找到约 7 条 “TR antagonist 1” 相关结果 （用时 0.15 秒）
| 目录号 | 产品名称 | 中文名称 | 靶点 |
|---|---|---|---|
| M14798 | TR antagonist 1 | TR antagonist 1 | Others |
| TR antagonist 1是高亲和力的甲状腺激素受体 (thyroid hormone receptor (TR)) 拮抗剂，对 TRα 和 TRβ 的IC50 值分别为 36 和 22 nM。 | |||
| M8611 | Ex26 | Ex26 | S1P Receptor |
| Ex26 is a peripherally-restricted biphenylcarboxamide derivative that acts as a highly potent and subtype-selective S1P1 antagonist (IC50 = 0.93 nM against S1PR1 and >3.1 μM against S1PR2/3/4/5). | |||
M9569
|
Etrumadenant | 伊曲地南 | Adenosine Receptor |
| AB928; A2aR/A2bR antagonist-1 | |||
| Etrumadenant（AB928，A2aR/A2bR antagonist-1）是一种口服生物可利用的，选择性的A2aR和A2bR腺苷受体的双重拮抗剂，具有免疫调节活性和抗肿瘤活性。 | |||
| M20639 | H3B-5942 | H3B-5942 | Estrogen Receptor |
| H3B-5942 is a selective and irreversible estrogen receptor covalent antagonist, inactivates both ERα WT and ERα mutation. The Ki values are 1 nM and 0.41 nM, respectively. | |||
| M20685 | Lerisetron | Lerisetron | 5-HT Receptor |
| F 0930, F 0930RS | |||
| Lerisetron is a 5-HT3 receptor antagonist with IC50 of 0.81μM. | |||
| M43594 | Estrogen receptor antagonist 8 | Estrogen receptor antagonist 8 | Estrogen Receptor |
| Estrogen receptor antagonist 8 是一种有效的雌激素受体 ER 拮抗剂，其EC50为4.160 μM。 | |||
| M58323
|
MK-2295 | MK-2295 | TRP Channel |
| TRPV1 antagonist 5 | |||
| MK-2295 (TRPV1 antagonist 5) 是一种有效的 TRPV1 拮抗剂。MK-2295 可用于慢性疼痛的研究。 | |||
