目录号 | 产品名称 | 产品简介 |
---|---|---|
M4953 | Bafilomycin A1 | 巴佛洛霉素A1 Bafilomycin A1(Baf-A1)是一种液泡H+-ATPase抑制剂,IC50为0.44 nM。 |
M20514 | Omeprazole Sodium | Omeprazole Sodium is the sodium salt form of omeprazole, which is a proton pump inhibitor and suppresses gastric acid secretion. |
M20496 | Ilaprazole sodium | Ilaprazole sodium is the sodium salt form of ilaprazole, which is a proton pump inhibitor. |
M20452 | Revaprazan Hydrochloride | Revaprazan Hydrochloride is a new reversible proton pump inhibitor with long-lasting acid-suppressive effects. |
M20434 | Rabeprazole | Rabeprazole is an oral inhibitor of proton pump and blocks the production of acid by the stomach. |
M20397 | Pantoprazole | Pantoprazole is a proton pump inhibitor used for short-term treatment of erosion and ulceration of the esophagus caused by gastroesophageal reflux disease. |
M20394 | NEXIUM (esomeprazole magnesium) | Esomeprazole Magnesium is a proton pump inhibitor to reduce gastric acid secretion. |
M14268 | Vonoprazan | Vonoprazan (TAK-438 free base) 是一种质子泵抑制剂 (PPI),是高效的,具有口服活性的钾竞争性酸阻断剂 (potassium-competitive acid blocker, P-CAB),具有抗分泌活性。 |
M14266 | Soraprazan | Soraprazan (BYK61359) 是选择性的钾通道竞争性的 H,K-ATPase (Ki=6.4 nM)的抑制剂,在胃腺的 IC50 为 0.19 μM。Soraprazan 与 H,K-ATPase 结合,Kd为 28.27 nM。Soraprazan 对酸分泌有直接抑制作用,对 H,K-ATPase 的选择性是 Na,K- 和 Ca- ATPases 的 2000 倍以上。 |
M14265 | Pantoprazole sodium hydrate | Pantoprazole sodium hydrate (BY1023 sodium hydrate) 是一种具有口服活性的,有效质子泵 (proton pump) 抑制剂 (PPI)。Pantoprazole sodium hydrate 是一种取代的苯并咪唑,是一种有效的 H+/K+-ATPase 抑制剂,IC50 为 6.8 μM。 |
M4953 | Bafilomycin A1 | 巴佛洛霉素A1 Bafilomycin A1(Baf-A1)是一种液泡H+-ATPase抑制剂,IC50为0.44 nM。 |
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