找到约 58 条 “Peptide R” 相关结果 （用时 0.065 秒）
| 目录号 | 产品名称 | 中文名称 | 靶点 |
|---|---|---|---|
M2007
|
Romidepsin (FK228) | 罗米地辛；罗米地新 | HDAC |
| FK228; ISTODAX; Depsipeptide; FR 901228; NSC 630176 | |||
| Romidepsin (FK228, Depsipeptide, FR 901228, NSC 630176) 是一种大环缩肽化合物，也是一种组蛋白去乙酰化酶 (HDAC) 抑制剂，可抑制HDAC1，HDAC2，HDAC4 和 HDAC6，IC50 值分别为 36 nM，47 nM，510 nM 和 1.4 μM。Romidepsin可诱导肿瘤细胞周期的停滞和凋亡。 | |||
| M1261
|
NFAT Inhibitor-1 (VIVIT peptide) | NFAT Inhibitor-1 (VIVIT peptide) | NFAT |
| VIVIT peptide; NFAT Inhibitor; ABM-7733 | |||
| NFAT Inhibitor-1 (VIVIT peptide) 是一种 NFAT 的细胞渗透性肽抑制剂，在抑制细胞提取物中钙调神经磷酸酶介导的NFAT1、NFAT2和NFAT4去磷酸化方面表现优异。 | |||
M9771
|
TRAP-6 | TRAP-6 | Peptides |
| Thrombin Receptor Activator Peptide 6; PAR-1 agonist peptide | |||
| TRAP-6 (Thrombin Receptor Activator Peptide 6) 是一种凝血酶受体激活肽，也是选择性的蛋白酶激活受体 1 (PAR1) 激动剂，TRAP-6 可以通过 PAR 1受体激活血小板并刺激血小板聚集。 | |||
| M10236
|
PAR-2 (1-6) (mouse, rat) | H-丝氨酰亮氨酰异亮氨酰甘氨酰精氨酰亮氨酰-OH | PAR |
| PAR-2 AGONIST PEPTIDE (SLIGRL), MOUSE | |||
| PAR-2 (1-6) (mouse, rat) 是一种 PAR2 的激活剂，它可以用于探索细胞中 PAR2 的信号传导。 | |||
| M10557
|
RGD peptide (GRGDNP) (TFA) | RGD peptide (GRGDNP) (TFA) | Integrin |
| GRGDNP TFA | |||
| RGD peptide TFA 是一种整合素（integrin）-配体相互作用的抑制剂，在细胞黏附、迁移、生长和分化中发挥重要作用。 | |||
| M11207
|
GLP-1(7-37) | 人胰高血糖素样肽-1 | GLP Receptor |
| Insulinotropin (human);Peptide GLP-1 (human glucose-lowering peptide-1) | |||
| GLP-1(7-37) 是一种肠道胰岛素激素，可以增强葡萄糖诱导的胰岛素分泌。 | |||
| M13495
|
Aviptadil | 阿肽地尔 | Others |
| Vasoactive Intestinal Peptide (human, rat, mouse, rabbit, canine, porcine) | |||
| Aviptadil 是一种血管活性肠多肽 (VIP) 类似物，具有强的血管舒张 (vasodilatory) 作用。Aviptadil 诱导肺血管扩张，抑制血管 SMCs 增殖、血小板聚集。Aviptadil 可用于肺纤维化、肺动脉高压 (PAH)、SARS-CoV-2 引起呼吸衰竭等的研究。 | |||
| M13496
|
Aviptadil acetate | 醋酸阿肽地尔 | Others |
| Vasoactive Intestinal Peptide acetate salt (human, rat, mouse, rabbit, canine, porcine) | |||
| Aviptadil acetate 是一种模拟血管活性肠多肽 (VIP) 类似物，具有强的血管舒张 (vasodilatory) 效应。。Aviptadil acetate 诱导肺血管扩张，抑制血管 SMCs 增殖、血小板聚集。Aviptadil acetate 可用于肺纤维化、肺动脉高压 (PAH)、SARS-CoV-2 引起呼吸衰竭等的研究。 | |||
| M13751
|
Arg-Gly-Asp-Ser | Arg-Gly-Asp-Ser | Integrin |
| RGDS peptide; Fibronectin tetrapeptide | |||
| Arg-Gly-Asp-Ser 是整联蛋白结合序列，抑制整联蛋白受体 (integrin receptor) 功能。Arg-Gly-Asp-Ser 直接并特异性地结合 pro-caspase-8，pro-caspase-9 和 pro-caspase-3，但不与 pro-caspase-1 结合。 | |||
| M13931
|
Calcitonin Gene Related Peptide (CGRP) (83-119), rat TFA | Calcitonin Gene Related Peptide (CGRP) (83-119), rat TFA | CGRP Receptor |
