找到约 38 条 “Antibiotic” 相关结果 （用时 0.087 秒）
| 目录号 | 产品名称 | 中文名称 | 靶点 |
|---|---|---|---|
M2790
|
K252a | K252a | PKC |
| SF 2370; Antibiotic K-252a | |||
| K252a 是BDNF 受体 TrkB 的抑制剂。K-252a 对 PKC、PKA、II型钙调素依赖性激酶和磷酸化酶激酶的 IC50 值分别为470 nM、140 nM、270 nM和1.7 nM。K-252a 抑制 NGF 受体 gp140trk 的酪氨酸蛋白激酶 (TRK) 活性，IC50 为 3 nM。 | |||
M6292
|
Ansamitocin P 3 | 安丝菌素P-3 | Microtubule |
| Antibiotic C 15003P3; Maytansinol butyrate | |||
| Ansamitocin P-3是一种微管抑制剂，也是一种大环抗肿瘤抗生素。 | |||
| M9780
|
Nigericin | Nigericin | Potassium Channel |
| Antibiotic K178, Antibiotic X464 | |||
| Nigericin is an antibiotic derived from Streptomyces hygroscopicus, it acts as an H+, K+, Pb2+ ionophore. | |||
| M9860
|
Bleomycin A5 Hydrochloride | 盐酸平阳霉素 (不含铜离子) | DNA/RNA Synthesis |
| BLEOCIN Antibiotic; Bleomycin A5 HCl | |||
| 博莱霉素A5盐酸盐是博莱霉素家族的一种独特的抗生素，对真核和原核细胞有毒。 | |||
| M11236
|
Lasalocid sodium | 拉沙洛西钠；拉沙里菌素钠；那塞罗钠 | Antibiotic |
| Lasalocid-A sodium; Ionophore X-537A sodium; Antibiotic X-537A | |||
| Lasalocid sodium (Lasalocid-A sodium) 是一个抗菌剂。 | |||
| M13469 | Lasalocid | Lasalocid | Antibiotic |
| Lasalocid-A; Ionophore X-537A; Antibiotic X-537A | |||
| Lasalocid (Lasalocid-A; Ionophore X-537A; Antibiotic X-537A) 是一种抗菌剂和抗球虫药, 用在饲料添加剂中。 | |||
| M21494
|
Sibofimloc | Sibofimloc | Antibiotic |
| Antibiotic-202 | |||
| Sibofimloc (Antibiotic-202) 是一类首创的(first-in-class)，肠道限制性的，具有口服活性的 FimH 粘附 (FimH adhesion ) 抑制剂。Sibofimloc 具有抗细菌感染活性，被开发用于炎症性肠病 (IBD) 的研究。 | |||
| M30025 | Malonomicin | Malonomicin | Antibiotic |
| Antibiotic K16 | |||
| Malonomicin (Antibiotic K16) 是一种具有抗原生动物和抗锥虫活性的抗生素。Malonomicin 在体内也显示出抗锥虫活性。 | |||
| M30504 | Pentachloropseudilin | Pentachloropseudilin | Myosin |
| Antibiotic A 15104 Y; PClP | |||
| Pentachloropseudilin (Antibiotic A 15104 Y; PClP) 是一种可逆的、变构有效的肌球蛋白 (Myo1s) 抑制剂，对 Myo1s 的 IC50 范围为 1 至 5 μM，对于 2 类和 5 类肌球蛋白，IC50 范围 > 90 μM。Pentachloropseudilin 是转化生长因子-β (TGF-β) 刺激的信号传导的有效抑制剂，对 TGF-β 的 IC50 值为 0.1-0.2 μM。 | |||
| M30588 | Leucinostatin A | Leucinostatin A | Antifungal |
| Antibiotic P168 | |||
| Leucinostatin A (Antibiotic P168) 是一种九肽，对白色念珠菌和新型隐球菌具有显着的活性。Leucinostatin A 是一种疏水性九肽抗生素。Leucinostatin A 通过减少前列腺基质细胞中胰岛素样生长因子-I 的表达来抑制前列腺癌的生长。具有抗原虫活性。 | |||
| M2637
|
Difloxacin hydrochloride | 盐酸双氟沙星 | Antibiotic |
| Difloxacin is a synthetic antibiotic that belongs to the fluoroquinolone class. | |||
| M2833
|
Meclocycline Sulfosalicylate | 磺基水杨酸甲氯环素；甲氯环素磺基水杨酸盐 | Antibiotic |
| Meclocycline is a tetracycline antibiotic. Meclocycline sulfosalicylate prevents bacterial protein synthesis through 30S ribosome-mediated chain elongation and blocks amino-acyl tRNA A-site binding. | |||
| M2950
|
