找到约 59 条 “Gly6” 相关结果 (用时 0.113 秒)

目录号 产品名称 中文名称 靶点
M12591 ChemBridge-6146494 ChemBridge化合物-6146494 Screening Compounds and Building Blocks
N-[3-(3-bromophenyl)-2-(2-furoylamino)acryloyl]glycine (6146494)
ChemBridge特有类药化合物/先导化合物-6146494,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M12625 ChemBridge-6220207 ChemBridge化合物-6220207 Screening Compounds and Building Blocks
N~1~-(2-bromophenyl)-N~2~-(4-ethoxyphenyl)-N~2~-(methylsulfonyl)glycinamide (6220207)
ChemBridge特有类药化合物/先导化合物-6220207,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M12671 ChemBridge-6402712 ChemBridge化合物-6402712 Screening Compounds and Building Blocks
N~1~-cyclopropyl-N~2~-(4-ethoxyphenyl)-N~2~-[(4-methylphenyl)sulfonyl]glycinamide (6402712)
ChemBridge特有类药化合物/先导化合物-6402712,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M12674 ChemBridge-6432139 ChemBridge化合物-6432139 Screening Compounds and Building Blocks
N-methyl-N-(6-nitro-1,3-benzothiazol-2-yl)glycine (6432139)
ChemBridge特有类药化合物/先导化合物-6432139,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M12768 ChemBridge-6723028 ChemBridge化合物-6723028 Screening Compounds and Building Blocks
ethyl 2-{[N-(2,3-dimethylphenyl)-N-(phenylsulfonyl)glycyl]amino}benzoate (6723028)
ChemBridge特有类药化合物/先导化合物-6723028,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M12771 ChemBridge-6739985 ChemBridge化合物-6739985 Screening Compounds and Building Blocks
methyl 2-({N-(2-methoxyphenyl)-N-[(4-methylphenyl)sulfonyl]glycyl}amino)benzoate (6739985)
ChemBridge特有类药化合物/先导化合物-6739985,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M12782 ChemBridge-6809058 ChemBridge化合物-6809058 Screening Compounds and Building Blocks
N-[4-(methylsulfonyl)-2-nitrophenyl]glycine (6809058)
ChemBridge特有类药化合物/先导化合物-6809058,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M12905 ChemBridge-7361080 ChemBridge化合物-7361080 Screening Compounds and Building Blocks
N-cyclohexyl-N-[(4-fluorophenyl)sulfonyl]glycine (7361080)
ChemBridge特有类药化合物/先导化合物-7361080,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M12909 ChemBridge-7402683 ChemBridge化合物-7402683 Screening Compounds and Building Blocks
methyl N-[4-(tert-butylamino)-6-(ethylamino)-1,3,5-triazin-2-yl]-N-cyanoglycinate (7402683)
ChemBridge特有类药化合物/先导化合物-7402683,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M14813 GPRP acetate GPRP acetate Peptides
Gly-Pro-Arg-Pro acetate; Pefa 6003 acetate
GPRP acetate (Gly-Pro-Arg-Pro acetate) 是一种纤维蛋白聚合抑制剂, 能够抑制纤维蛋白原与血小板膜糖蛋白 Ⅱb/IIIa 复合物(糖蛋白 IIb/IIIa 受体)之间的相互作用。
M24887 Torapsel Torapsel Others
42-89-glycoprotein; WAY164339; pMT21:PL85
Torapsel (42-89-glycoprotein; WAY164339) 是一种与免疫球蛋白融合的蛋白。Torapsel 可用于研究缺血再灌注损伤的预防。
M30472 GPRP GPRP Integrin
Gly-Pro-Arg-Pro; Pefa 6003
GPRP 是一种纤维蛋白聚合抑制剂,能够抑制纤维蛋白原与血小板膜糖蛋白 Ⅱb/IIIa 复合物(糖蛋白 IIb/IIIa 受体)之间的相互作用。
M45637 ChemBridge-5634520 ChemBridge化合物-5634520 Screening Compounds and Building Blocks
methyl N-(4-methylphenyl)-N-(methylsulfonyl)glycinate (5634520)
ChemBridge特有类药化合物/先导化合物-5634520,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M45776 ChemBridge-6012256 ChemBridge化合物-6012256 Screening Compounds and Building Blocks
N~1~-cyclopentyl-N~2~-(3,4-dimethoxyphenyl)-N~2~-[(4-methylphenyl)sulfonyl]glycinamide (6012256)