| Calcitonin Gene Related Peptide (CGRP) (83-119), rat (TFA) 是一种由 37 个氨基酸组成的降钙素家族神经肽，通过 (CRLR) 起作用。 | |||
| M13957
|
Carperitide acetate | Carperitide acetate | Endothelin Receptor |
| Atrial Natriuretic Peptide (ANP) (1-28), human, porcine acetate | |||
| Carperitide acetate (Atrial Natriuretic Peptide (ANP) (1-28), human, porcine acetate) 是一种含 28 个氨基酸的激素，由心脏产生并分泌，以响应心脏损伤和机械拉伸。Carperitide acetate 抑制内皮素-1 (endothelin-1) 分泌。 | |||
| M14026 | Peptide YY (PYY) (3-36), porcine TFA | Peptide YY (PYY) (3-36), porcine TFA | Others |
| Peptide YY (PYY) (3-36), porcine TFA 是一种肠胃激素肽，作为 Y2 受体的激动剂，能够降低食欲。 | |||
| M14808 | (Arg)9 TFA | (Arg)9 TFA | Peptides |
| Nona-L-arginine TFA; Peptide R9 TFA | |||
| (Arg)9 TFA (Nona-L-arginine TFA)是可渗透细胞的多肽，在谷氨酸模型实验模型中保护神经的IC50值为0.78 μM。 | |||
| M14818
|
Myelin Oligodendrocyte Glycoprotein Peptide (35-55), mouse, rat TFA | Myelin Oligodendrocyte Glycoprotein Peptide (35-55), mouse, rat TFA | Peptides |
| MOG (35-55) (TFA) | |||
| Myelin Oligodendrocyte Glycoprotein Peptide (35-55), mouse, rat (TFA) 是中枢神经鞘的一个次要成分。Myelin Oligodendrocyte Glycoprotein Peptide (35-55), mouse, rat (TFA)引发复发缓解性神经系统疾病，伴有广泛的斑块样脱髓鞘。还能诱导强效的 T细胞和 B 细胞反应，同时是高度脑源性的。 | |||
| M20872
|
RGD peptide (GRGDNP) | RGD peptide (GRGDNP) | Integrin |
| RGD peptide (GRGDNP) is an inhibitor of binding of integrins to the extracellular matrixs. RGD peptide (GRGDNP) induces apoptosis presumably through direct activation of caspase-3. | |||
| M21347
|
Recombinant Human NPPB (E.coli, N-6His) | 重组人NPPB蛋白 (E.coli, N-6His) | Cytokines and Growth Factors |
| Natriuretic Peptides B; Gamma-Brain Natriuretic Peptide | |||
| 重组人钠尿酸肽B是由大肠杆菌表达系统生产的，编码His27-His134的目标基因在N端有一个6His标签。蛋白编号：P16860。 | |||
| M21348
|
Recombinant Human NT-proBNP ( E.coli, N-6His-Flag) | 重组人NT-proBNP蛋白 ( E.coli, N-6His-Flag) | Cytokines and Growth Factors |
| Natriuretic peptides B; Gamma-brain natriuretic peptide | |||
| 重组人脑型钠尿酸肽由大肠杆菌表达系统生产，编码His27-Arg102的目标基因在N端有一个6His、Flag标签。蛋白编号：P16860。 | |||
| M28094 | Peptide YY (PYY) (3-36), porcine | Peptide YY (PYY) (3-36), porcine | Neuropeptide Receptor |
| Peptide YY (PYY) (3-36), porcine 是一种肠胃激素肽，作为 Y2 受体的激动剂，能够降低食欲。 | |||
| M31218
|
Neuropeptide Y (3-36) (human, rat) | Neuropeptide Y (3-36) (human, rat) | Neuropeptide Receptor |
| Neuropeptide Y (3-36) (human, rat) 是由二肽基肽酶4 (DPP4) 形成的神经肽Y (NPY) 代谢产物，是一种选择性 Y2 受体激动剂。Neuropeptide Y (3-36) (human, rat) 是由二肽基肽酶 4 (DPP4) 形成的 NPY 代谢产物。Neuropeptide Y (3-36) (human, rat) 通过 Y2 受体减少去甲肾上腺素的释放。 | |||
