POT-4 - 搜索结果 | AbMole中文官网

找到约 34 条 “POT-4” 相关结果（用时 0.073 秒）

目录号	产品名称	中文名称	靶点
M3173	Potassium canrenoate	坎利酸钾	Mineralocorticoid Receptor
	Aldadiene potassium, SC-14266
	Canrenoate potassium 是一种释放 canrenone 的前药，也是一种有效的竞争性盐皮质激素受体 (mineralocorticoid receptor) 拮抗剂。Canrenoate potassium 作为一种利尿剂，用于高血压的研究。
M11700	ChemBridge-5141951	ChemBridge化合物-5141951	Screening Compounds and Building Blocks
	potassium 4-{[4-(allyloxy)-3,5-dibromophenyl]sulfonyl}-2,6-dibromobenzenolate (5141951)
	ChemBridge特有类药化合物/先导化合物-5141951，由AbMole（奥默生物）独家提供。具体售价货期请咨询AbMole（奥默生物）。运费额外计算。
M45466	ChemBridge-5152690	ChemBridge化合物-5152690	Screening Compounds and Building Blocks
	potassium 7-hydroxy-4,5-dihydronaphtho[1,2-c][1,2,5]oxadiazole-5-sulfonate 3-oxide (5152690)
	ChemBridge特有类药化合物/先导化合物-5152690，由AbMole（奥默生物）独家提供。具体售价货期请咨询AbMole（奥默生物）。运费额外计算。
M54080	POT-4	POT-4	Complement System
	POT-4 (AL-78898A)，一种 Compstatin 衍生物，是补体因子 C3 激活的有效抑制剂。
M2144	Topotecan hydrochloride	盐酸拓扑替康；盐酸拓普替康；拓普替康	Topoisomerase
	Hycamtin, NSC 609669
	Topotecan HCl是一种拓扑异构酶I（Topoisomerase I）抑制剂，作用于MCF-7 Luc细胞和DU-145 Luc细胞，IC50分别为13 nM和2 nM。
M2181	ML133 hydrochloride	ML133 hydrochloride	Potassium Channel
	ML133 HCl
	ML133 HCl是一种选择性钾离子通道（Potassium Channel）抑制剂，作用于K_ir2.1， IC50为1.8 μM (pH 7.4)和290 nM (pH 8.5)，对K_ir1.1没有作用效果，对K_ir4.1和K_ir7.1具有微弱的作用活性。
M2608	Kobe0065	Kobe0065	Ras
	Kobe0065 is a novel and effective small-molecule compound inhibiting Ras–Raf interaction by SBDD, exhibits potent activity to competitively inhibit the binding of H-Ras·GTP to c-Raf-1 RBD with a Ki value of 46 ± 13 μM.
M5029	WHI-P180	WHI-P180	CDK
	Janex 3
	WHI-P180 is a potent EGFR and Cdk2 inhibitors with IC50 of 4.0 and 1.0 uM, respectively.
M5078	(S)-Willardiine	(S)-Willardiine	GluR
	(-)-Willardiine
	(S)-Willardiine is a potent agonist of AMPA/kainate receptors with EC50 of 44.8 uM.
M6508	BIO 5192	BIO 5192	Others
	BIO 5192 is a highly potent and selective inhibitor of integrin α ₄β ₁.
M6606	Cinalukast	西那司特	Others
	Cinalukast is a potent, selective CysLT ₁(LTD ₄) antagonist; orally active.
M6642	CYM 50260	CYM 50260	S1P Receptor
	CYM 50260 is a potent and selective S1P₄ agonist.
M6701	Eggmanone	Eggmanone	Others
	Eggmanone is a potent and selective PDE4 inhibitor; suppresses hedgehog signaling.
M6716	ER 819762	ER 819762	Others
	ER 819762 is a potent EP ₄ receptor antagonist; orally bioavailable.
M7222	RS 25344 hydrochloride	RS 25344 hydrochloride	Others
	RS 25344 hydrochloride is a potent PDE4 inhibitor.
M7250	SB 204070	SB 204070	Others
	SB 204070 is a potent and selective 5-HT ₄ antagonist.
M7292	SIB 1508Y maleate	SIB 1508Y maleate	Others
	SIB 1508Y maleate is a potent agonist of α4β2, α2β4, α4β4 and α3β4 nACh receptors.
M7378	TC-N 22A	TC-N 22A	Others
	TC-N 22A is a potent, selective mGlu ₄ positive allosteric modulator.
M7399	TC-T 6000	TC-T 6000	Others
	TC-T 6000 is a potent equilibrative nucleoside transporter 4 (ENT4) inhibitor.
M7467	VU 0155041	VU 0155041	Others
	VU 0155041 is a potent, positive allosteric mGlu ₄ agonist.
M7468	VU 0155041 sodium salt	VU 0155041 sodium salt	Others
	VU 0155041 sodium salt is a potent, positive allosteric mGlu 4 agonist.
M7479	VUF 8430 dihydrobromide	VUF 8430 dihydrobromide	Others
	VUF 8430 dihydrobromide is a potent, high affinity H ₄ agonist.
M7731	CHIC-35	CHIC-35	Others
	CHIC-35 is cell-permeable, metabolically stable, and very potent inhibitor of SIRT1; IC₅₀ of S-isomer is 60 nM; IC₅₀ of mixed isomers is 124 nM.
M7828	Hypothemycin	寄端霉素	Others
	Hypothemycin, one of the highly oxygenated analogues in the group of 14-membered resorcylic acid lactones (RAL).
M7935	ML 10302	ML 10302	Others
	Potent, selective 5-HT₄ serotonin receptor agonist.
M8158	SDZ-205,557 hydrochloride	SDZ-205,557 hydrochloride	Others
	Potent, selective 5-HT₄ serotonin receptor antagonist.
M8223	VU591	VU591	Potassium Channel
	VU591 is a Potassium Inwardly-Rectifying Channel (KCNJ1 or ROMK) specific inhibitor (IC50 = 240 nM) that is closely related to VU590.
M8282	Deformylflustrabromine hydrochloride	Deformylflustrabromine hydrochloride	Others
	Deformylflustrabromine hydrochloride; dFBr hydrochloride
	Desformylflustrabromine (dFBr) is a potent, selective positive allosteric modulator of α4β2 nicotinic receptor; increases efficacy and potency of acetylcholine.
M8415	CID44216842	CID44216842	Others
	CID44216842 is a potent and selective non-competitive allosteric inhibitor of Cdc42 GTPase that does not inhabit Rho and Rac.
M8431	CYM50358	CYM50358	S1P Receptor
	CYM50358 is a potent, selective antagonist of the sphingosine-1-phosphate receptor 4 (S1P₄).
M8496	NSC687852	NSC687852	Others
	NSC687852 is a cell-permeable, potent, reversible and selective inhibitor of 19S regulatory-particle-associated deubiquitinases (DUBs) UCHL5 and USP14, with no effect on UCH-L1, UCH-L3, USP2, USP7, USP8 and BAP1.
M8503	SB-207266	SB-207266	5-HT Receptor
	SB-207266 is a potent, selective, orally active and long-acting 5-HT4 antagonist in vivo.
M8557	CS1	CS1	Others
	CS1 is a selective and potent inhibitor of topoisomerase IIα (TopoIIα) that potently inhibits a proliferation of cancer cell lines including MDA-MB-231 and A548 cells, with less toxicity than etoposide.
M8598	ZQ-16	ZQ-16	Others
	ZQ-16 is a potent and selective agonist for medium-chain free fatty acid receptor GPR84 (G protein-coupled receptor 84).

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