M2206
|
TH-302 (Evofosfamide) |
TH-302是一种选择性低氧激活的前体药物,靶向作用于实体瘤的hypoxic区域,IC50为19 nM,在缺氧条件下比在有氧条件下细胞毒性增强270倍,细胞色素P450代谢稳定。 |
M6098
|
Baicalein |
Baicalein(5,6,7-Trihydroxyflavone,Noroxylin,黄芩素)是一种存在于黄芩,木蝴蝶,百里香等植物中的天然黄酮类化合物,具有抗炎和抗癌活性。Baicalein可明显抑制PI3K/Akt/NF-κB途径,同时也可通过上调GPX4,抑制黑素细胞的铁死亡(ferroptosis),用于白癜风和肿瘤的相关研究。 |
M9325
|
EGTA |
EGTA是一种特殊的钙离子螯合剂,在生理 pH 值 (7.4) 下,Kd 为 60.5 nM,对 Ca2+ 比对 Mg2+ 有很高的特异性。EGTA 显著抑制炎性巨噬细胞的底物粘附能力。 |
M9330
|
Brij-35 |
Brij-35(月桂醇聚氧乙烯醚)是一种无毒的非离子表面活性剂,可降低非特定蛋白质的吸附,应用于红曲霉深层发酵时,能显著提高红曲色素产量。 |
M6154
|
2-PMPA tetrasodium |
2-PMPA(PMPA tetrasodium salt)是高效选择性的谷氨酸羧肽酶II (GCPII)抑制剂,IC50值为300 pM。 |
M2250
|
Pamidronate disodium |
Pamidronate Disodium(帕米膦酸二钠)是一种含氮的双磷酸盐类化合物,具有抑制骨吸收的作用,可用于癌症相关的溶骨性病变等研究。 |
M9916
|
DPPH |
DPPH (2,2-Diphenyl-1-picrylhydrazyl,2,2-联苯基-1-苦基肼基) 是一种稳定的自由基,可用于测量抗氧化剂的自由基清除活性。 |
M9194
|
Insulin (human) |
Insulin (human) 是一种多肽激素,其调节血液中的糖(葡萄糖)水平并且由胰岛的β细胞产生。 |
M3409
|
Formestane |
Formestane(4-hydroxyandrostenedione,福美司坦)是第二代选择性芳香酶抑制剂,IC50为80 nM。 |
M9665
|
N-(2-amino-2-oxoethyl)acrylamide |
N-(2-Amino-2-oxoethyl)acrylamide(N-acryloyl-glycinamide,丙烯酰基甘氨酰胺)是一种单体,其聚合物能制备水凝胶,并用于酶的固定化。 |
M20085
|
WAY-320049 |
WAY-320049 can modulate mitochondrial reactive oxygen species production |
M20084
|
WAY-320008 |
WAY-320008 is a tropomyosin-related kinase a inhibitor |
M20083
|
WAY-313218 |
WAY-313218 is a 11β-hydroxysteroid dehydrogenase type 1 modulator |
M20081
|
WAY-312602 |
WAY-312602 is a maternal embryonic leucine zipper kinase inhibitor. |
M20080
|
WAY-312567 |
WAY-312567 is a Mycobacterium tuberculosis shikimate kinase inhibitor. |
M20079
|
WAY-312157 |
WAY-312157 has ATP-utilizing enzyme inhibitory activity |
M20078
|
WAY-311972 |
WAY-311972 is a inhibitor of ATP-kinases. |
M20076
|
WAY-310944 |
WAY-310944 is a Mycobacterium tuberculosis shikimate kinase inhibitor |
M20074
|
WAY-310507 |
WAY-310507 is a Mycobacterium tuberculosis shikimate kinase inhibitor. |
M20073
|
WAY-310334 |
WAY-310334 is a mPGES-1 inhibitor |
M20072
|
WAY-300442 |
WAY-300442 is a inhibitor of ATP-kinases. |
M20071
|
WAY-300385 |
WAY-300385 is a Mycobacterium tuberculosis shikimate kinase inhibitor. |
M20070
|
WAY-300062 |
WAY-300062 is a Mycobacterium tuberculosis shikimate kinase inhibitor. |
M20068
|
WAY-299590 |
WAY-299590 is a inhibitor against Mycobacterium tuberculosis Enoyl acyl carrier protein reductase |
M20067
|
WAY-299369 |
WAY-299369has inhibition of AR dimerization and/or DNA binding |
M20064
|
WAY-298350 |
WAY-298350 is a inhibitor of A kinase anchor protein/protein kinase A interaction. |
M20057
|
WAY-278559-A |
WAY-278559-A is a ethanolamine kinase inhibitor. |
M20054
|
WAY-278459-A |
WAY-278459-A is a inhibitor of wild type and mutant HIV-1 reverse transcriptase |
M20053
|
WAY-277054 |
WAY-277054 is a tyrosine kinase inhibitor |
M20052
|
WAY-273170 |
WAY-273170 is a Myt1 Kinase inhibitor. |