| M20927
|
Betahistine mesylate |
Betahistine mesylate is the mesylate salt form of Betahistine, a histamine analog and H3 receptor agonist that serves as a vasodilator. |
| M20813
|
Cyclizine |
Cyclizine is a piperazine first-generation antagonist of histamine 1 receptor. |
| M20574
|
Thonzylamine |
Thonzylamine is an antihistamine and anticholinergic drug. |
| M20520
|
Chloropyramine hydrochloride |
Chloropyramine hydrochloride is a histamine receptor H1 antagonist and has anti-cholinergic, antispasmodic, and antiallergic effects. |
| M20515
|
Emedastine |
Emedastine is a potent, high affinity histamine H1-receptor-selective antagonist with Ki of 1.3 ±0.1 nM for H1-receptors while considerably weaker at H2- (K1 = 49,067 ± 11,113 nM) and H3-receptors (Ki = 12,430 ± 1,282 nM). |
| M20511
|
Betahistine |
Betahistine Dihydrochloride is a histamine H3 receptors inhibitor used as an antivertigo drug. |
| M20495
|
Cloperastine hydrochloride |
Cloperastine is a drug with a central antitussive effect, and is also endowed with an antihistaminic activity. |
| M20424
|
CarbinoxaMine Maleate |
Carbinoxamine maleate is a histamine-H1 receptor blocking agent with antihistamine and anticholinergic properties. |
| M13995
|
Adriforant hydrochloride |
Adriforant hydrochloride (PF-3893787 hydrochloride) 是一种新型的，具有口服活性的组胺 H4 受体亲和型拮抗剂 (Ki=2.4 nM)，同时也是H4 受体功能性拮抗剂 (Ki=1.56 nM)。可用于银屑病的相关研究。 |
| M13994
|
N-Acetylhistamine |
N-Acetylhistamine 是一种组胺代谢物。N-acetylhistamine 可用作过敏反应中组氨酸代谢的生物标志物。 |
| M13992
|
Chlorcyclizine hydrochloride |
Chlorcyclizine hydrochloride 是一种组胺 H1 拮抗剂。 |
| M13991
|
Bepotastine |
Bepotastine 是一种选择性的具有口服活性的第二代组胺 H1 受体 (histamine H1 receptor) 拮抗剂。Bepotastine 可用于过敏性鼻炎，过敏性结膜炎和荨麻疹/瘙痒症的研究。 |
| M11287
|
JNJ-39758979 |
JNJ-39758979是一种选择性的、具有口服活性的、高亲和力的组胺 H4 受体 (histamine H4 receptor) 拮抗剂，对人，小鼠，猴子的组胺 H4 受体的 Ki 值分别为 12.5、5.3 和 25 nM。JNJ-39758979 对组胺诱导的 cAMP 抑制作用具有拮抗作用，pA2 为 7.9。JNJ-39758979 具有良好的抗炎、止痒作用。 |
