl T315l mutant and wild-type Abl kinases. |
| M7155
|
PPPA |
PPPA is a competitive NR2A antagonist. |
| M7154
|
PPDA |
PPDA is a subtype-selective NR2C/NR2D antagonist. |
| M7153
|
PP 3 |
PP 3是PP 2的阴性对照。 |
| M7151
|
Polygodial |
Polygodial is a tRPA1 channel activator; analgesic and antifungal. |
| M7150
|
PNU 96415E |
PNU 96415E is a d
4 and 5-HT
2A antagonist; antipsychotic. |
| M7149
|
PNU 37883 hydrochloride |
PNU 37883 hydrochloride is a vascular K
ir6 (K
ATP) channel blocker. |
