找到约 32 条 “Phosphatase” 相关结果 (用时 0.107 秒)

目录号 产品名称 中文名称 靶点
M7528 Phosphatase Inhibitor Cocktail (EDTA-Free) 磷酸酶抑制剂Cocktail(不含EDTA) Inhibitor Cocktails
AbMole磷酸酶抑制剂Cocktail 是由2 支(8 种) 独立的磷酸酶抑制剂(不含EDTA) 配置而成的磷酸酶抑制剂混合物。分为A、B 两管:A 管中是磷酸根类似物,以阻止研究中蛋白和脂类的磷酸化状态丢失;B 管则是新兴的天然产物,为蛋白磷酸化提供更加全面的保护。
M9403 TPI-1 TPI-1 Phosphatase
Tyrosine Phosphatase Inhibitor 1
TPI-1是一种SHP-1的抑制剂,它抑制重组SHP-1的IC50值为40 nM。
M9518 BN82002 BN82002 Phosphatase
CDC25 Phosphatase Inhibitor I
BN82002(别名CDC25 Phosphatase Inhibitor I)是一种CDC25磷酸酶家族的有效,选择性和不可逆抑制剂,对于25A,25B2,25B3,25C和25C-cat的IC50值分别为2.4,3.9,6.3,5.4和4.6 µM。
M11157 Alkaline phosphatase (E. coli) 碱性磷酸酶 (E. coli) Metabolite/Endogenous Metabolite
Alkaline phosphatase 是一种膜结合糖蛋白,在碱性 pH 值下催化磷酸单酯的水解。Alkaline phosphatase 可用于分子生物学和酶免分析。
M42551 Phosphatase-IN-1 Phosphatase-IN-1 Phosphatase
Phosphatase-IN-1 是一种 propranolol 衍生物,是一种磷脂酸磷酸酶 (Pah) 抑制剂。
M52602 Adenosine triphosphatase Adenosine triphosphatase Metabolite/Endogenous Metabolite
Adenosine triphosphatase 是一种催化 ATP 分解为 ADP 和游离磷酸根离子 (Pi) 的酶。
M2865 Sodium Monofluorophosphate 单氟磷酸钠 Pyruvate Kinase
Sodium Monofluorophosphate 是一种竞争性的丙酮酸激酶(PK)和碱性磷酸酶(ALP)抑制剂,Ki分别为3.4 mM和69 μM,也不可逆地抑制磷酸化酶磷酸酶(phosphorylase phosphatase),Ki为0.5 mM。
M2922 Pentamidine dihydrochloride 戊烷脒 Parasite
MP601205 dihydrochloride
Pentamidine HCl是一种 PRL Phosphatases 抑制剂,也可以抑制DNA, RNA和蛋白质的合成。
M2993 Sal003 Sal003 Phosphatase
Sal003 是一种有效的细胞渗透性 eIF-2α phosphatase 抑制剂。
M5767 Menadione (Vitamin K3) 维生素K3;甲萘醌 DNA/RNA Synthesis
Menadione(Vitamin K3,维生素K3,甲萘醌),一种脂溶性化合物,是Cdc25 phosphatase的抑制剂,也是mitochondrial DNA polymerase γ (pol γ)的抑制剂,常被用作营养添加剂。
M9081 Sodium Stibogluconate Sodium Stibogluconate Phosphatase
Stibogluconate sodium
Sodium Stibogluconate是一种有效的蛋白酪氨酸磷酸酶protein tyrosine phosphatase 抑制剂。
M9467 F1063-0967 F1063-0967 Phosphatase
F1063-0967 is a novel inhibitor of dual-specificity phosphatase 26 (DUSP26), inducing apoptosis in IMR-32 cell line.
M10278 Raphin1 Raphin1 Phosphatase
Raphin1 是一种选择性的,具有口服活性的 R15B (PPP1R15B, 一种蛋白磷酸酶1的调节亚基) 抑制剂,与 R15B-PP1c holophosphatase 结合的Kd值为33 nM。
M14486 BN82002 hydrochloride BN82002 hydrochloride Phosphatase
BN82002 hydrochloride 是 CDC25 phosphatase 家族的有效,选择性和不可逆的泛抑制剂。 BN82002 hydrochloride抑制 CDC25A,CDC25B2,CDC25B3,CDC25C CDC25A 和 25C-cat 的 IC50 值分别为 2.4、3.9、6.3、5.4 和 4.6 µM。 BN82002 hydrochloride 显示出比 CD45 酪氨酸磷酸酶高约 20 倍的选择性。
M14498 TCS 401 TCS 401 Phosphatase
TCS 401 是选择性的蛋白酪氨酸磷酸酶 1B (protein tyrosine phosphatase 1B) 抑制剂。
M20176 WAY-382818 WAY-382818 Others
WAY-382818 has mitogen-activated protein kinase phosphatase-1 inhibitory activity.
M20490 1-Naphthyl phosphate potassium salt 1-Naphthyl phosphate potassium salt Phosphatase
α-Naphthyl acid phosphate monopotassium salt
1-Naphthyl phosphate potassium salt is a non-specific phosphatase inhibitor which acts on acid, alkaline, and protein phosphatases.
M20719 Raphin1 acetate Raphin1 acetate Phosphatase
Raphin1 acetate is an orally bioavailable, selective inhibitor of the regulatory phosphatase PPP1R15B (R15B). Raphin1 acetate binds strongly to the R15B-PP1c holophosphatase with Kd of 0.033 μM.
