找到约 10 条 “Lidocaine” 相关结果 (用时 0.128 秒)
目录号 | 产品名称 | 中文名称 | 靶点 |
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M5741
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Lidocaine | 利多卡因 | Animal experimental anesthetics |
Alphacaine | |||
Lidocaine是一种选择性的,逆向外周组胺H1受体激动剂,IC50大于32 μM。Lidocaine (Lignocaine) 还抑制涉及复杂电压和依赖性的钠通道 (sodium channels)。 | |||
M5742
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Lidocaine HCl | 盐酸利多卡因 | Animal experimental anesthetics |
Lidocaine HCL, Lidothesin | |||
Lidocaine hydrochloride是一种局部麻醉剂及心脏抑制剂,被用作抗心律失常剂。 | |||
M7884 | Lidocaine N-ethyl chloride | Lidocaine N-ethyl chloride | Others |
Lidocaine N-ethyl chloride is an intracellular voltage-gated sodium channel blocker. | |||
M7892 | Lidocaine hydrochloride monohydrate | 盐酸利多卡因一水合物 | Animal experimental anesthetics |
Lidocaine hydrochloride monohydrate is an Na+ channel blocker; class IB antiarrhythmic that is rapidly absorbed after parenteral administration. | |||
M21430
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Lidocaine N-ethyl bromide | Lidocaine N-ethyl bromide | Animal experimental anesthetics |
QX-314 | |||
Lidocaine N-ethyl bromide(QX-314)是一种利多卡因衍生物,同时也是钠离子通道(Sodium Channel)阻断剂,可用于动物实验的局部麻醉。 | |||
M7180
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QX 314 bromide | QX 314 bromide | Sodium Channel |
QX-314 bromide | |||
QX 314 bromide是lidocaine的一种膜不渗透四元衍生物,同时也是电压激活 Na+通道(Sodium Channel)的阻断剂。此外,在细胞内 QX 314 还能抑制海马 CA1 锥体神经元的钙电流。 | |||
M8032 | Prilocaine hydrochloride | 盐酸丙胺卡因 | Animal experimental anesthetics |
Prilocaine hydrochloride is used for local nerve block and for spinal anesthesia; pharmacological properties are similar to those of lidocaine. | |||
M8226 | MEGX | MEGX | Others |
Monoethylglycinexylidide (MEGX) is an active metabolite of lidocaine. | |||
M49731 | Glycinexylidide | Glycinexylidide | MEK |
Glycinexylidide (GX) 是 Lidocaine 的活性代谢物。 | |||
M56949 | Carcainium chloride | Carcainium chloride | Others |
Carcainium chloride (QX 572) 是 Lidocaine 的四元衍生物。有镇咳作用。 |