Piromidic Acid | 吡咯酸；吡咯米酸 | Antibiotic |
| Piromidic acid is a quinolone antibiotic. | |||
| M3644
|
Demeclocycline hydrochloride | 盐酸地美环素 | Antibiotic |
| Demeclocycline HCl | |||
| Demeclocycline HCl 是一种四环素antibiotic可抑制细菌的蛋白合成，能用于细菌感染的相关研究。 | |||
| M4904
|
Clindamycin Phosphate | 克林霉素磷酸酯 | Antibiotic |
| NSC 618653 | |||
| Clindamycin Phosphate is a lincosamide antibiotic for Plasmodium falciparum with IC50 of 12 nM. | |||
| M4906
|
Doripenem Hydrate | 多尼培南 | Antibiotic |
| S-4661 | |||
| Doripenem Hydrate is an ultra-broad-spectrum injectable antibiotic, used to treat complicated intra-abdominal infections and complicated urinary tract infections. | |||
| M4941
|
Lomefloxacin | 洛美沙星 | Antibiotic |
| Maxaquin,SC47111A | |||
| Lomefloxacin (SC47111A) 是一种广谱喹诺酮类 (antibiotic)抗生素，具有抗菌活性。 | |||
| M4947
|
Streptomycin sulfate | 硫酸链霉素 | Antibiotic |
| Streptomycin sulfate（硫酸链霉素）是一种氨基糖苷类抗生素（antibiotic），它通过抑制蛋白质合成中的起始和延伸过程来发挥作用。 | |||
| M7125 | PF 945863 | PF 945863 | Others |
| PF 945863 is a macrolide antibiotic. | |||
| M7340 | Sulopenem | 硫培南 | Others |
| Sulopenem is a penem antibiotic. | |||
| M7436 | Trovafloxacin mesylate | 曲伐沙星甲磺酸；曲伐沙星甲磺酸盐 | Others |
| Trovafloxacin mesylate is a antibiotic; inhibits bacterial DNA synthesis. | |||
| M7720 | Caerulomycin A | 浅蓝霉素 | Others |
| Caerulomycins produced by Streptomyces caeruleus are bipyridinic molecules endowed with antibiotic properties. | |||
| M7721 | Chrysomycin B | 金黄霉素B | Others |
| Antibiotic from Streptomyces sp. | |||
| M7756 | Dihydroeponemycin | Dihydroeponemycin | Others |
| Dihydroeponemycin is an active derivative of eponemycin an antitumor antibiotic isolated from Streptomyces hygroscopicus. | |||
| M7893 | Leptomycin A | 来普霉素A | Others |
| Leptomycins are antifungal antibiotics with unique unsaturated, branched-chain fatty acid structures. | |||
| M8006 | PD 404,182 | PD 404,182 | Others |
| Potential antibiotic of gram negative bacteria. | |||
| M8276
|
Pleuromutilin | 泰妙菌素 | Antibiotic |
| Drosophilin B; Mutilin 14-glycolate | |||
| Pleuromutilin is an antibiotic natural product that inhibits bacterial protein synthesis by binding to bacterial ribosomes in the peptidyl transferase center and inhibiting peptide bond formation. | |||
| M8378 | DCAP | DCAP | Others |
| DCAP is a potent broad-spectrum antibiotic that specifically targets the membranes of both Gram-positive and Gram-negative bacteria. | |||
| M8412 | Pivmecillinam | 匹美西林；氮卓脒青霉素双酯；吡呋氮卓脒青霉素 | Others |
| Amdinocillin pivoxil | |||
| Pivmecillinam is a gram negative antibiotic, and inhibitor of penicillin-binding protein 2 (PBP2). | |||
| M8417 | Geldanamycin-Biotin | Geldanamycin-Biotin | Others |