M20734 (E/Z)-BCI (E/Z)-BCI Phosphatase
BCI, NSC 150117
(E/Z)-BCI (BCI, NSC 150117) is an inhibitor of dual specific phosphatase 1/6 (DUSP1/DUSP6) and mitogen-activated protein kinase with EC50 of 13.3 μM and 8.0 μM for DUSP6 and DUSP1 in cells, respectively. (E)-BCI induces apoptosis via generation of reactive oxygen species (ROS) and activation of intrinsic mitochondrial pathway in H1299 lung cancer cells.
M20794 Menadione bisulfite sodium Menadione bisulfite sodium Phosphatase
Menadione sodium bisulfite, Vitamin K3 sodium bisulfite
Menadione(Vitamin K3) bisulfite sodium, a fat-soluble compound, is an inhibitor of Cdc25 phosphatase and mitochondrial DNA polymerase γ (pol γ), used as a nutritional supplement.
M20854 L-Homoarginine hydrochloride L-Homoarginine hydrochloride Phosphatase
L-Homoarginine is a specific inhibitor of liver-type alkaline phosphatase.
M28961 TH1217 TH1217 Anti-infection
ZINC1775962367
TH1217 (ZINC1775962367) 是一种有效的、选择性的 dCTPase pyrophosphatase 1 (dCTPase) 抑制剂,IC50 值为 47 nM。TH1217 可增强胞苷类似物在白血病细胞中的细胞毒性作用。TH1217 还可以调节 SARS-Cov-2 相互作用体,因此它具有抗 COVID-19 的活性。
M29832 Managlinat dialanetil Managlinat dialanetil Others
MB06322; CS-917
Managlinat dialanetil (MB06322) 是一种可口服利用的 fructose 1,6-bisphosphatase (FBPase) 抑制剂,作用于 2 型糖尿病。
M43825 APS-5 APS-5 Fluorescent Dye
Lumigen APS-5
APS-5 是 alkaline phosphatase (ALP) 的底物,APS-5 可用于测定 ALP 的活性。
M50340 Organophosphorus acid anhydrolase Organophosphorus acid anhydrolase Enzymes & Coenzymes
Organophosphorus acid anhydrolase (Diisopropylfluorophosphatase) 是一种生化试剂,可作为生物材料或有机化合物,用于生命科学相关研究。
M52552 Microcystin-RR Microcystin-RR Phosphatase
Microcystin-RR (Cyanoviridin RR) 是一种有效的口服活性蛋白磷酸酶 (protein phosphatase) 抑制剂。
M52779 p-fin4 p-fin4 GluR
p-fin4 是 STEP Phosphatase-GluA2 AMPA 受体相互作用的肽抑制剂,Ki 为 0.4 μM。
M54738 Recombinant Human ICA 512/PTPRN Protein (293AA, E.coli, N-6His) 重组人ICA 512/PTPRN 蛋白 (293AA, E.coli, N-6His) Cytokines and Growth Factors
IA2; R-PTP-N; Islet cell antigen 512
ICA 512/PTPRN Protein belongs to the protein-tyrosine phosphatase family and receptor class 8 subfamily. ICA 512/PTPRN implicated in neuroendocrine secretory processes. It may be involved in processes specific for neurosecretory granules, such as their biogenesis, trafficking or regulated exocytosis or may have a general role in neuroendocrine functions.
M54739 Recombinant Human ICA 512/PTPRN Protein (80AA&94AA, E.coli, N-6His) 重组人ICA 512/PTPRN 蛋白 (80AA&94AA, E.coli, N-6His) Cytokines and Growth Factors
IA2; R-PTP-N; Islet cell antigen 512
ICA 512/PTPRN Protein belongs to the protein-tyrosine phosphatase family and receptor class 8 subfamily. ICA 512/PTPRN implicated in neuroendocrine secretory processes. It may be involved in processes specific for neurosecretory granules, such as their biogenesis, trafficking or regulated exocytosis or may have a general role in neuroendocrine functions.
M55360 4-Methylumbelliferyl phosphate 4-甲基伞形酮磷酸酯 Phosphatase
4-MUP
4-Methylumbelliferyl phosphate (4-MUP) 是一种阴离子有机磷酸酯,是一种酸性和碱性磷酸酶 (phosphatase) 的荧光底物。
M55404 Recombinant Mouse Pleiotrophin/PTN (HEK293, C-6His) 重组小鼠Pleiotrophin/PTN (HEK293, C-6His) Cytokines and Growth Factors
HBBM; HBGF-8; OSF-1
Pleiotrophin (PTN) is a secreted, strongly heparinbinding, developmentally regulated cytokine. PTN is involved in development of brain, bone, and organs undergoing branching morphogenesis. PTN causes PTPRB dimerization and inactivates its phosphatase activity, which allows increased tyrosine phosphorylation of its substrates. Increased expression of PTN is correlated with neuronal development or stresses such as brain ischemia and Parkinson’s disease.
M56678 DL-AP3  DL-AP3  Metabolite/Endogenous Metabolite
DL-AP3 是一种竞争性的 mGluR1 和 mGluR5 拮抗剂。DL-AP3 也是磷酸丝氨酸磷酸酶 (phosphoserine phosphatase) 的抑制剂。








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