ChemBridge特有类药化合物/先导化合物-6012256,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M45845 ChemBridge-6187162 ChemBridge化合物-6187162 Screening Compounds and Building Blocks
N~1~-cyclopentyl-N~2~-(3-methoxyphenyl)-N~2~-(phenylsulfonyl)glycinamide (6187162)
ChemBridge特有类药化合物/先导化合物-6187162,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M45859 ChemBridge-6226431 ChemBridge化合物-6226431 Screening Compounds and Building Blocks
methyl N-(2-ethylphenyl)-N-(methylsulfonyl)glycinate (6226431)
ChemBridge特有类药化合物/先导化合物-6226431,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M45896 ChemBridge-6388833 ChemBridge化合物-6388833 Screening Compounds and Building Blocks
N~1~-bicyclo[2.2.1]hept-2-yl-N~2~-(3-methoxyphenyl)-N~2~-[(4-methylphenyl)sulfonyl]glycinamide (6388833)
ChemBridge特有类药化合物/先导化合物-6388833,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M45898 ChemBridge-6403648 ChemBridge化合物-6403648 Screening Compounds and Building Blocks
N~1~-bicyclo[2.2.1]hept-2-yl-N~2~-(3-methoxyphenyl)-N~2~-(phenylsulfonyl)glycinamide (6403648)
ChemBridge特有类药化合物/先导化合物-6403648,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M45918 ChemBridge-6460000 ChemBridge化合物-6460000 Screening Compounds and Building Blocks
N~1~-bicyclo[2.2.1]hept-2-yl-N~2~-(3,4-dimethoxyphenyl)-N~2~-(phenylsulfonyl)glycinamide (6460000)
ChemBridge特有类药化合物/先导化合物-6460000,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M45967 ChemBridge-6664973 ChemBridge化合物-6664973 Screening Compounds and Building Blocks
N~2~-benzyl-N~2~-[(2,5-dichlorophenyl)sulfonyl]-N~1~-methylglycinamide (6664973)
ChemBridge特有类药化合物/先导化合物-6664973,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M45989 ChemBridge-6792161 ChemBridge化合物-6792161 Screening Compounds and Building Blocks
N~2~-benzyl-N~2~-[(2,5-dichlorophenyl)sulfonyl]glycinamide (6792161)
ChemBridge特有类药化合物/先导化合物-6792161,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M45996 ChemBridge-6817802 ChemBridge化合物-6817802 Screening Compounds and Building Blocks
N~1~-[4-(anilinosulfonyl)phenyl]-N~2~-(4-methoxyphenyl)-N~2~-(methylsulfonyl)glycinamide (6817802)
ChemBridge特有类药化合物/先导化合物-6817802,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M46049 ChemBridge-7016027 ChemBridge化合物-7016027 Screening Compounds and Building Blocks
N-(4-bromophenyl)-2-{[N-(2-hydroxyethyl)glycyl]amino}-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxamide (7016027)
ChemBridge特有类药化合物/先导化合物-7016027,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M46128 ChemBridge-7356480 ChemBridge化合物-7356480 Screening Compounds and Building Blocks
N-benzyl-N-[(2,5-dichlorophenyl)sulfonyl]glycine (7356480)
ChemBridge特有类药化合物/先导化合物-7356480,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M46190 ChemBridge-7636042 ChemBridge化合物-7636042 Screening Compounds and Building Blocks
N~1~-2-biphenylyl-N~2~-(2,3-dihydro-1,4-benzodioxin-6-yl)-N~2~-(methylsulfonyl)glycinamide (7636042)
ChemBridge特有类药化合物/先导化合物-7636042,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M46246 ChemBridge-7742661 ChemBridge化合物-7742661 Screening Compounds and Building Blocks
N~1~-bicyclo[2.2.1]hept-2-yl-N~2~-(2,3-dihydro-1,4-benzodioxin-6-yl)-N~2~-(phenylsulfonyl)glycinamide (7742661)
