找到约 50 条 “OT-82” 相关结果 (用时 0.096 秒)
目录号 | 产品名称 | 中文名称 | 靶点 |
---|---|---|---|
M3379 | Trifluridine | 曲氟胸苷;曲氟尿苷 | DNA/RNA Synthesis |
Trifluridine; FTD; 5-Trifluorothymidine; NSC 529182; NSC 75520 | |||
Trifluridine(曲氟胸苷,曲氟尿苷)是一种氟化嘧啶核苷,同时也是胸苷酸合酶的抑制剂,具有抗肿瘤活性,对1型和2型单纯疱疹病毒表现出有效的抑制作用。此外,Trifluridine还具有抗癌活性,能在细胞摄取后掺入癌细胞的DNA中,从而在细胞复制过程中干扰DNA功能。可用于角膜炎和结膜炎的相关研究。 | |||
M5116 | Formoterol Hemifumarate | 富马酸福莫特罗 | Adrenergic Receptor |
Eformoterol, CGP 25827A, NSC 299587, YM 08316 | |||
Formoterol Hemifumarate 是一种强效、选择性和长效的β2-肾上腺素受体( β2-adrenoceptor)激动剂。 | |||
M10214 | Agouti-related Protein (AGRP) (25-82), human | Agouti-related Protein (AGRP) (25-82), human | Peptides |
Agouti-related protein (AgRP) is a neuropeptide produced in the brain by the AgRP/NPY neuron. | |||
M11666 | ChemBridge-5131382 | ChemBridge化合物-5131382 | Screening Compounds and Building Blocks |
N'-(2-hydroxybenzylidene)isonicotinohydrazide (5131382) | |||
ChemBridge特有类药化合物/先导化合物-5131382,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M11949 | ChemBridge-5273682 | ChemBridge化合物-5273682 | Screening Compounds and Building Blocks |
1-(4-bromobenzoyl)-1H-1,2,3-benzotriazole (5273682) | |||
ChemBridge特有类药化合物/先导化合物-5273682,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M12280 | ChemBridge-5682321 | ChemBridge化合物-5682321 | Screening Compounds and Building Blocks |
4-{[3,6-bis(ethoxycarbonyl)-4,5,6,7-tetrahydrothieno[2,3-c]pyridin-2-yl]amino}-4-oxobutanoic acid (5682321) | |||
ChemBridge特有类药化合物/先导化合物-5682321,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M12822 | ChemBridge-6948261 | ChemBridge化合物-6948261 | Screening Compounds and Building Blocks |
N-(2-ethoxy-4-nitrophenyl)-2-(3-oxo-3,4-dihydro-2H-1,4-benzothiazin-2-yl)acetamide (6948261) | |||
ChemBridge特有类药化合物/先导化合物-6948261,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M12872 | ChemBridge-7117827 | ChemBridge化合物-7117827 | Screening Compounds and Building Blocks |
5-(2-thienyl)-2-thioxo-2,3-dihydrothieno[2,3-d]pyrimidin-4(1H)-one (7117827) | |||
ChemBridge特有类药化合物/先导化合物-7117827,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M13014 | ChemBridge-7826786 | ChemBridge化合物-7826786 | Screening Compounds and Building Blocks |
methyl 2-{[({4-[(1-adamantylamino)sulfonyl]phenyl}amino)carbonothioyl]amino}-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate (7826786) | |||
ChemBridge特有类药化合物/先导化合物-7826786,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M13105 | ChemBridge-7958223 | ChemBridge化合物-7958223 | Screening Compounds and Building Blocks |
2-[(4,6-diamino-2-pyrimidinyl)thio]-N-(6-ethoxy-1,3-benzothiazol-2-yl)acetamide (7958223) | |||
ChemBridge特有类药化合物/先导化合物-7958223,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M13128 | ChemBridge-7980582 | ChemBridge化合物-7980582 | Screening Compounds and Building Blocks |
4-hydroxy-3-methoxy-N,N-dimethylbenzenecarbothioamide (7980582) | |||
