找到约 4 条 “ET receptor antagonist 1” 相关结果 （用时 0.109 秒）
| 目录号 | 产品名称 | 中文名称 | 靶点 |
|---|---|---|---|
| M43590 | ET receptor antagonist 1 | ET receptor antagonist 1 | Estrogen Receptor |
| ET receptor antagonist 1 是一种 ET 受体拮抗剂 (IC50=0.18 nM)，可用于肺动脉高压 (PAH) 研究。 | |||
| M8700 | PCS1055 dihydrochloride | PCS1055 dihydrochloride | Others |
| PCS1055 is a potent and selective muscarinic M4 acetylcholine receptor competitive antagonist that exhibits >100-fold selectivity over M1-, M3-, and M5-receptors and 30-fold selectivity at the M2 receptor. | |||
M8764
|
MM11253 | MM11253 | RAR/RXR |
| SR11253 | |||
| MM11253 (SR11253) is a high-affinity RARγ-selective retinoid acid (RA) receptor antagonist (IC50 = 44 nM against ATRA for binding RARγ; IC50 =1 μM in case of RARα, RARβ, RXRα). | |||
| M20685 | Lerisetron | Lerisetron | 5-HT Receptor |
| F 0930, F 0930RS | |||
| Lerisetron is a 5-HT3 receptor antagonist with IC50 of 0.81μM. | |||