ChemBridge特有类药化合物/先导化合物-7742661,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M48121 ChemBridge-44647926 ChemBridge化合物-44647926 Screening Compounds and Building Blocks
N~1~-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-N~2~-methylglycinamide (44647926)
ChemBridge特有类药化合物/先导化合物-44647926,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M48681 ChemBridge-67485854 ChemBridge化合物-67485854 Screening Compounds and Building Blocks
7-(1,3-benzothiazol-2-yl)-4-glycyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol hydrochloride (67485854)
ChemBridge特有类药化合物/先导化合物-67485854,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M48807 ChemBridge-73521846 ChemBridge化合物-73521846 Screening Compounds and Building Blocks
N~1~-(biphenyl-4-ylmethyl)-N~2~-methyl-N~2~-piperidin-4-ylglycinamide (73521846)
ChemBridge特有类药化合物/先导化合物-73521846,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M49283 ChemBridge-96305102 ChemBridge化合物-96305102 Screening Compounds and Building Blocks
4-(N,N-dimethylglycyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol (96305102)
ChemBridge特有类药化合物/先导化合物-96305102,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M1845 LY335979 trihydrochloride 唑喹达三盐酸盐 P-glycoprotein
Zosuquidar trihydrochloride; RS 33295-198 trihydrochloride
Zosuquidar (LY335979) 3HCl是一种有效的P-glycoprotein(P-糖蛋白)介导的多药耐抗性的调节剂,Ki为60 nM。
M3909 Glycyrrhizic acid 甘草酸;甘草甜素 HMGB1
NSC 167409; Glycyrrhizin
Glycyrrhizic acid (NSC 167409) 是一种直接的高迁移率族蛋白1(HMGB1)的抑制剂,抑制依赖于HMGB1的炎症分子表达和氧化应激反应。Glycyrrhizic acid的生物活性代谢物是甘草次酸,Glycyrrhizic acid是11-β-羟基类固醇脱氢酶有效抑制剂。
M5881 Piperine 胡椒碱 P-glycoprotein
Bioperine; 1-Piperoylpiperidine
Piperine是从胡椒中分离的天然生物碱,可以抑制P-glycoprotein and CYP3A4的活性,在HeLa细胞中的IC50值为61.94±0.054 μg/mL。
M11233 Recombinant Human KRAS(G12C, His, E.coli) 重组人 KRAS 蛋白 G12C( His, E.coli) Cytokines and Growth Factors
Ki-Ras; c-K-ras; KRAS2
重组人 KRAS 蛋白 (G12C, His) 由大肠杆菌表达系统产生,编码 Thr2-Cys185(Gly12Cys) 的靶基因在 N 末端用 6His 标签表达。
M8662 PDD00017273 PDD00017273 Others
PDD-17273
PDD00017273 是一种有效的、选择性的聚(ADP-核糖)糖水解酶 poly (ADP ribose) glycohydrolase (PARG)抑制剂,IC50为26 nM。PDD00017273催化 ADP-核糖聚合物的 O-糖苷键的水解,逆转聚(ADP-核糖)聚合酶 (PARP) 的作用。
M11496 FGF-basic, Rat (E. coli) FGF-basic, Rat (E. coli) Cytokines and Growth Factors
Fibroblast Growth Factor-basic; FGF-2; BFGF; FGFB; HBGF-2; bFGF; Prostatropin
FGF-basic, Rat(E. coli) 蛋白构造:Expressed with an N-terminal Gly.FGF-basic (Pro10-Ser154) Accession # P13109。 生物活性:ED50 < 0.25 ng/ml,采用3T3细胞增殖法测定,对应> 4.0 × 106单位/mg。
M13442 Recombinant Mouse IL-36 gamma (E.coli) 重组小鼠 IL-36 gamma蛋白(E.coli) Cytokines and Growth Factors
IL-36 gamma(E.coli)
重组小鼠IL-36 γ由我们的大肠杆菌表达系统产生,并表达了编码Gly13-Ser164的目的基因。
M19968 Glycol chitosan 乙二醇壳聚糖;羟乙基脱乙酰壳多糖 Anti-infection
Glycol chitin; deacetylated
Glycol chitosan 乙二醇壳聚糖是一种具有亲水性乙二醇分支的壳聚糖衍生物。乙二醇壳聚糖增强甘氨酸max Harosoy 63W细胞的膜渗透性和铅。
M15078 Recombinant Mouse Noggin/NOG (HEK293,C-6His) 重组小鼠Noggin/NOG蛋白 (HEK293,C-6His) Cytokines and Growth Factors
Noggin; Nog
Noggin is a secreted homodimeric glycoprotein that is an antagonist of bone morphogenetic proteins (BMPs). Noggin binds some BMPs such as BMP4 with high affinity and others such as BMP7 with lower affinity. It antagonizes BMP bioactivities by blocking epitopes on BMPs that are needed for binding to both type I and type II receptors. Accession # : P97466.
