找到约 44 条 “Glycine” 相关结果 (用时 0.067 秒)
目录号 | 产品名称 | 中文名称 | 靶点 |
---|---|---|---|
M2558 | DMOG | 二甲基草酰甘氨酸 | HIF |
Dimethyloxalylglycine | |||
DMOG(Dimethyloxalylglycine,二甲基草酰甘氨酸)是一种α-酮戊二酸类似物,同时也是α-酮戊二酸辅助因子的拮抗剂。此外,DMOG还是竞争性的,细胞可渗透的缺氧诱导因子脯氨酰羟化酶 (HIF-PH)抑制剂,以及缺氧诱导因子-1α(HIF-1α)的激活剂,具有神经保护活性。 | |||
M1500 | Sarcosine | 肌氨酸 | Others |
N-Methylglycine | |||
Sarcosine(肌氨酸)是甘氨酸合成和降解过程中的中间体和副产物。 | |||
M7987 | N-Oleoylglycine | N-Oleoylglycine | Metabolite/Endogenous Metabolite |
Enzymatically produced in mammals. | |||
M9408 | Glycochenodeoxycholic acid | 甘氨鹅脱氧胆酸 | Metabolite/Endogenous Metabolite |
Chenodeoxycholylglycine | |||
Glycochenodeoxycholic acid(GCDC,甘氨鹅脱氧胆酸)是在肝内形成的胆汁盐,是胆汁酸(BA)的一种成分,可诱导原代人类肝细胞坏死,并可通过STAT3途径,促进肝细胞癌(HCC)的化疗耐药性。 | |||
M9409 | Glycoursodeoxycholic acid | 甘氨熊脱氧胆酸 | Metabolite/Endogenous Metabolite |
Ursodeoxycholylglycine | |||
Glycoursodeoxycholic acid是一种酰基甘氨酸和胆汁酸-甘氨酸缀合物。它是一种通过肠道微生物菌丛而产生的次级胆汁酸。 | |||
M9517 | Sodium hippurate | 马尿酸钠 | Others |
N-Benzoylglycine Sodium Salt | |||
Hippuric acid is a low molecular weight phenolic carboxylic acid urinary metabolite that may be a useful urinary biomarker for certain cancers such as gastric cancer and oxidative stress. | |||
M9566 | Glycine | 甘氨酸 | GluR |
Glycine甘氨酸是一种重要的抑制性神经神经递质(Inhibitory neurotransmitter)和NMDA受体的变构调节剂。 | |||
M10251 | Gly-β-MCA | Gly-β-MCA | Farnesoid X Receptor |
Glycine-β-muricholic Acid | |||
Gly-β-MCA 是一种有效的,稳定的,肠特异性的,具有口服生物活性的法尼酯X受体 (FXR) 抑制剂。 | |||
M10389 | Aminoethoxyvinyl glycine hydrochloride | Aminoethoxyvinyl glycine hydrochloride | Others |
AVG-HCl | |||
Aminoethoxyvinyl glycine hydrochloride (AVG-HCl) 是乙烯生物合成的抑制剂,1 µM 时可阻断 ACS 和 ACO 的活性。 | |||
M11510 | DL-Propargylglycine | DL-炔丙基甘氨酸 | Others |
PAG | |||
DL-Propargylglycine(DL-丙炔甘氨酸(PAG))是胱硫醚γ-裂解酶(GCL)的不可逆抑制剂,该酶是一种参与谷胱甘肽合成 ,调节同型半胱氨酸浓度,并介导半胱氨酸合成的代谢转硫途径的关键酶。 | |||
M12591 | ChemBridge-6146494 | ChemBridge化合物-6146494 | Screening Compounds and Building Blocks |
N-[3-(3-bromophenyl)-2-(2-furoylamino)acryloyl]glycine (6146494) | |||
ChemBridge特有类药化合物/先导化合物-6146494,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M12674 | ChemBridge-6432139 | ChemBridge化合物-6432139 | Screening Compounds and Building Blocks |
N-methyl-N-(6-nitro-1,3-benzothiazol-2-yl)glycine (6432139) | |||
ChemBridge特有类药化合物/先导化合物-6432139,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M12782 | ChemBridge-6809058 | ChemBridge化合物-6809058 | Screening Compounds and Building Blocks |
N-[4-(methylsulfonyl)-2-nitrophenyl]glycine (6809058) | |||
