M2206
|
TH-302 (Evofosfamide) |
TH-302是一种选择性低氧激活的前体药物,靶向作用于实体瘤的hypoxic区域,IC50为19 nM,在缺氧条件下比在有氧条件下细胞毒性增强270倍,细胞色素P450代谢稳定。 |
M6098
|
Baicalein |
Baicalein(5,6,7-Trihydroxyflavone,Noroxylin,黄芩素)是一种存在于黄芩,木蝴蝶,百里香等植物中的天然黄酮类化合物,具有抗炎和抗癌活性。Baicalein可明显抑制PI3K/Akt/NF-κB途径,同时也可通过上调GPX4,抑制黑素细胞的铁死亡(ferroptosis),用于白癜风和肿瘤的相关研究。 |
M9325
|
EGTA |
EGTA是一种特殊的钙离子螯合剂,在生理 pH 值 (7.4) 下,Kd 为 60.5 nM,对 Ca2+ 比对 Mg2+ 有很高的特异性。EGTA 显著抑制炎性巨噬细胞的底物粘附能力。 |
M9330
|
Brij-35 |
Brij-35(月桂醇聚氧乙烯醚)是一种无毒的非离子表面活性剂,可降低非特定蛋白质的吸附,应用于红曲霉深层发酵时,能显著提高红曲色素产量。 |
M6154
|
2-PMPA tetrasodium |
2-PMPA(PMPA tetrasodium salt)是高效选择性的谷氨酸羧肽酶II (GCPII)抑制剂,IC50值为300 pM。 |
M2250
|
Pamidronate disodium |
Pamidronate Disodium(帕米膦酸二钠)是一种含氮的双磷酸盐类化合物,具有抑制骨吸收的作用,可用于癌症相关的溶骨性病变等研究。 |
M9916
|
DPPH |
DPPH (2,2-Diphenyl-1-picrylhydrazyl,2,2-联苯基-1-苦基肼基) 是一种稳定的自由基,可用于测量抗氧化剂的自由基清除活性。 |
M9194
|
Insulin (human) |
Insulin (human) 是一种多肽激素,其调节血液中的糖(葡萄糖)水平并且由胰岛的β细胞产生。 |
M3409
|
Formestane |
Formestane(4-hydroxyandrostenedione,福美司坦)是第二代选择性芳香酶抑制剂,IC50为80 nM。 |
M9665
|
N-(2-amino-2-oxoethyl)acrylamide |
N-(2-Amino-2-oxoethyl)acrylamide(N-acryloyl-glycinamide,丙烯酰基甘氨酰胺)是一种单体,其聚合物能制备水凝胶,并用于酶的固定化。 |
M20249
|
WAY-637493 |
WAY-637493 is a Fyn kinase inhibitor. |
M20240
|
WAY-634964 |
WAY-634964 is a tyrosine kinase inhibitor. |
M20231
|
WAY-632021 |
WAY-632021 is a TIE-2 and Raf kinase inhibitor |
M20230
|
WAY-631545 |
WAY-631545 is a protein kinase inhibitor |
M20218
|
WAY-620147 |
WAY-620147 is a monoamine oxidase a inhibitor |
M20217
|
WAY-620099 |
WAY-620099 is a tyrosine kinase inhibitor |
M20216
|
WAY-619999 |
WAY-619999 is a inhibitor of CK2 and GSK3β. |
M20214
|
WAY-616763 |
WAY-616763 is a Inhibitor of T. brucei and T. cruzi Phosphofructokinase. |
M20211
|
WAY-615029 |
WAY-615029 is a Kinase Inhibitor. |
M20207
|
WAY-612763 |
WAY-612763 is a altering the lifespan of eukaryotic organisms |
M20206
|
WAY-612698 |
WAY-612698 is a altering the lifespan of eukaryotic organisms |
M20204
|
WAY-612453 |
WAY-612453 is a Mycobacterium tuberculosis shikimate kinase inhibitor. |
M20202
|
WAY-607738 |
WAY-607738 is a inhibitor of Mcl-1 |
M20200
|
WAY-607324 |
WAY-607324 is a inhibitor of Mcl-1 |
M20188
|
WAY-602219 |
WAY-602219 is a Trypanosoma brucei hexokinase inhibitor |
M20186
|
WAY-601258 |
WAY-601258 is a Mycobacterium tuberculosis shikimate kinase inhibitor. |
M20178
|
WAY-384934 |
WAY-384934 is a inhibitor of pyruvate kinase |
M20176
|
WAY-382818 |
WAY-382818 has mitogen-activated protein kinase phosphatase-1 inhibitory activity. |
M20174
|
WAY-359594 |
WAY-359594 inhibiting G protein coupled receptor 6 kinase. |
M20172
|
WAY-358667-A |
WAY-358667-A is a inhibitor of human protein kinase CK2 |