M15084 Recombinant Mouse Sonic Hedgehog/Shh (E.coli) 重组小鼠 Sonic Hedgehog/Shh 蛋白(E.coli) Cytokines and Growth Factors
Sonic Hedgehog Protein; SHH; HHG-1; SHH
利用大肠杆菌表达系统制备了重组小鼠Sonic Hedgehog基因,并表达了编码Cys25-Gly198的目的基因。Accession #: Q62226。
M16107 Glycozolinine 3-甲基-6-羟基咔唑 Alkaloids
Glycozolinine 3-甲基-6-羟基咔唑
M18181 6,7,4'-Trihydroxyisoflavone 6,7,4'-三羟基异黄酮 CDK
Desmethylglycitein (4',6,7-Trihydroxyisoflavone),大豆苷元的代谢产物,来源于大豆 Glycine max,具有抗氧化性和抗癌活性。
M20644 TH34 TH34 HDAC
TH34 is a HDAC inhibitor that shows pronounced selectivity for HDACs 6, 8 and 10 over HDACs 1, 2 and 3. In a NanoBRET assay, TH34 strongly binds HDAC6, 8 and 10 with low-micromolar IC50 concentrations (HDAC6: 4.6 µM, HDAC8: 1.9 µM, HDAC10: 7.7 µM).
M21677 Recombinant Human Follistatin 288 (HEK293, C-6His) 重组人Follistatin 288 蛋白 (HEK293, C-6His) Cytokines and Growth Factors
FST; follistatin isoform FST317
Follistatin 288 是一种分泌型糖蛋白,为卵巢卵泡液中的促卵泡激素抑制物质。人卵泡抑素 288 cDNA 编码具有 29 个氨基酸信号序列和 288 个氨基酸成熟区的 317 个氨基酸 (aa) 蛋白。重组人卵泡抑素/FST 由哺乳动物表达系统产生,编码 Gly30-Asn317 的靶基因在 C 末端用 6His 标签表达。
M21202 Recombinant Human Lipocalin-2/NGAL/LCN2 (E. coli, C-6His) 重组人Lipocalin-2/NGAL/LCN2 蛋白 (E. coli, C-6His) Cytokines and Growth Factors
Neutrophil gelatinase-associated lipocalin; NGAL
人中性粒细胞明胶酶相关脂质运载蛋白(Lipocalin-2/NGAL/LCN2)由大肠杆菌表达系统生产,编码Gln21-Gly198的目标基因在C端有一个6His标签。Protein number:P80188。
M21448 Recombinant Mouse IL-15RA (HEK293, C-Fc) 重组小鼠IL-15RA 蛋白 (HEK293, C-Fc) Cytokines and Growth Factors
Interleukin-15 receptor subunit alpha
重组小鼠白细胞介素15受体亚基α由哺乳动物表达系统产生,编码Gly33-Lys205的目标基因在c端带有Fc标签表达。蛋白编号:Q60819。
M21664 Recombinant Human F13A (HEK293, C-6His) 重组人凝血因子 XIII A 链蛋白 (HEK293, C-6His) Cytokines and Growth Factors
Coagulation Factor XIII A Chain
重组人凝血因子 XIII A 链 (F13A) 由哺乳动物表达系统产生,编码 Gly39-Met732 的靶基因在 C 端用 6His 标签表达。凝血因子 XIII 是凝血级联反应中最后激活的酶原。血浆因子 XIII 是由 2 个 A 亚基和 2 个 B 亚基组成的异四聚体。A亚基具有催化功能,B亚基不具有酶活性。
M25536 Recombinant Human CXCL13/BCA-1 (E. coli) 重组人CXCL13/BCA-1蛋白 (E. coli) Cytokines and Growth Factors
CXC chemokine BLC; Small-inducible cytokine B13
CXCL13, also known as B-lymphocyte chemoattractant (BLC), is a CXC chemokine that is constitutively expressed in secondary lymphoid organs. Recombinant human CXCL13 is a single non-glycosylated polypeptide chain containing 87 amino acids and mature human BCA-1 shares 64 % amino acid sequence similarity with the murine protein and 23–34 % amino acid sequence identity with other known CXC chemokines. Determined by a chemotaxis bioassay using human B cells, the biological activity is in a concentration range of 1.0-10 ng/ml.