ChemBridge特有类药化合物/先导化合物-6809058,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M12905 | ChemBridge-7361080 | ChemBridge化合物-7361080 | Screening Compounds and Building Blocks |
N-cyclohexyl-N-[(4-fluorophenyl)sulfonyl]glycine (7361080) | |||
ChemBridge特有类药化合物/先导化合物-7361080,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M14365 | Glycylglycine | Glycylglycine | Metabolite/Endogenous Metabolite |
Glycylglycine 是最简单的多肽,可作为谷氨酰胺 (gamma-glutamyl) 的受体。 | |||
M14395 | N-Methylsarcosine | N-Methylsarcosine | Metabolite/Endogenous Metabolite |
Dimethylglycine; DMG; N,N-Dimethylglycine | |||
N-Methylsarcosine是用于合成蛋白质的氨基酸砌块,在体内少量存在。 | |||
M15091 | 2-(2-Phenylacetamido)acetic acid | 2-(2-Phenylacetamido)acetic acid | Metabolite/Endogenous Metabolite |
Phenaceturic Acid; Phenacetylglycine | |||
2-(2-Phenylacetamido)acetic acid 是一种内源性代谢产物。 | |||
M21460 | Cinnamoylglycine | Cinnamoylglycine | Metabolite/Endogenous Metabolite |
Cinnamoylglycine 是人体尿液代谢物,一种肉桂酸和的甘氨酸结合物。Cinnamoylglycine 被用作的尿液标志物,可作为在抗生素研究期之后定殖耐药性的标志物。 | |||
M21543 | N-(2-Cyanoethyl)glycine | N-(2-氰乙基)氨基乙酸 | Peptides |
AVG | |||
N-(2-Cyanoethyl)glycine(N-(2-氰乙基)氨基乙酸)是一种甘氨酸衍生物。 | |||
M22403 | Glycine methyl ester hydrochloride | 甘氨酸甲酯盐酸盐 | Others |
Glycine methyl ester hydrochloride | |||
M22404 | Glycine ethyl ester hydrochloride | 甘氨酸乙酯盐酸盐 | Others |
Glycine ethyl ester hydrochloride | |||
M22405 | Glycine benzyl ester p-toluenesulfonate salt | 甘氨酸苄酯对甲苯磺酸盐 | Others |
Glycine benzyl ester p-toluenesulfonate salt | |||
M30390 | N-Ethylglycine | N-Ethylglycine | Amino Acid Derivatives |
N-Ethylglycine 是一种甘氨酸衍生物。 | |||
M30460 | gamma-DGG | gamma-DGG | GluR |
γDGG; γ-D-Glutamylglycine | |||
gamma-DGG 是一种竞争性的 AMPA 受体阻断剂。 | |||
M31102 | Tricine | 三羟甲基甲基甘氨酸 | Solvents & Excipients |
N-tris(hydroxymethyl)methylglycine | |||
Tricine(三羟甲基甲基甘氨酸)是一种良好的缓冲物质,20 ℃时pKa = 8.15。 | |||
M39103 | 2-Phenylglycine | 2-Phenylglycine | Metabolite/Endogenous Metabolite |
2-Phenylglycine (DL-α-Phenylglycine) 是在 W2 至 W4 泌乳期间母乳中的代谢产物。 | |||
M39278 | (S)-(+)-2-Phenylglycine methyl ester hydrochloride | (S)-(+)-2-苯甘氨酸甲酯 盐酸盐 | Amino Acid Derivatives |
(S)-(+)-2-Phenylglycine methyl ester hydrochloride 是一种甘氨酸衍生物。 | |||
M39308 | Glycine tert-butyl ester hydrochloride | Glycine tert-butyl ester hydrochloride | Amino Acid Derivatives |
Glycine tert-butyl ester hydrochloride 是一种甘氨酸衍生物。 | |||
M39354 | N-(4-Cyanophenyl)glycine | N-(4-Cyanophenyl)glycine | Amino Acid Derivatives |
