找到约 40 条 “Compound E” 相关结果 （用时 0.172 秒）
| 目录号 | 产品名称 | 中文名称 | 靶点 |
|---|---|---|---|
M5534
|
Cortisone | 可的松 | GCR |
| 17-Hydroxy-11-dehydrocorticosterone; Kendall's compound E | |||
| Cortisone是一种用于治疗感染或过敏的激素药物 | |||
| M7043 | NPS ALX Compound 4a dihydrochloride | NPS ALX Compound 4a dihydrochloride | Others |
| NPS ALX Compound 4a dihydrochloride is a potent and selective 5-HT 6 antagonist. | |||
| M9505
|
Compound E | Compound E | Gamma-secretase/Beta-secretase |
| GSI-XXI; γ-secretase inhibitor XXI; γ-Secretase-IN-1 | |||
| Compound E 是一种可透过细胞的强效选择性γ-分泌酶（γ-secretase）和Notch抑制剂。 | |||
| M11655 | ChemBridge-5126190 | ChemBridge化合物-5126190 | Screening Compounds and Building Blocks |
| 3,7-dihydro-1H-purine-2,6-dione (5126190) | |||
| ChemBridge特有类药化合物/先导化合物-5126190，由AbMole（奥默生物）独家提供。具体售价货期请咨询AbMole（奥默生物）。运费额外计算。 | |||
| M12301 | ChemBridge-5713492 | ChemBridge化合物-5713492 | Screening Compounds and Building Blocks |
| 1-(2-chloro-4-nitrophenyl)-4-[(5-methyl-3-phenyl-4-isoxazolyl)carbonyl]piperazine (5713492) | |||
| ChemBridge特有类药化合物/先导化合物-5713492，由AbMole（奥默生物）独家提供。具体售价货期请咨询AbMole（奥默生物）。运费额外计算。 | |||
| M12806 | ChemBridge-6881166 | ChemBridge化合物-6881166 | Screening Compounds and Building Blocks |
| 4-[(2-{[1-(4-ethylphenyl)-2,4,6-trioxotetrahydro-5(2H)-pyrimidinylidene]methyl}phenoxy)methyl]benzoic acid (6881166) | |||
| ChemBridge特有类药化合物/先导化合物-6881166，由AbMole（奥默生物）独家提供。具体售价货期请咨询AbMole（奥默生物）。运费额外计算。 | |||
| M20547
|
Rabeprazole Related Compound E | Rabeprazole Related Compound E | Proton Pump |
| Rabeprazole thioether; Rabeprazole Sulfide | |||
| Rabeprazole Related Compound E是 Rabeprazole 的活性代谢产物，同时也是一种具有口服活性的质子泵抑制剂，能通过与胃壁细胞中的 (H+/K+)-ATPase 相互作用来抑制胃酸分泌。此外，Rabeprazole Related Compound E 还能显著抑制幽门螺旋杆菌的活性，可用于各种消化系统疾病的相关研究。 | |||
| M20688 | B-Raf inhibitor 1 (Compound 13) dihydrochloride | B-Raf inhibitor 1 (Compound 13) dihydrochloride | Raf |
| B-Raf inhibitor 1 (Compound 13) is a type IIA Raf inhibitor which bind to the DFG-out conformation with ki of 1 nM,1 nM,and 0.3 nM for B-Raf(WT), B-Raf(V600E) and C-Raf, respectively. | |||
| M21681
|
Compound 48/80 trihydrochloride | Compound 48/80 trihydrochloride | Phospholipase |
| C48/80 trihydrochloride | |||
| Compound 48/80 trihydrochloride 作为选择性肥大细胞激活剂广泛用于动物和组织模型。Compound 48/80 作用于肥大细胞膜，刺激三聚体 G 蛋白，并通过磷脂酶 C 和 D 途径诱导脱颗粒。 | |||
| M55555 | PI3K/Akt/CREB activator 1 | PI3K/Akt/CREB activator 1 | PI3K |
| compound AE-18 | |||
| PI3K/Akt/CREB activator 1 (compound AE-18) 是一种口服有效的 PI3K/Akt/CREB 的激活剂。PI3K/Akt/CREB activator 1 通过 PI3K/Akt/CREB 通路上调脑源性神经营养因子，促进神经元增殖，诱导 Neuro-2a 细胞分化成神经元样形态，加速海马原代神经元轴突-树突极化的建立。 | |||
| M56074 | NPS ALX Compound 4a dihydrochloride | NPS ALX Compound 4a dihydrochloride | 5-HT Receptor |
| NPS ALX Compound 4a dihydrochloride 是一种有效的、选择性的 5-羟色胺受体 6 (5-HT6) 受体拮抗剂，IC50 值为 7.2 nM，且具有高亲和力，Ki 值为 0.2 nM。 | |||
| M58107 | PD-1/PD-L1-IN-9 | PD-1/PD-L1-IN-9 | PD-1/PD-L1 |
