找到约 7 条 “Thyroid Hormone Receptor” 相关结果 (用时 0.219 秒)
目录号 | 产品名称 | 中文名称 | 靶点 |
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M40874
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Recombinant Human PTH1R (HEK293, C-6His) | 重组人PTH1R (HEK293, C-6His) | Cytokines and Growth Factors |
Parathyroid Hormone 1 Receptor | |||
Parathyroid hormone 1 receptor (PTH1R) is a protein that in humans is encoded by the PTH1R gene, it belongs to the G-protein coupled receptor 2 family. PTH1R functions as a receptor for parathyroid hormone (PTH) and for parathyroid hormone-related protein (PTHrP). | |||
M43608 | Thyroid hormone receptor beta agonist-1 | Thyroid hormone receptor beta agonist-1 | Thyroid Hormone Receptor |
Thyroid hormone receptor beta agonist-1 是thyroid beta 的激动剂。 | |||
M58468
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Thyroid hormone receptor antagonist (1-850) | Thyroid hormone receptor antagonist (1-850) | Thyroid Hormone Receptor |
THR antagonist 1-850 | |||
Thyroid hormone receptor antagonist (1-850) 是一种竞争性、选择性、高亲和力的甲状腺激素受体 (TR) 拮抗剂,拮抗 T3 对 TR 的影响的 IC50 为 1.5 μM。 | |||
M5828
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Octinoxate | 对甲氧基肉桂酸辛酯 | Thyroid Hormone Receptor |
2-Ethylhexyl 4-methoxycinnamate; Octyl methoxycinnamate | |||
Octinoxate(对甲氧基肉桂酸辛酯)是一种紫外线过滤剂和甲状腺激素受体(thyroid hormone receptor)的激动剂。Octinoxate 还可以抑制 CYP1A1 和 CYP1B1,IC50值分别约为1 µM和586 nM,并以依赖于 PI3K 通路的方式调节角质形成细胞中的透明质酸代谢。 | |||
M8278 | MLS000389544 | MLS000389544 | Others |
MLS000389544 is a selective and potent methylsulfonylnitrobenzoa |
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M14798 | TR antagonist 1 | TR antagonist 1 | Others |
TR antagonist 1是高亲和力的甲状腺激素受体 (thyroid hormone receptor (TR)) 拮抗剂,对 TRα 和 TRβ 的IC50 值分别为 36 和 22 nM。 | |||
M57253 | 3,5-Diiodothyropropionic acid | 3,5-Diiodothyropropionic acid | Thyroid Hormone Receptor |
3,5-Diiodothyropropionic acid 是甲状腺激素类似物,可诱导 α-肌球蛋白重链 mRNA 表达,与甲状腺激素受体 (thyroid hormone receptors (TR)) 结合,对 TRα1 和 TRβ1 的 Ka 值分别为 2.40 和 4.06 M-1。 |