找到约 32 条 “CH 275” 相关结果 (用时 0.217 秒)
目录号 | 产品名称 | 中文名称 | 靶点 |
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M3483
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Flavopiridol hydrochloride | 弗拉平度盐酸盐;盐酸阿伏西地 | CDK |
NSC 649890 HCl; Alvocidib hydrochloride; L86 8275 HCl; HMR-1275 HCl | |||
Flavopiridol HCl (Alvocidib HCl) 是一种 CDK 的广谱抑制剂,与 ATP 竞争性地抑制 CDK1,CDK2 和 CDK4 的活性,IC50 值分别为 30, 170, 100 nM。 | |||
M11578 | ChemBridge-4102756 | ChemBridge化合物-4102756 | Screening Compounds and Building Blocks |
(2-imidazo[2,1-b][1,3]thiazol-6-ylethyl)amine dihydrochloride (4102756) | |||
ChemBridge特有类药化合物/先导化合物-4102756,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M11581 | ChemBridge-5100275 | ChemBridge化合物-5100275 | Screening Compounds and Building Blocks |
pentacyclo[6.6.6.0~2,7~.0~9,14~.0~15,20~]icosa-2(7),4,9,11,13,15,17,19-octaene-3,6-dione (5100275) | |||
ChemBridge特有类药化合物/先导化合物-5100275,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M11586 | ChemBridge-5101275 | ChemBridge化合物-5101275 | Screening Compounds and Building Blocks |
3-(2,5-diethoxyphenyl)-1-(2-thienyl)-2-propen-1-one (5101275) | |||
ChemBridge特有类药化合物/先导化合物-5101275,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M11621 | ChemBridge-5112759 | ChemBridge化合物-5112759 | Screening Compounds and Building Blocks |
1-(2-furylmethylene)-6-methyl-4-thioxo-4,5-dihydrofuro[3,4-c]pyridin-3(1H)-one (5112759) | |||
ChemBridge特有类药化合物/先导化合物-5112759,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M11859 | ChemBridge-5227511 | ChemBridge化合物-5227511 | Screening Compounds and Building Blocks |
5,5-dimethyl-1,3-cyclohexanedione 1-[N-(4-methylphenyl)thiosemicarbazone] (5227511) | |||
ChemBridge特有类药化合物/先导化合物-5227511,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M11871 | ChemBridge-5232755 | ChemBridge化合物-5232755 | Screening Compounds and Building Blocks |
2-hydroxy-1-naphthaldehyde 1,3-benzothiazol-2-ylhydrazone (5232755) | |||
ChemBridge特有类药化合物/先导化合物-5232755,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M11951 | ChemBridge-5275107 | ChemBridge化合物-5275107 | Screening Compounds and Building Blocks |
ethyl 3-amino-6-(3-pyridinyl)thieno[2,3-b]pyridine-2-carboxylate (5275107) | |||
ChemBridge特有类药化合物/先导化合物-5275107,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M11952 | ChemBridge-5275805 | ChemBridge化合物-5275805 | Screening Compounds and Building Blocks |
2-[5-(4-bromobenzylidene)-4-oxo-2-thioxo-1,3-thiazolidin-3-yl]-3-methylbutanoic acid (5275805) | |||
ChemBridge特有类药化合物/先导化合物-5275805,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M12001 | ChemBridge-5327543 | ChemBridge化合物-5327543 | Screening Compounds and Building Blocks |
5-(1-naphthylmethylene)-2-thioxodihydro-4,6(1H,5H)-pyrimidinedione (5327543) | |||
ChemBridge特有类药化合物/先导化合物-5327543,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M12445 | ChemBridge-5927508 | ChemBridge化合物-5927508 | Screening Compounds and Building Blocks |
N,N'-bis(1,3-benzodioxol-5-ylmethyl)isophthalamide (5927508) | |||
ChemBridge特有类药化合物/先导化合物-5927508,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M12479 | ChemBridge-5977961 | ChemBridge化合物-5977961 | Screening Compounds and Building Blocks |
ethyl 2-{[(3-chlorophenoxy)acetyl]amino}-4,5-dimethyl-3-thiophenecarboxylate (5977961) | |||
ChemBridge特有类药化合物/先导化合物-5977961,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M12627 | ChemBridge-6227564 | ChemBridge化合物-6227564 | Screening Compounds and Building Blocks |
2-methoxy-4-[(4-oxo-2-thioxo-1,3-thiazolidin-5-ylidene)methyl]phenyl 2-nitrobenzenesulfonate (6227564) | |||
ChemBridge特有类药化合物/先导化合物-6227564,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M13091 | ChemBridge-7939275 | ChemBridge化合物-7939275 | Screening Compounds and Building Blocks |
5-chloro-7-{[4-(2-pyridinyl)-1-piperazinyl]methyl}-8-quinolinol (7939275) | |||
ChemBridge特有类药化合物/先导化合物-7939275,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M13183 | ChemBridge-9022755 | ChemBridge化合物-9022755 | Screening Compounds and Building Blocks |
6-(2-ethoxyphenyl)-3-(2-methyl-3-furyl)[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole (9022755) | |||
ChemBridge特有类药化合物/先导化合物-9022755,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M45427 | ChemBridge-5102751 | ChemBridge化合物-5102751 | Screening Compounds and Building Blocks |
4,4'-(1,2-ethenediylbis{[5-(benzoylamino)-2,1-phenylene]sulfonylimino})dibenzoic acid (5102751) | |||