| PD-1/PD-L1-IN-9 是一种有效和具有口服活性的 PD-1/PD-L1 相互作用抑制剂，IC50 值为 3.8 nM。PD-1/PD-L1-IN-9 可以增强免疫细胞对肿瘤细胞的杀伤活性。PD-1/PD-L1-IN-9 在 CT26 小鼠模型中表现出显着的体内抗肿瘤活性。 | |||
| M2896
|
OAC1 | OAC1 | Others |
| OAC1 (Oct4-activating compound 1)是一种有效的 Oct4 激活剂，能激活 Oct4 和 Nanog 启动子，促进诱导多功能干细胞 (iPSC) 的形成，以及通过上调 HOXB4 表达激活 OCT4。此外，OAC1 还能增加Oct4-Nanog-Sox2 三联体和 TET1 的转录，并可通过提高效率和缩短重编程时间，促进细胞的重编程。 | |||
| M4088
|
Ginsenoside Compound-K | 人参皂苷CK | COX |
| Ginsenoside K; Ginsenoside C-K | |||
| Ginsenoside Compound-K(人参皂苷CK)是一种 Ginsenoside Rb1 细菌代谢物，通过抑制诱生型一氧化氮合酶 (iNOS) 和 COX-2，从而发挥抗炎作用。 | |||
| M4902
|
Chloroxine | 氯喔星；克氯辛 | Antibiotic |
| Chloroxine is a synthetic antibacterial compound that is effective in the treatment of dandruff and seborrheic dermatitis when incorporated in a shampoo. | |||
| M4924
|
Dehydroacetic acid | 脱氢乙酸 | Antibiotic |
| Biocide 470F | |||
| Dehydroacetic acid is an organic compound, classified as a pyrone derivative and is used mostly as a fungicide and bactericide. | |||
| M4961
|
CB72666407 | CB72666407 | mTOR |
| Pyrimidine substituted purine compounds as kinase (S) inhibitors. | |||
| M4987
|
Procyanidin B4 | Procyanidin B4 | Others |
| A series of dimeric procyanidins (1-9) and some related polyphenols (10-15) were chosen as model compounds in a comparative investigation for various biological activities in order to obtain structure-activity relationships. | |||
| M5007
|
Hexyl Chloroformate | 己基甲酸氯 | Others |
| The Carbonochloridic acid,hexyl ester, belongs to the following product categories: (1)Acid Halides; (2)Carbonyl Compounds; (3)Organic Building Blocks. It has the systematic name of hexyl carbonochloridate. | |||
| M6285
|
Glutaminase C-IN-1 | Glutaminase C-IN-1 | Glutaminase |
| Compound 968 | |||
| Glutaminase C-IN-1 (Compound 968) 是一种Glutaminase C变构抑制剂。 | |||
| M7400 | Teijin compound 1 | Teijin compound 1 | Others |
| Teijin compound 1 is a potent CCR2b antagonist. | |||
| M7946 | Naloxone methiodide | Naloxone methiodide | Others |
| Quaternary salt of naloxone that, like the parent compound, is a nonselective antagonist at opioid receptors. | |||
| M8161 | SE 175 | SE 175 | Others |
| An organic nitrate compound that acts as an NO donor in vivo following reductive transformation of the nitrate group to nitric oxide. | |||
| M8166 | Sulindac sulfide | 硫化舒林酸 | Others |
| Sulindac sulfide is a non-steroidal anti-inflammatory compound with a preference for COX-1; it is an inhibitor of Ras activation of Raf-1. | |||
| M8211
|
Triacetyl resveratrol | 乙酰化白藜芦醇 | STAT |
| Triacetyl resveratrol displays superior bioavailability to the parent compound, resveratrol. | |||
| M8246 | GPR35 Agonist, Compound 10 | GPR35 Agonist, Compound 10 | Others |
| GPR35 agonist Compound 10 is a GPR35 agonist the binds with higher affinity than other known agonists, such as kynurenic acid and zaprinast. | |||
| M8609 | MM-206 | MM-206 | Others |