ChemBridge特有类药化合物/先导化合物-7980582,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M20622 | Naquotinib(ASP8273) | Naquotinib(ASP8273) | EGFR/HER2 |
Naquotinib(ASP8273) is an orally available, irreversible, mutant-selective, epidermal growth factor receptor (EGFR) inhibitor, with potential antineoplastic activity. | |||
M20823 | OT-82 | OT-82 | NAMPT |
OT-82 is a novel nicotinamide phosphoribosyltransferase (NAMPT) inhibitor with average IC50s of 13.03 nM in non-HP cancer cells and 2.89 nM in HP cancer cells, respectively. | |||
M45520 | ChemBridge-5248266 | ChemBridge化合物-5248266 | Screening Compounds and Building Blocks |
3-chloro-N-[3-(4-morpholinyl)propyl]-1-benzothiophene-2-carboxamide (5248266) | |||
ChemBridge特有类药化合物/先导化合物-5248266,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M45770 | ChemBridge-5976826 | ChemBridge化合物-5976826 | Screening Compounds and Building Blocks |
N-[2-({2-[(4-isopropylphenyl)amino]-2-oxoethyl}thio)-1,3-benzothiazol-6-yl]-2-[(1-phenyl-1H-tetrazol-5-yl)thio]acetamide (5976826) | |||
ChemBridge特有类药化合物/先导化合物-5976826,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M45810 | ChemBridge-6082112 | ChemBridge化合物-6082112 | Screening Compounds and Building Blocks |
2-[(2,4,6-trioxotetrahydro-5(2H)-pyrimidinylidene)methyl]phenyl 2-naphthalenesulfonate (6082112) | |||
ChemBridge特有类药化合物/先导化合物-6082112,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M46011 | ChemBridge-6898204 | ChemBridge化合物-6898204 | Screening Compounds and Building Blocks |
N-(3-chloro-2-methylphenyl)-4-methyl-1-piperazinecarbothioamide (6898204) | |||
ChemBridge特有类药化合物/先导化合物-6898204,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M46033 | ChemBridge-6982699 | ChemBridge化合物-6982699 | Screening Compounds and Building Blocks |
7-(2-chlorophenyl)-5-(4-fluorophenyl)-4,7-dihydrotetrazolo[1,5-a]pyrimidine (6982699) | |||
ChemBridge特有类药化合物/先导化合物-6982699,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M46060 | ChemBridge-7112828 | ChemBridge化合物-7112828 | Screening Compounds and Building Blocks |
2-(1H-benzimidazol-2-ylthio)-N-(2-{[2-(tert-butylamino)-2-oxoethyl]thio}-1,3-benzothiazol-6-yl)acetamide (7112828) | |||
ChemBridge特有类药化合物/先导化合物-7112828,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M46275 | ChemBridge-7787282 | ChemBridge化合物-7787282 | Screening Compounds and Building Blocks |
N-(5-chloro-2-methoxyphenyl)-1-pyrrolidinecarbothioamide (7787282) | |||
ChemBridge特有类药化合物/先导化合物-7787282,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M46298 | ChemBridge-7803828 | ChemBridge化合物-7803828 | Screening Compounds and Building Blocks |
ethyl 4-({[(4-chloro-2,5-dimethoxyphenyl)amino]carbonothioyl}amino)benzoate (7803828) | |||
ChemBridge特有类药化合物/先导化合物-7803828,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M46325 | ChemBridge-7822325 | ChemBridge化合物-7822325 | Screening Compounds and Building Blocks |
4-({[(1,3-benzodioxol-5-ylamino)carbonothioyl]amino}methyl)benzoic acid (7822325) | |||