N-(4-Cyanophenyl)glycine 是一种甘氨酸衍生物。 | |||
M39355 | Boc-D-Cyclopropylglycine | Boc-D-Cyclopropylglycine | Amino Acid Derivatives |
Boc-D-Cyclopropylglycine 是一种小分子多肽,可用于化合物的合成。 | |||
M2584 | MDL-29951 | MDL-29951 | GluR |
MDL-29951 is a novel glycine antagonist of NMDA receptor activation (Ki=0.14 mM, [3H]glycine binding) in vitro and in vivo with IC50 value of 0.14 mM ([3H]glycine binding). | |||
M5464 | Bitopertin | 比拓喷丁 | GlyT |
RG1678, RO-4917838 | |||
Bitopertin (RG1678, RO-4917838)是有效的GlyT1(glycine transporter 1)抑制剂,在CHO细胞中IC50为25 nM。 | |||
M6691 | D-Serine | D-丝氨酸 | GluR |
D-Serine is a potentiator, acts at glycine site. | |||
M6745 | Gavestinel | Gavestinel | Others |
Gavestinel is a potent and selective glycine site antagonist; orally available and active in vivo. | |||
M6801 | Hypotaurine | 亚牛磺酸 | Others |
2-Aminoethanesulfinic acid | |||
Hypotaurine is a non-selective endogenous glycine receptor agonist. | |||
M8226 | MEGX | 去乙基利多卡因 | Others |
Monoethylglycinexylidide (MEGX) is an active metabolite of lidocaine. | |||
M8547 | Thiocolchicoside | 硫秋水仙苷;噻可撒可 | Others |
Thiocolchicoside is a potent competitive γ-aminobutyric acid type A (GABAA) receptor antagonist and glycine receptor agonist with muscle relaxant, anti-inflammatory, and analgesic activity. | |||
M8733 | K67 | K67 | Others |
K67 is a specific inhibitor against the interaction between KEAP1 (Kelch-like ECH-associated protein 1) DC (double glycine repeat and C-terminal region) domain and S349-phosphorylated (human Ser349, mouse Ser351) KIR (Keap1-interacting region). | |||
M14228 | MRZ 2-514 | MRZ 2-514 | GluR |
MRZ 2-514 是一种 NMDA receptor (glycineB) 的拮抗剂,Ki 值为 33 μM。 | |||
M18181 | 6,7,4'-Trihydroxyisoflavone | 6,7,4'-三羟基异黄酮 | CDK |
Desmethylglycitein (4',6,7-Trihydroxyisoflavone),大豆苷元的代谢产物,来源于大豆 Glycine max,具有抗氧化性和抗癌活性。 | |||
M20559 | Brucine sulfate heptahydrate | Brucine sulfate heptahydrate | Others |
Brucine is an alkaloid that acts as an antagonist at glycine receptors and paralyzes inhibitory neurons. | |||
M27771 | Soyasaponin IV | Soyasaponin IV | Others |
Soyasaponin IV 可从 Glycine soya 中分离得到,具有肝脏保护作用。 | |||
M28817 | ZD-9379 | ZD-9379 | GluR |
ZD-9379 是一种有效的,具有口服活性的,可穿过血脑屏障的 NMDA 受体甘氨酸位点 (glycine site) 拮抗剂。 | |||
M39137 | Betaine | 甜菜碱 | Metabolite/Endogenous Metabolite |
Betaine (Trimethylglycine) 是许多食物中发现的天然化合物,也是一种可维持正常 DNA 甲基化模式的活性甲基供体。Betaine 广泛存在于植物,动物,微生物和丰富的膳食来源中,包括海鲜,菠菜和麦麸。 |
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