找到约 33 条 “Xanthone” 相关结果 (用时 0.056 秒)
目录号 | 产品名称 | 中文名称 | 靶点 |
---|---|---|---|
M4191 | Polygalaxanthone-III | 远志山酮III | Cytochrome P450 (e.g. CYP17) |
Polygalaxanthone III 从远志 polygala tenuifolia wild 中提取,对 CYP450 酶具有抑制作用。Polygalaxanthone III抑制由 CYP2E1 催化的氯唑沙宗 6-羟基化,IC50 为 50.56μM。 | |||
M10680 | AH 6809 | 6-异丙氧基-9-氧代氧杂蒽-2-羧酸 | Prostaglandin Receptor |
6-Isopropoxy-9-xanthone-2-carboxylicacid | |||
AH 6809 是一种 EP 和 DP 受体的拮抗剂,对克隆的人类 EP1,EP2,EP3-III 和 DP 受体的 Ki 值分别为 1217、1150、1597 和 1415 nM,对小鼠 EP2 受体的 Ki 值为 350 nM。 | |||
M13478 | Xanthone | 呫吨酮 | Antibiotic |
Xanthone 是从山竹果中分离得到的,在癌变的不同阶段可控制细胞分裂和生长,凋亡,炎症和转移。Xanthone 具有抗氧化,抗肿瘤,抗过敏,抗炎,抗细菌,抗真菌和抗病毒活性。 | |||
M17871 | 1,5,8-Trihydroxy-3-methoxy-2-prenylxanthone | 1,5,8-Trihydroxy-3-methoxy-2-prenylxanthone | Xanthones |
1,5,8-Trihydroxy-3-methoxy-2-prenylxanthone | |||
M17872 | 1,7-Dihydroxy-3-methoxy-2-prenylxanthone | 1,7-Dihydroxy-3-methoxy-2-prenylxanthone | Xanthones |
1,7-Dihydroxy-3-methoxy-2-prenylxanthone | |||
M17873 | 1-Hydroxy-2,3,4,7-tetramethoxyxanthone | 1-Hydroxy-2,3,4,7-tetramethoxyxanthone | Xanthones |
1-Hydroxy-2,3,4,7-tetramethoxyxanthone | |||
M17874 | 3,6-Dihydroxy-1,2,7-trimethoxyxanthone | 3,6-二羟基-1,2,7-三甲氧基呫吨酮 | Xanthones |
3,6-Dihydroxy-1,2,7-trimethoxyxanthone 3,6-二羟基-1,2,7-三甲氧基呫吨酮 | |||
M17875 | 1,3,5,7-Tetrahydroxy-8-prenylxanthone | 1,3,5,7-Tetrahydroxy-8-prenylxanthone | Xanthones |
1,3,5,7-Tetrahydroxy-8-prenylxanthone | |||
M17876 | 1,7-Dihydroxy-2,3-dimethoxyxanthone | 1,7-二羟基-2,3-二甲氧基呫吨酮 | Xanthones |
1,7-Dihydroxy-2,3-dimethoxyxanthone 1,7-二羟基-2,3-二甲氧基呫吨酮 | |||
M17877 | 3,6-Dihydroxy-1,7-dimethoxyxanthone | 3,6-二羟基-1,7-二甲氧基呫吨酮 | Xanthones |
3,6-Dihydroxy-1,7-dimethoxyxanthone 3,6-二羟基-1,7-二甲氧基呫吨酮 | |||
M17878 | 1,5,6-Trihydroxy-3-methoxyxanthone | 1,5,6-三羟基-3-甲氧基呫吨酮 | Xanthones |
1,5,6-Trihydroxy-3-methoxyxanthone 1,5,6-三羟基-3-甲氧基呫吨酮 | |||
M17879 | 1,3,7-Trihydroxy-2-prenylxanthone | 1,3,7-Trihydroxy-2-prenylxanthone | Xanthones |
1,3,7-Trihydroxy-2-prenylxanthone | |||
M17880 | 1,7-Dihydroxy-4-methoxyxanthone | 1,7-二羟基-4-甲氧基呫吨酮 | Xanthones |
1,7-Dihydroxy-4-methoxyxanthone 1,7-二羟基-4-甲氧基呫吨酮 | |||
M17881 | 1,2,3,6,7-Pentamethoxyxanthone | 1,2,3,6,7-五甲氧基呫吨酮 | Xanthones |
1,2,3,6,7-Pentamethoxyxanthone 1,2,3,6,7-五甲氧基呫吨酮 | |||