ChemBridge特有类药化合物/先导化合物-7822325,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M46326 | ChemBridge-7822832 | ChemBridge化合物-7822832 | Screening Compounds and Building Blocks |
4-({[(5-tert-butyl-2-methoxyphenyl)amino]carbonothioyl}amino)benzenesulfonamide (7822832) | |||
ChemBridge特有类药化合物/先导化合物-7822832,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M46329 | ChemBridge-7826969 | ChemBridge化合物-7826969 | Screening Compounds and Building Blocks |
N-[4-({[(4-isopropylphenyl)amino]carbonothioyl}amino)phenyl]-N-methylacetamide hydrochloride (7826969) | |||
ChemBridge特有类药化合物/先导化合物-7826969,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M46331 | ChemBridge-7829543 | ChemBridge化合物-7829543 | Screening Compounds and Building Blocks |
N-(3,4-dichlorophenyl)-4-({[(3,4-dimethoxyphenyl)amino]carbonothioyl}amino)benzenesulfonamide (7829543) | |||
ChemBridge特有类药化合物/先导化合物-7829543,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M46425 | ChemBridge-7932782 | ChemBridge化合物-7932782 | Screening Compounds and Building Blocks |
7-(4-fluorophenyl)-5-(3-pyridinyl)-4,5,6,7-tetrahydrotetrazolo[1,5-a]pyrimidine (7932782) | |||
ChemBridge特有类药化合物/先导化合物-7932782,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M46445 | ChemBridge-7947827 | ChemBridge化合物-7947827 | Screening Compounds and Building Blocks |
3-chloro-N-[3-(4-morpholinylsulfonyl)phenyl]-1-benzothiophene-2-carboxamide (7947827) | |||
ChemBridge特有类药化合物/先导化合物-7947827,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M46574 | ChemBridge-8824789 | ChemBridge化合物-8824789 | Screening Compounds and Building Blocks |
ethyl 4-{[({4-[(2-methyl-1-piperidinyl)sulfonyl]phenyl}amino)carbonothioyl]amino}benzoate (8824789) | |||
ChemBridge特有类药化合物/先导化合物-8824789,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M46576 | ChemBridge-8825115 | ChemBridge化合物-8825115 | Screening Compounds and Building Blocks |
isopropyl 4-({[(3,5-dimethoxyphenyl)amino]carbonothioyl}amino)benzoate (8825115) | |||
ChemBridge特有类药化合物/先导化合物-8825115,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M46577 | ChemBridge-8826004 | ChemBridge化合物-8826004 | Screening Compounds and Building Blocks |
N-(tert-butyl)-4-({[(4-isopropylphenyl)amino]carbonothioyl}amino)benzenesulfonamide (8826004) | |||
ChemBridge特有类药化合物/先导化合物-8826004,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M2150 | Oprozomib | 奥泼佐米 | Proteasome |
ONX 0912, PR-047 | |||
Oprozomib (ONX 0912)是一种口服生物有效的抑制剂,抑制20S proteasome(20S蛋白酶体)β5/LMP7的CT-L活性,IC50为36 nM/82 nM。 | |||
M6206 | ARV-825 | ARV-825 | Epigenetic Reader Domain |
ARV-825 是一种 PROTAC 类的 BRD4 抑制剂。ARV-825 对 BRD4 的 BD1 和 BD2 结构域具有高亲和力,Kds 值分别为 90 和 28 nM | |||
M7834 | HMBA | HMBA | Others |
HMBA is an Inhibitor of microtubule polymerization; apoptosis inducer. | |||
M8330 | Carboxyamidotriazole | Carboxyamidotriazole | Others |
Carboxyamidotriazole (L-651582) is an orally active calcium channel blocker. | |||
M9749 | Cotadutide acetate | 醋酸可妥度肽 | GLP Receptor |
MEDI0382 acetate | |||