ChemBridge特有类药化合物/先导化合物-5102751,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M45544 | ChemBridge-5315275 | ChemBridge化合物-5315275 | Screening Compounds and Building Blocks |
1,4-phenylenebis[(4-methoxy-1-naphthyl)methanone] (5315275) | |||
ChemBridge特有类药化合物/先导化合物-5315275,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M46107 | ChemBridge-7275454 | ChemBridge化合物-7275454 | Screening Compounds and Building Blocks |
N-[3-(aminocarbonyl)-6-propyl-4,5,6,7-tetrahydro-1-benzothien-2-yl]tetrahydro-2-furancarboxamide (7275454) | |||
ChemBridge特有类药化合物/先导化合物-7275454,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M46108 | ChemBridge-7275695 | ChemBridge化合物-7275695 | Screening Compounds and Building Blocks |
4-(5-chloro-2-hydroxyphenyl)-4-azatetracyclo[5.3.2.0~2,6~.0~8,10~]dodec-11-ene-3,5-dione (7275695) | |||
ChemBridge特有类药化合物/先导化合物-7275695,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M46135 | ChemBridge-7402751 | ChemBridge化合物-7402751 | Screening Compounds and Building Blocks |
ethyl 3-[(3-cyclohexylpropanoyl)amino]benzoate (7402751) | |||
ChemBridge特有类药化合物/先导化合物-7402751,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M46334 | ChemBridge-7832758 | ChemBridge化合物-7832758 | Screening Compounds and Building Blocks |
N-(4-sec-butylphenyl)-N'-(3,4-diethoxybenzyl)thiourea (7832758) | |||
ChemBridge特有类药化合物/先导化合物-7832758,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M46343 | ChemBridge-7842754 | ChemBridge化合物-7842754 | Screening Compounds and Building Blocks |
N-(4-sec-butylphenyl)-N'-[3-(1H-pyrazol-1-ylmethyl)phenyl]thiourea (7842754) | |||
ChemBridge特有类药化合物/先导化合物-7842754,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M46768 | ChemBridge-9012750 | ChemBridge化合物-9012750 | Screening Compounds and Building Blocks |
4-({[5-(2-furyl)-4-phenyl-4H-1,2,4-triazol-3-yl]thio}methyl)-1,3-thiazol-2-amine (9012750) | |||
ChemBridge特有类药化合物/先导化合物-9012750,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M46788 | ChemBridge-9027577 | ChemBridge化合物-9027577 | Screening Compounds and Building Blocks |
3-(1,3-benzodioxol-5-yl)-5-(4-methylphenyl)-1,2,4-oxadiazole (9027577) | |||
ChemBridge特有类药化合物/先导化合物-9027577,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M46808 | ChemBridge-9041275 | ChemBridge化合物-9041275 | Screening Compounds and Building Blocks |
N-(4-cyanophenyl)-1-(2-furoyl)piperidine-4-carboxamide (9041275) | |||
ChemBridge特有类药化合物/先导化合物-9041275,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M47129 | ChemBridge-9275388 | ChemBridge化合物-9275388 | Screening Compounds and Building Blocks |
7-(1,3-benzodioxol-5-yl)-3-(4-fluorophenyl)-2-methylpyrazolo[1,5-a]pyrido[3,4-e]pyrimidin-6(7H)-one (9275388) | |||
ChemBridge特有类药化合物/先导化合物-9275388,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M47400 | ChemBridge-15275036 | ChemBridge化合物-15275036 | Screening Compounds and Building Blocks |
3-[2-(4-fluorophenyl)morpholin-4-yl]propan-1-ol (15275036) | |||
ChemBridge特有类药化合物/先导化合物-15275036,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M47550 | ChemBridge-21275089 | ChemBridge化合物-21275089 | Screening Compounds and Building Blocks |
1-{5-[(4-cyclopentyl-1,4-diazepan-1-yl)carbonyl]-2-methylphenyl}-2-imidazolidinone (21275089) | |||
ChemBridge特有类药化合物/先导化合物-21275089,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M47551 | ChemBridge-21275538 | ChemBridge化合物-21275538 | Screening Compounds and Building Blocks |
3-{[4-(1,2,4-oxadiazol-3-yl)piperidin-1-yl]carbonyl}-4,5,6,7-tetrahydro-1H-indazole (21275538) | |||
ChemBridge特有类药化合物/先导化合物-21275538,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M47707 | ChemBridge-27529496 | ChemBridge化合物-27529496 | Screening Compounds and Building Blocks |
(3,5-dimethoxybenzyl)({1-[2-(3-fluorophenyl)ethyl]-4-piperidinyl}methyl)methylamine (27529496) | |||
ChemBridge特有类药化合物/先导化合物-27529496,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M1942
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Alectinib | 艾乐替尼;阿来替尼 | ALK |
CH5424802; AF802 | |||
Alectinib (CH5424802) 是一种有效的ALK抑制剂,IC50为1.9 nM,对L1196M突变型敏感。Alectinib (CH5424802) 还抑制 ALK F1174L 和 ALK R1275Q,其 IC50 分别为 1 nM 和 3.5 nM。Alectinib 还具有有效的中枢神经系统 (CNS) 渗透能力。 | |||
M47708 | ChemBridge-27540064 | ChemBridge化合物-27540064 | Screening Compounds and Building Blocks |
trans-N-[2-(4-chlorophenyl)ethyl]-3-hydroxy-N-(pyridin-3-ylmethyl)cyclohexanecarboxamide (27540064) | |||
ChemBridge特有类药化合物/先导化合物-27540064,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 |