| M41862 | Dipeptide diaminobutyroyl benzylamide diacetate | Dipeptide diaminobutyroyl benzylamide diacetate | AChR/AChE |
| Dipeptide diaminobutyroyl benzylamide diacetate 是一种 Wagerlin-1 模拟肽，是一种 mAChR 拮抗剂。 | |||
| M43248 | IRAK-4 Peptide substrate | IRAK-4 Peptide substrate | Others |
| IRAK-4 Peptide substrate (IRAK-1 (360-380)) 是一种有生物活性的肽。 | |||
| M43256 | Myristoyl tetrapeptide Ala-Ala-Pro-Val | Myristoyl tetrapeptide Ala-Ala-Pro-Val | Others |
| Myristoyl tetrapeptide Ala-Ala-Pro-Val 是一种有生物活性的肽。 | |||
| M43267 | CCK1-specific peptide substrate | CCK1-specific peptide substrate | Others |
| CCK1-specific peptide substrate 是一种有生物活性的肽。 | |||
| M49714 | MEK1 Derived Peptide Inhibitor 1 | MEK1 Derived Peptide Inhibitor 1 | ERK |
| MEK1 Derived Peptide Inhibitor 1 是一种肽抑制剂。 | |||
| M49718 | Myristoyl-MEK1 Derived Peptide Inhibitor 1 | Myristoyl-MEK1 Derived Peptide Inhibitor 1 | ERK |
| Myristoyl-MEK1 Derived Peptide Inhibitor 1 是 MEK1 Derived Peptide Inhibitor 1 的豆蔻酰化形式。 | |||
| M49754 | C-Peptide 1 (rat) | C-Peptide 1 (rat) | GSK-3 |
| C-Peptide 1 (rat) 是一种肽，是 β-catenin/GSK-3β 激活剂。 | |||
| M50405 | Syk Kinase Peptide Substrate | Syk Kinase Peptide Substrate | Syk |
| Syk Kinase Peptide Substrate 是Syk 激酶多肽底物。 | |||
| M50418 | Gastric Inhibitory Polypeptide (1-30), porcine | Gastric Inhibitory Polypeptide (1-30), porcine | Insulin Receptor |
| Gastric Inhibitory Polypeptide (1-30), porcine 缺乏天然胃抑制多肽 (GIP) C端 12 个氨基酸残基，能够增强胰岛素和生长抑素的释放而发挥生物活性。 | |||
| M50431 | Phospho-Glycogen Synthase Peptide-2(substrate) | Phospho-Glycogen Synthase Peptide-2(substrate) | GSK-3 |
| Phospho-Glycogen Synthase Peptide-2 (substrate) 是糖原合酶激酶-3 (GSK-3) 的肽底物，可用于蛋白丝氨酸激酶的亲和纯化。 | |||
| M51065 | MLCK Peptide, control | MLCK Peptide, control | Others |
| MLCK Peptide, control是一种肌球蛋白轻链激酶。 | |||
| M2976
|
RGD | RGD | Integrin |
| Arg-Gly-Asp | |||
| RGD (Arg-Gly-Asp) Peptides是一种细胞粘附序列，可以模仿细胞粘附蛋白并与整合素（integrin）结合。 | |||
| M40855
|
Recombinant Human Siglec-7 Protein (HEK293, C-6His) | 重组人Siglec-7蛋白 (HEK293, C-6His) | Receptor Proteins |
| sialic acid binding Ig-like lectin 7; CD328 antigen; p75/AIRM1; QA79 | |||
| Human Siglec-7 encodes a 467 amino acid (aa) polypeptide with a hydrophobic signal peptide, an N-terminal Ig-like V-type domain, two Ig-like C2-type domains, a transmembrane region and a cytoplasmic tail. It binds equally well to both alpha 2,3- and alpha 2,6-linked sialic acid. | |||
