找到约 13 条 “66-84-2” 相关结果 （用时 0.112 秒）
| 目录号 | 产品名称 | 中文名称 | 靶点 |
|---|---|---|---|
M2807
|
LDN-57444 | LDN-57444 | Deubiquitinase |
| LDN-57444是一种可逆的竞争性的蛋白酶体抑制剂，抑制UCch-L1时，IC50为0.88 μM，比作用于亚型Uch-L3选择性高30倍。 | |||
| M3280
|
Clopidogrel | 氯吡格雷 | P2 Receptor |
| SR-25990C; Clopidogrelum | |||
| Clopidogrel是一种具有口服活性的P2Y12受体阻断剂。Clopidogrel 可降低血小板聚集，用于抑制冠状动脉、周围血管和脑血管中的血凝块。 | |||
| M6292
|
Ansamitocin P 3 | 安丝菌素P-3 | Microtubule |
| Antibiotic C 15003P3; Maytansinol butyrate | |||
| Ansamitocin P-3是一种微管抑制剂，也是一种大环抗肿瘤抗生素。 | |||
| M14086
|
Glucosamine hydrochloride | 盐酸氨基葡萄糖 | Metabolite/Endogenous Metabolite |
| D-(+)-Glucosamine hydrochloride; Chitosamine hydrochloride | |||
| Glucosamine hydrochloride (D-Glucosamine hydrochloride) 是一种氨基糖, 是糖基化蛋白和脂质生化合成的突出前体, 用作膳食补充剂。Glucosamine hydrochloride也是软骨基质和滑液中糖胺聚糖的天然成分，当外用时，对骨关节炎软骨和软骨细胞具有药理作用。 | |||
| M20730
|
KGA-2727 | KGA-2727 | SGLT |
| KGA-2727 is a potent, selective, high-affinity inhibitor of sodium glucose cotransporter 1 (SGLT1) with Ki of 97.4 nM and 43.5 nM for human SGLT1 and rat SGLT1, respectively. The selectivity ratios (Ki for SGLT2/Ki for SGLT1) of KGA-2727 are 140 (human) and 390 (rat). KGA-2727 exhibits antidiabetic efficacy in rodent models. | |||
| M21293 | BCPyr | BCPyr | BTK |
| BCPyr 是一种新的候选 BTK 降解剂 （DC50 = 800 nM）。 | |||
| M30749 | UCK2 Inhibitor-2 | UCK2 Inhibitor-2 | Dehydrogenase |
| UCK2 Inhibitor-2 是一种非竞争性尿苷胞苷激酶 2 (UCK2) 抑制剂，IC50 值为 3.8 µM。UCK2 Inhibitor-2 可以抑制细胞中尿苷的回收。 | |||
| M48662 | ChemBridge-66846217 | ChemBridge化合物-66846217 | Screening Compounds and Building Blocks |
| 1'-(4-fluorobenzyl)-4,5-dihydro-2H-spiro[cyclopenta[c]pyrazole-6,3'-piperidine] (66846217) | |||
| ChemBridge特有类药化合物/先导化合物-66846217，由AbMole（奥默生物）独家提供。具体售价货期请咨询AbMole（奥默生物）。运费额外计算。 | |||
| M51669 | Cys-Arg-Gly-Asp-Phe-Pro-Ala-Ser-Ser-Cys (Disulfide bridge:cys1-cys10) | Cys-Arg-Gly-Asp-Phe-Pro-Ala-Ser-Ser-Cys (Disulfide bridge:cys1-cys10) | Others |
| Cys-Arg-Gly-Asp-Phe-Pro-Ala-Ser-Ser-Cys (Disulfide bridge:cys1-cys10)，一种含有环状 RGD 活性序列的十肽，是整合素 (Integrin) αIIbβ3 拮抗剂，可抑制血小板和 proMMP-13 的粘附。 | |||
| M51940 | Z-D-Lys(Boc)-OH | Z-D-Lys(Boc)-OH | Amino Acid Derivatives |
| Z-D-Lys(Boc)-OH 是一种赖氨酸衍生物。 | |||
| M7057 | NSC 663284 | NSC 663284 | Others |
| DA-3003-1 | |||
| NSC 663284是一种有效的、选择性的Cdc25磷酸酶抑制剂。 | |||
| M20715 | CS-2660 (JNJ-38158471) | CS-2660 (JNJ-38158471) | VEGFR/PDGFR |
| CS-2660 (JNJ-38158471) is a well tolerated, orally available, highly selective VEGFR-2 inhibitor with IC50 of 40 nM. CS-2660 (JNJ-38158471) also inhibits closely related tyrosine kinases such as Ret and Kit with IC50 of 180 nM and 500 nM，while it has no significant activity (>1 microM) against VEGFR-1 and VEGFR-3. | |||
| M52945 | CR 665 | CR 665 | Opioid Receptor |
| CR 665 (JNJ 38488502) 是一种外周选择性κ-阿片类激动剂。 | |||