M17882 | 1,2,3,7-Tetramethoxyxanthone | 1,2,3,7-四甲氧基呫吨酮 | Xanthones |
1,2,3,7-Tetramethoxyxanthone 1,2,3,7-四甲氧基呫吨酮 | |||
M17883 | 5-Hydroxy-1-methoxyxanthone | 5-羟基-1-甲氧基呫吨酮 | Xanthones |
5-Hydroxy-1-methoxyxanthone 5-羟基-1-甲氧基呫吨酮 | |||
M17884 | 1,5,6-Trihydroxyxanthone | 1,5,6-三羟基呫吨酮 | Xanthones |
1,5,6-Trihydroxyxanthone 1,5,6-三羟基呫吨酮 | |||
M17885 | 1,6,7-Trihydroxyxanthone | 1,6,7-三羟基呫吨酮 | Xanthones |
1,6,7-Trihydroxyxanthone 1,6,7-三羟基呫吨酮 | |||
M17886 | O-Demethylforbexanthone | O-Demethylforbexanthone | Xanthones |
O-Demethylforbexanthone | |||
M17888 | 1,5-Dihydroxyxanthone | 1,5-二羟基呫吨酮 | Xanthones |
1,5-Dihydroxyxanthone 1,5-二羟基呫吨酮 | |||
M17889 | 2,3-Dimethoxyxanthone | 2,3-二甲氧基呫吨酮 | Xanthones |
2,3-Dimethoxyxanthone 2,3-二甲氧基呫吨酮 | |||
M17890 | 1,7-Dimethoxyxanthone | 1,7-二甲氧基呫吨酮 | Xanthones |
1,7-Dimethoxyxanthone 1,7-二甲氧基呫吨酮 | |||
M17891 | Isocudraniaxanthone A | Isocudraniaxanthone A | Xanthones |
Isocudraniaxanthone A | |||
M17892 | Isogarciniaxanthone E | 异藤黄氧蒽酮 E | Xanthones |
Isogarciniaxanthone E 异藤黄氧蒽酮 E | |||
M17893 | Polygalaxanthone XI | 远志口山酮XI | Xanthones |
Polygalaxanthone XI 远志口山酮XI | |||
M17895 | Griffipavixanthone | Griffipavixanthone | Xanthones |
Griffipavixanthone | |||
M17896 | 2-Hydroxyxanthone | 2-羟基呫吨酮 | Xanthones |
2-Hydroxyxanthone 2-羟基呫吨酮 | |||
M17897 | 4-Hydroxyxanthone | 4-羟基呫吨酮 | Xanthones |
4-Hydroxyxanthone 4-羟基呫吨酮 | |||
M17900 | Dulcisxanthone B | Dulcisxanthone B | Xanthones |
Dulcisxanthone B | |||
M17901 | Assiguxanthone B | Assiguxanthone B | Xanthones |
Assiguxanthone B | |||
M4482 | Neomangiferin | 新芒果苷 | Others |
Neomangiferin,一种天然的 C-glucosyl xanthone,是从干燥的 Anemarrhena asphodeloides 的根茎中分离得到的。Neomangiferin 有效减轻大鼠高脂饮食诱导的非酒精性脂肪性肝病 (NAFLD)。 | |||
M4621 | Garcinone-C | 伽升沃C | ATM/ATR |
Garcinone C 是一种呫吨酮 (xanthone) 衍生物,是从长叶藤 (Garcinia oblongifolia Champ) 中提取的天然化合物。Garcinone C 刺激 ATR 和 4E-BP1 的表达水平,同时有效抑制细胞周期蛋白 B1,细胞周期蛋白 D1,细胞周期蛋白 E2,cdc2,Stat3 和 CDK7 的表达水平。 | |||
M10671 | Garcinone E | 伽升沃E | Apoptosis |
Garcinone-E | |||
Garcinone E is the most active xanthone from mangosteen, which has potent cytotoxic effect against hepatocellular carcinoma cell lines. Garcinone E might inhibit metastasis of an oral cancer cell line by blocking invasion, migration and MMP production. |
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