M2206
|
TH-302 (Evofosfamide) |
TH-302是一种选择性低氧激活的前体药物，靶向作用于实体瘤的hypoxic区域，IC50为19 nM，在缺氧条件下比在有氧条件下细胞毒性增强270倍，细胞色素P450代谢稳定。 |
| M6098
|
Baicalein |
Baicalein（5,6,7-Trihydroxyflavone，Noroxylin，黄芩素）是一种存在于黄芩，木蝴蝶，百里香等植物中的天然黄酮类化合物，具有抗炎和抗癌活性。Baicalein可明显抑制PI3K/Akt/NF-κB途径，同时也可通过上调GPX4，抑制黑素细胞的铁死亡（ferroptosis），用于白癜风和肿瘤的相关研究。 |
| M9325
|
EGTA |
EGTA是一种特殊的钙离子螯合剂，在生理 pH 值 (7.4) 下，Kd 为 60.5 nM，对 Ca2+ 比对 Mg2+ 有很高的特异性。EGTA 显著抑制炎性巨噬细胞的底物粘附能力。 |
| M9330
|
Brij-35 |
Brij-35（月桂醇聚氧乙烯醚）是一种无毒的非离子表面活性剂，可降低非特定蛋白质的吸附，应用于红曲霉深层发酵时，能显著提高红曲色素产量。 |
| M6154
|
2-PMPA tetrasodium |
2-PMPA（PMPA tetrasodium salt）是高效选择性的谷氨酸羧肽酶II (GCPII)抑制剂，IC50值为300 pM。 |
| M2250
|
Pamidronate disodium |
Pamidronate Disodium（帕米膦酸二钠）是一种含氮的双磷酸盐类化合物，具有抑制骨吸收的作用，可用于癌症相关的溶骨性病变等研究。 |
| M9916
|
DPPH |
DPPH (2,2-Diphenyl-1-picrylhydrazyl，2,2-联苯基-1-苦基肼基) 是一种稳定的自由基，可用于测量抗氧化剂的自由基清除活性。 |
| M9194
|
Insulin (human) |
Insulin (human) 是一种多肽激素，其调节血液中的糖（葡萄糖）水平并且由胰岛的β细胞产生。 |
| M3409
|
Formestane |
Formestane（4-hydroxyandrostenedione，福美司坦）是第二代选择性芳香酶抑制剂，IC50为80 nM。 |
| M9665
|
N-(2-amino-2-oxoethyl)acrylamide |
N-(2-Amino-2-oxoethyl)acrylamide（N-acryloyl-glycinamide，丙烯酰基甘氨酰胺）是一种单体，其聚合物能制备水凝胶，并用于酶的固定化。 |
| M7349
|
TAK 21d |
TAK 21d is a potent FAAH inhibitor. |
| M7348
|
TACA |
TACA is a gABA
A agonist. Also GABA-T substrate and GABA uptake inhibitor. |
| M7347
|
Tabimorelin hemifumarate |
Tabimorelin hemifumarate is a potent, orally active ghrelin receptor agonist. |
| M7345
|
T 98475 |
T 98475 is a gnRH receptor antagonist. |
| M7344
|
T 5601640 |
T 5601640 is a selective LIMK2 inhibitor; antitumor. |
| M7338
|
Sulfidefluor 7 AM |
Sulfidefluor 7 AM is a h
2S fluorescent probe. |
| M7337
|
STOCK2S 26016 |
STOCK2S 26016 is a lysine deficient protein kinase (WNK) signaling inhibitor. |
| M7335
|
STEARDA |
硬脂酰胺是一种内源性活性脂类
体内< em > < / em >。内香素对TRPV1受体的作用增强。 |
| M7334
|
ST 1936 oxalate |
ST 1936 oxalate is a selective, high affinity 5-HT
6 agonist. |
| M7333
|
SSR 69071 |
SSR 69071 is a potent, orally active human leukocyte elastase inhibitor. |
| M7332
|
SR 7826 |
SR 7826 is a potent and selective LIMK inhibitor; antitumor. |
| M7331
|
SR 57227 hydrochloride |
SR 57227 hydrochloride is a potent, selective 5-HT
3 agonist. |
| M7329
|
SR 3576 |
SR 3576 is a highly potent and selective JNK3 inhibitor. |
| M7328
|
SR 33805 oxalate |
SR 33805 oxalate is a ca
2+ channel blocker; binds allosterically to distinct site on L-type channels. |
| M7326
|
SR 142948 |
SR 142948 is a highly potent NT receptor antagonist. |
| M7324
|
SR 12813 |
SR 12813 is a pregnane X receptor agonist. |
| M7320
|
Spiperone hydrochloride |
Spiperone hydrochloride is a 5-HT
2A antagonist. Also D
2-like antagonist. |
| M7313
|
SN 2 |
SN 2 is a selective TRPML3 channel activator. |
| M7311
|
SMBA 1 |
SMBA 1 is a high affinity and selective activator of Bax. |
| M7310
|
SMANT hydrochloride |
SMANT hydrochloride is a inhibits Smoothened (Smo) accumulation. |