Cotadutide acetate(MEDI0382 acetate)是Cotadutide的乙酸盐形式,同时也是一种有效的胰高血糖素样肽-1受体(GLP-1R)和胰高血糖素受体(GCGR)的双重肽激动剂,EC50值分别为6.9 pM和10.2 pM。 | |||
M9824 | MZ 1 | MZ 1 | PROTAC |
MZ1 | |||
MZ 1是一种PROTAC BRD4降解剂,对BRD4 BD1/2,BRD3 BD1/2和BRD2 BD1/2的Kd值分别为382/120,119/115和307/228 nM。 | |||
M13686 | MKC8866 | MKC8866 | IRE1 |
MKC8866 是一种水杨醛类似物,有效的选择性 IRE1 RNase 抑制剂,在体外的 IC50 为 0.29 μM。 MKC8866 强烈抑制 Dithiothreitol 诱导的 XBP1s 表达,EC50 为 0.52 μM。MKC8866 抑制无应激 RPMI 8226 细胞,IC50 为 0.14 μM。 MKC8866 抑制乳腺癌细胞中的 IRE1 RNase 导致促肿瘤发生因子减少,同时也能抑制前列腺癌 (PCa) 肿瘤的生长。 | |||
M14139 | Naquotinib mesylate | Naquotinib mesylate | EGFR/HER2 |
ASP8273 (mesylate) | |||
Naquotinib mesylate (ASP8273 mesylate) 是有口服活性,不可逆的 EGFR 突变体抑制剂;对EGFR突变体和EGFR的 IC50 值分别为8-33和230 nM。 | |||
M14871 | Gefitinib-based PROTAC 3 | Gefitinib-based PROTAC 3 | PROTAC |
Gefitinib-based PROTAC 3,通过 linker 将 EGFR 结合元件与 von Hippel-Lindau 配体结合,作用于 HCC827 (外显子 19 缺失) 和 H3255 (L858R 突变) 细胞,诱导 EGFR 降解,DC50 分别为 11.7 nM 和 22.3 nM。 | |||
M20515 | Emedastine | Emedastine | Histamine Receptor |
Emedastine is a potent, high affinity histamine H1-receptor-selective antagonist with Ki of 1.3 ±0.1 nM for H1-receptors while considerably weaker at H2- (K1 = 49,067 ± 11,113 nM) and H3-receptors (Ki = 12,430 ± 1,282 nM). | |||
M20742 | Y06036 | Y06036 | Epigenetic Reader Domain |
Y06036 (compound 6i) is a potent and selective inhibitor of BET with antitumor activity. Y06036 binds to the BRD4(1) bromodomain with Kd of 82 nM. | |||
M24987 | Baloramotide | Baloramotide | Others |
Baloramotide 是一种含有 182 个氨基酸的重组蛋白 NY-ESO-1。Baloramotide 可以增强免疫系统对肿瘤的反应。 | |||
M28236 | OTS447 | OTS447 | FLT3 |
OTS447 是一种有效的 FLT3 抑制剂,IC50 为 21 nM (WO2012016082A1, compound 335)。 | |||
M31215 | Cotadutide | 可妥度肽 | Glucagon Receptor |
Cotadutide (MEDI0382) 是一种有效的胰高血糖素样肽-1 (GLP-1) 和胰高血糖素受体 (GCGR) 双重激动剂,EC50 值分别为 6.9 pM 和 10.2 pM。Cotadutide 可控制血糖,以及减轻纤维化。Cotadutide 可用于肥胖和 2 型糖尿病 (T2D) 的研究。 | |||
M31351 | Dirucotide | Dirucotide | Others |
MBP8298 | |||
Dirucotide(MBP8298)是一种包含17 个氨基酸的合成肽,其序列与部分人髓鞘碱性蛋白(MBP)的序列相同,同时也是一种MBP调节剂。可用于多发性硬化症 (MS) 等中枢神经系统自身免疫性疾病的研究。 | |||
M43435 | PROTAC BRD4 Degrader-17 | PROTAC BRD4 Degrader-17 | PROTAC |
PROTAC BRD4 Degrader-17 是一种有效的 PROTAC BRD4 降解剂,IC50 值为 29.54 nM (BRD4 (BD1) ) 和 3.82 nM (BRD4 (BD2))。 | |||
M51324 | Agouti-Related Protein (54-82) (human) | Agouti-Related Protein (54-82) (human) | Others |
Agouti-Related Protein (54-82) (human) (AGRP (54-82) (human)) 是刺鼠关联蛋白 (AGRP) 的氨基末端 54-82 氨基酸片段。 | |||
M51547 | C3bot(154-182) | C3bot(154-182) | Others |
C3bot(154-182) 是一种 C3 肽,通过改善下行纤维束的再生生长来增强脊髓损伤的恢复能力。 | |||
M51617 | C-Reactive Protein (CRP) (77-82) | C-Reactive Protein (CRP) (77-82) | Others |
C-Reactive Protein (CRP) 77-82 是 C-反应蛋白的 77-82 片段。 | |||
M54343 | Myelin Basic Protein (MBP) (68-82), guinea pig | Myelin Basic Protein (MBP) (68-82), guinea pig | Others |
Myelin Basic Protein (MBP) (68-82), guinea pig 是髓鞘碱性蛋白 (MBP) 的一个片段。 |
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