| M11232
|
Recombinant Mouse Beta-NGF Protein (110AA, E. coli) | 重组小鼠β-NGF蛋白 (110AA, E. coli) | Cytokines and Growth Factors |
| β-NGF; NGFB | |||
| Mouse beta -NGF is a homodimer of two 120 amino acid polypeptides. β-NGF acts as a growth and differentiation factor for B lymphocytes, and enhances B-cell survival. | |||
| M6875
|
L-152,804 | L-152,804 | Neuropeptide Receptor |
| L-152804 | |||
| L-152,804（L-152804）是一种具有口服活性和脑渗透性的，有效的、选择性的非肽类Neuropeptide Y Receptor（NPYR）拮抗剂，Ki值为 26 nM，比作用于hY1、hY2和hY4受体的选择性高300倍。此外，L-152804还能通过调节食物摄入和能量消耗，减轻饮食诱导的肥胖小鼠的体重，可用于摄食，体重调节以及血糖的相关研究。 | |||
| M6911 | LM11A 31 dihydrochloride | LM11A 31 dihydrochloride | Others |
| LM11A 31 dihydrochloride is a nonpeptide p75 NTR ligand; neuroprotective. | |||
| M7008
|
Muramyl Dipeptide | 佐剂肽 | p38 MAPK |
| MDP | |||
| Muramyl dipeptide（MDP）是一种合成的免疫反应肽，它是细菌细胞壁肽聚糖的共有结构单元，广泛存在于革兰氏阳性菌和革兰氏阴性菌中。MDP具有较强的免疫调节作用，MDP作为NOD2受体的激动剂可以激活NF-κB并促进炎症因子的释放，MDP还可激活NLRP3，进一步增强免疫反应，它还常作为一种免疫佐剂使用，可增强疫苗或抗原的免疫效果。此外，MDP还能诱导成骨细胞的分化并抑制破骨细胞的分化。 | |||
| M7257 | SB 222200 | SB 222200 | Others |
| SB 222200 is a potent, selective non-peptide NK 3 antagonist. Brain penetrant. | |||
| M7283 | SDM25N hydrochloride | SDM25N hydrochloride | Others |
| SDM25N hydrochloride is a potent, selective non-peptide δ antagonist; also inhibits dengue virus replication. | |||
| M7586 | AC-7954 | AC-7954 | Others |
| Nonpeptide GPR14 / urotensin-UII (UII) receptor agonist that has an EC50 of 300 nM at the human UII receptor (h-UTR). | |||
| M7629
|
BIBP3226 TFA | BIBP3226 TFA | Neuropeptide Receptor |
| BIBP3226 TFA是第一个选择性的，有效的 Neuropeptide Y (神经肽Y) Y1 (NPY Y1) 受体拮抗剂，对 rNPY Y1，hNPFF2，rNPFF的Ki分别为1.1、79、108 nM。可用于心血管的相关研究。 | |||
| M7735
|
CP-96345 | CP-96345 | Neurokinin Receptor |
| CP96345 | |||
| CP-96345 is a highly potent and selective, orally active tachykinin and substance P receptor non-peptide inhibitor. | |||
| M7888 | Levocabastine hydrochloride | 左旋多巴 | Others |
| Non-peptide histamine H1 receptor antagonist; neurotensin NTS2 receptor ligand. | |||
| M7896 | LWH-63 hydrochloride | LWH-63 hydrochloride | Others |
| Non-peptide CRF1 corticotrophin-releasing factor antagonist. | |||
| M7912 | Mastoparan-7 | Mastoparan-7 | Others |
| Mastoparan 7 | |||