M28216 6''-O-Acetylglycitin  6''-O-Acetylglycitin  Others
6''-O-Acetylglycitin 6''-O-乙酰黄豆黄苷是一种乙酰基葡萄糖苷,大豆异黄酮异构体之一,其含量根据储存温度,包装条件和异黄酮异构体种类不同会显示出不同程度的含量降低。
M31176 Recombinant Human CD40L Protein (E. coli) 重组人CD40L蛋白 (E. coli) Cytokines and Growth Factors
CD40 Ligand; CD154; TRAP
CD40 Ligand (CD40L/CD154/TRAP) is a type II transmembrane glycoprotein that belongs to the TNF superfamily. The CD40 ligand stimulates B-cell proliferation and secretion of all immunoglobulin isotypes in the presence of cytokines. Recombinant Human CD40 Ligand is produced by E.coli expression system and the target gene encoding Met113-Leu261 is expressed.
M38644 Stearyl glycyrrhetinate 硬脂醇甘草亭酸酯 Antibiotic
Stearyl glycyrrhetinate 是甘草提取物中的主要成分之一,对金黄色葡萄球菌菌株的 MIC 大于 256 mg/L。Stearyl glycyrrhetinate 具有抗菌 (antibacterial) 作用。
M38776 1-(26-Hydroxyhexacosanoyl)-glycerol 1-(26-Hydroxyhexacosanoyl)-glycerol Parasite
1-(26-Hydroxyhexacosanoyl)-glycerol 是一种有效的抗疟剂。1-(26-Hydroxyhexacosanoyl)-glycerol 具有抗疟活性,对 Plasmodium falciparum 的 IC50 值为 9.48 µM。
M39028 Picrotin 苦亭 GABA Receptor
Picrotin 是一种活性化合物,也是 picrotoxin(GABAA 受体 (GABAARs) 和甘氨酸受体 (GlyRs) 的拮抗剂)的成分之一。Picrotin 对甘氨酸受体 (GlyRs) 具有敏感性,IC50 值范围为 5.2 μM 至 106 μM。
M39059 Isoglycycoumarin Isoglycycoumarin Cytochrome P450 (e.g. CYP17)
Isoglycycoumarin 是从Glycyrrhiza uralensis 根中提取的黄酮类化合物。Isoglycycoumarin 是一种高度选择性的人细胞色素 P450 2A6 (CYP2A6) 探针。
M39972 Notoginsenoside T5 Notoginsenoside T5 Others
Notoginsenoside T5 是一种 dammarane 61 glycoside. Notoginsenoside T5 是从 P. 62 notoginseng 的根皂苷酸性脱糖基中分离出来的。
M40606 Recombinant Human C5a Protein (E.coli) 重组人补体C5a (E.coli) Cytokines and Growth Factors
Complement C5; C5a anaphylatoxin
Human Complement 5a (C5a) is an enzymatically generated glycoprotein that belongs to a family of structurally and functionally related proteins known as anaphylatoxins. Recombinant Human C5a expressed the target gene encoding Thr678-Arg751.
M42282 Dehydroglyasperin D Dehydroglyasperin D Aldose Reductase
DeHydroglyasperin D 抑制大鼠和人醛糖还原酶 (Aldose Reductase (AR)) (IC50 分别为 62.4 μM 和 176.2μM)。
M45395 1-Oleoyl-2-hydroxy-sn-glycero-3-phosphoethanolamine 1-Oleoyl-2-hydroxy-sn-glycero-3-phosphoethanolamine Others
1-Oleoyl-2-hydroxy-sn-glycero-3-phosphoethanolamine是溴氰菊酯在体外被原核蛋白(CYP6A14和CYP6N6)复合物代谢的主要降解产物。
M50815 Cbz-Glu-Gly-OH Cbz-Glu-Gly-OH Others
Cbz-Glu-Gly-OH (NSC 186902) 是一种多肽,能够由多肽筛选发现。








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