| MM-206 is a cell-permeable, non-cytotoxic naphthalene sulfonamide compound effectively inhibits STAT3 DNA-binding activity (IC50 = 2. | |||
| M8635 | Displurigen | Displurigen | Others |
| Displurigen is a cell-permeable, phenylthiochromen-4-one derived compound that disrupts the pluripotency of human embryonic stem cells by targeting HSPA8/HSC70 and affects its binding to Oct4. | |||
| M8639 | STK16-IN-1 | STK16-IN-1 | Others |
| STK16-IN-1 is a cell-permeable pyrrolonaphthyridinone compound that acts as an ATP-competitive inhibitor against NAK (Numb Associated Kinase) family serine/threonine kinase STK16 (IC50/substrate = 0. | |||
| M8640
|
SW044248 | SW044248 | Topoisomerase |
| SW044248 is a cell permeable, indolotriazine-based compound that selectively inhibits topoisomerase 1 (Top 1), but not Top 2, catalyzed DNA decatenation in a manner distinct from that of camptothecin (Cat. | |||
| M8647
|
Raptinal | Raptinal | Caspase |
| Raptinal is a cell-permeable bifluorene-dicarbaldehyde compound that acts as a rapid activator of mitochondrial pathway-mediated intrinsic apoptosis. | |||
| M8668 | MI-4F | MI-4F | Others |
| MI-4F is mesoionic compound that exhibits potent anticancer activity against multiple cancer cell lines and in vivo. | |||
| M8706 | NSC57969 | NSC57969 | Others |
| NSC57969 is a MDR-selective compound that exhibits a robust Pgp-dependent toxic activity across diverse cancer cell lines. | |||
| M8717 | PBOX-6 | PBOX-6 | Others |
| PBOX-6 belongs to a group of tubulin-targeting pyrrolo-1,5-benzoxazepine (PBOX) compounds that potently induce apoptosis in a wide spectrum of cancer cells, including those originating from the four main types of leukemia. | |||
| M8723 | PBOX-15 | PBOX-15 | Others |
| PBOX-15 belongs to a group of tubulin-targeting pyrrolo-1,5-benzoxazepine (PBOX) compounds that potently induce apoptosis in a wide spectrum of cancer cells, including those originating from the four main types of leukemia. | |||
| M8884
|
Febantel | 非班太尔 | Parasite |
| Rintal, Combotel | |||
| Febantel is a veteran anthelmintic (wormer) compound belonging to the chemical class of the benzimidazoles. | |||
| M9031
|
6-Methylcoumarin | 6-Methylcoumarin | Others |
| Toncarine | |||
| 6-Methylcoumarin belongs to the class of organic compounds known as coumarins and derivatives. | |||
| M9461
|
Oxyclozanide | 氯羟柳胺；五氯柳胺；羟氯柳苯胺 | Anti-infection |
| 五氯柳胺Oxyclozanide is a salicylanilide anthelmintic compound, which acts by uncoupling oxidative phosphorylation in flukes. | |||
| M10351
|
IKarisoside A | 大花淫羊藿苷 A | Others |
| Baohuoside II | |||
| IKarisoside A is a natural compound isolated from Epimedium koreanum (Berberidaceae) with anti-inflammatory properties. | |||
| M10418
|
Malvidin chloride | 氯化锦葵素；锦葵色素；氯化锦葵色素 | Others |
| Syringidin | |||
| Malvidin (chloride) is a bioactive compound demonstrates antioxidant capacity with free radical scavenging properties in vitro. | |||