| G protein activator via Gαi and Gαo stimulation, similar to G protein-coupled receptors; peptide originally isolated from wasp venom. | |||
| M7947 | NSCI | NSCI | Others |
| NSCI is a nonpeptide caspase 3 selective inhibitor. | |||
| M7974 | Netropsin dihydrochloride | 水合纺锤菌素氟安定 | Others |
| Netropsin is an unusual n-methylpyrrole-containin |
|||
| M8150 | SB-668875 | SB-668875 | Others |
| SB-668875 is a novel, selective peptide agonist at OX2 orexin receptors. | |||
| M8205 | SR 142948A | SR 142948A | Others |
| SR 142948A is a non-peptide Neurotensin receptor antagonist. | |||
| M8210 | FR-171113 | FR-171113 | Others |
| FR171113 was the first non-peptide antagonist of the Protease Activated Receptor-1 (PAR1), also termed thrombin receptor. | |||
| M8276
|
Pleuromutilin | 泰妙菌素 | Antibiotic |
| Drosophilin B; Mutilin 14-glycolate | |||
| Pleuromutilin is an antibiotic natural product that inhibits bacterial protein synthesis by binding to bacterial ribosomes in the peptidyl transferase center and inhibiting peptide bond formation. | |||
| M8402 | LM11A-31 dihydrochloride | LM11A-31 dihydrochloride | Others |
| LM11A-31 is a non-peptide ligand of the p75 neurotrophin receptor (p75NTR). | |||
| M8432 | CYM50769 | CYM50769 | Neuropeptide Receptor |
| CYM50769 is a potent, specific antagonist of the Neuropeptide B and Neuropeptide W receptor, NPBWR1 (IC50 = 120 nM). | |||
| M8491 | Nap-FF | Nap-FF | Others |
| Nap-FF (2-Naa-FF) is a cell penetrant dipeptide that self-assembly and adopt the β-sheet structures to form prion-like nanofibrils of small molecules (PriSM). | |||
| M8539 | G3335 | G3335 | Others |
| G3335 ( L-tryptophyl-L-glutamic acid) is a cell-permeable dipeptide that acts as a selective and reversible PPARγ antagonist with a Kd value of 8. | |||
| M8814 | Trap-101 hydrochloride | Trap-101 hydrochloride | Others |
| Trap-101 Hydrochloride is a nociceptin/orphanin FQ peptide (NOP) receptor blocker. | |||
| M8853 | WIN 62,577 | WIN 62,577 | Others |
| Non-peptide NK1 tachykinin receptor antagonist. | |||
| M9190
|
Lixisenatide | 利西拉肽；利司那肽 | GLP Receptor |
| Lyxumia; Adlyxin; ZP10A peptide | |||
| Lixisenatide（Lyxumia, Adlyxin, ZP10A peptide）是一种glucagon-like peptide-1 (GLP-1) receptor激动剂(GLP-1RA)，其对人源GLP-1受体的IC50值为1.4 nM。 | |||
| M9656
|
FLAG peptide | FLAG peptide | Peptides |
| DYKDDDDK Peptide | |||
| FLAG peptide是一个多肽（Asp-Ty-rLys-Asp-Asp-Asp-Asp-Lys）由八个氨基酸组成，具有肠激酶切割位点，可用于抗体介导的重组蛋白识别和纯化。 | |||