| Geldanamycin-Biotin is a benzoquinone ansamycin antitumor antibiotic. | |||
| M8578 | Undecylprodigiosin hydrochloride | Undecylprodigiosin hydrochloride | Others |
| Undecylprodigiosin is a tri-pyrolle antibiotic isolated from Streptomyces coelicolor A3 that exhibits immunosuppressive and apoptotic activities as well as antibacterial, antioxidative and UV protective properties. | |||
| M8711 | Delafloxacin | 德拉沙星API | Others |
| Delafloxacinum; RX-3341; WQ-3034; ABT492; ABT 492; ABT-492 | |||
| Delafloxacin is a fluoroquinolone antibiotic active against both Gram-negative and Gram-positive bacteria such as MRSA. | |||
| M8803 | Thiolutin | 硫藤黄素；硫藤黄菌素 | Others |
| Sulfur-containing antibiotic, which is a potent inhibitor of bacterial and yeast RNA polymerases. | |||
| M19137
|
Amoxicillin | 阿莫西林 | Antibiotic |
| Amoxicillin (Amoxycillin) 是一种具有良好口服吸收和广谱抗菌活性的抗生素 (antibiotic)。Amoxicillin 抑制细胞壁中多肽的生物合成，从而抑制细胞生长。 | |||
| M19865
|
Sulfacetamide sodium salt hydrate | Sulfacetamide sodium salt hydrate | Autophagy |
| Sulfacetamide is a sulfonamide antibiotic that blocks the synthesis of dihydrofolic acid by inhibiting the enzyme dihydropteroate synthase(DHPS) with IC50 of 9.5 μM. Sulfacetamide is a competitive inhibitor of bacterial para-aminobenzoic acid (PABA), which is required for bacterial synthesis of folic acid. | |||
| M19867
|
Gatifloxacin hydrochloride | Gatifloxacin hydrochloride | Topoisomerase |
| AM-1155 hydrochloride; CG5501 hydrochloride; BMS-206584 hydrochloride; PD135432 hydrochloride | |||
| Gatifloxacin (AM-1155, CG5501, BMS-206584, PD135432) hydrochloride is a potent fluoroquinolone antibiotic with broad-spectrum antibacterial activity. Gatifloxacin hydrochloride inhibits bacterial type II topoisomerases with IC50 of 13.8 μg/ml and 0.109 μg/ml for S. aureus topoisomerase IV and E. coli DNA gyrase, respectively. | |||
| M19869
|
Lefamulin acetate (Xenleta) | Lefamulin acetate (Xenleta) | Antibiotic |
| BC-3781 acetate | |||
| Lefamulin acetate (Xenleta, BC-3781 acetate) is a pleuromutilin antibiotic for community-acquired bacterial pneumonia (CABP) treatment. Lefamulin acetate inhibits protein synthesis by binding to the peptidyl transferase center of the 50S bacterial ribosome, thus preventing the binding of transfer RNA for peptide transfer. | |||
| M19870
|
Delafloxacin Meglumine | Delafloxacin Meglumine | Antibiotic |
| ABT-492; RX-3341; WQ-3034; Baxdela | |||
| Delafloxacin (ABT-492, RX-3341, WQ-3034, Baxdela) meglumine is a broad-spectrum fluoroquinolone antibiotic against multiple pathogens. | |||
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