Others 抑制剂/激活剂/调节剂 Others

目录号 产品名称 产品简介
M6098 Baicalein Baicalein(5,6,7-Trihydroxyflavone,Noroxylin,黄芩素)是一种存在于黄芩,木蝴蝶,百里香等植物中的天然黄酮类化合物,具有抗炎和抗癌活性。Baicalein可明显抑制PI3K/Akt/NF-κB途径,同时也可通过上调GPX4,抑制黑素细胞的铁死亡(ferroptosis),用于白癜风和肿瘤的相关研究。
M9325 EGTA EGTA是一种特殊的钙离子螯合剂,在生理 pH 值 (7.4) 下,Kd 为 60.5 nM,对 Ca2+ 比对 Mg2+ 有很高的特异性。EGTA 显著抑制炎性巨噬细胞的底物粘附能力。
M9330 Brij-35 Brij-35(月桂醇聚氧乙烯醚)是一种无毒的非离子表面活性剂,可降低非特定蛋白质的吸附,应用于红曲霉深层发酵时,能显著提高红曲色素产量。
M6154 2-PMPA tetrasodium 2-PMPA(PMPA tetrasodium salt)是高效选择性的谷氨酸羧肽酶II (GCPII)抑制剂,IC50值为300 pM。
M2250 Pamidronate disodium Pamidronate Disodium(帕米膦酸二钠)是一种含氮的双磷酸盐类化合物,具有抑制骨吸收的作用,可用于癌症相关的溶骨性病变等研究。
M9916 DPPH DPPH (2,2-Diphenyl-1-picrylhydrazyl,2,2-联苯基-1-苦基肼基) 是一种稳定的自由基,可用于测量抗氧化剂的自由基清除活性。
M9194 Insulin (human) Insulin (human) 是一种多肽激素,其调节血液中的糖(葡萄糖)水平并且由胰岛的β细胞产生。
M3409 Formestane Formestane(4-hydroxyandrostenedione,福美司坦)是第二代选择性芳香酶抑制剂,IC50为80 nM。
M9665 N-(2-amino-2-oxoethyl)acrylamide N-(2-Amino-2-oxoethyl)acrylamide(N-acryloyl-glycinamide,丙烯酰基甘氨酰胺)是一种单体,其聚合物能制备水凝胶,并用于酶的固定化。
M7791 Exo-1 Exo1是一种可逆的细胞外渗(exocytosis)抑制剂,也是高尔基ARF 1(ADP-Ribosylation Factor)GTP酶的激活剂。Exo1抑制细胞外渗,其IC50约为20μM。
M7817 GYKI 52466 hydrochloride Selective allosteric AMPA receptor antagonist; anti­convulsant; skeletal muscle relaxant.
M7815 GW2974 Potent and selective dual inhibitor of EGFR (IC50 = 0.
M7814 Guvacine hydrochloride GABA uptake inhibitor.
M7812 Formoterol fumarate dihydrate β2-Adrenoreceptor agonist.
M7809 FM19G11 FM19G11 is an inhibitor of Hypoxia Inducible Factors α (HIFα), reported to affect self-renewal and differentiation of stem cells.
M7808 FR-900098 monosodium salt 1-脱氧-d -木酮糖5-磷酸还原异构酶(DXR)是一种酶,在革兰氏阴性、革兰氏阳性细菌、植物和导致最致命疟疾的疟原虫——恶性疟原虫(哺乳动物产生)的非甲戊酸途径中,参与类异戊二烯生物合成的第一步。
M7807 Fusaric acid Dopamine β-hydroxylase inhibitor.
M7806 Fluorocurarine chloride Short-acting selective sympathetic ganglioblocker with weak antagonist activity on the nicotinic receptor at the neuromuscular junction; hypotensive.
M7803 FAUC 213 Highly selective D4 dopamine receptor full antagonist.
M7801 6-Fluoromevalonate Mevalonate-pyrophosphate decarboxylase inhibitor.
M7800 Fenvalerate Type II pyrethroid.
M7798 FPL 64176 Potent Ca2+ channel (L-type) activator.
M7797 FPL-55712 CysLT1 leukotriene receptor antagonist.
M7794 Encainide hydrochloride Encainide hydrochloride is a sodium channel blocker and class Ic antiarrhythmic.
M7789 Exo2 Exo2 acts as a chemical probe of intracellular transport.
M7788 Ethopropazine hydrochloride Ethoproprazine hydrochloride is an inhibitor of butyrylcholinesterase; antiparkinsonian.
M7787 Eupatorin Eupatorin acts as an antiproliferative in cells expressing the CYP1A- family.
M7786 17-Epiestriol 17-雌二醇是一种雌二醇代谢物,也是一种选择性雌激素受体(ER) -激动剂。
M7784 16-Epiestriol 16-Epiestriol is an estradiol metabolite that exhibits significant anti-inflammatory activity without glycogenic activity.
M7783 Efaroxan hydrochloride (+)-Isomer is a selective α-adrenoceptor antagonist; (−)-isomer is an imidazoline ligand that induces insulin secretion, mediated by the blockade of ATP-sensitive potassium channels in pancreatic β cells; I1 imidazoline binding site antagonist.








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