找到约 37 条 “Pyrazole” 相关结果 (用时 0.088 秒)

目录号 产品名称 中文名称 靶点
M4834 Propyl pyrazole triol (PPT) Propyl pyrazole triol (PPT) Estrogen Receptor
propyl pyrazole triol
PPT是一种有效的亚型选择性雌激素受体 α (ERα) 激动剂,具有EC50 ~ 200 pM,对ERα的选择性比ERβ高410倍。
M5663 Fomepizole 4-甲基吡唑 Dehydrogenase
4-methylpyrazole, Antizol, Antizol-Vet
Fomepizole是一种竞争性乙醇脱氢酶抑制剂。
M9967 Methylpiperidino pyrazole 甲基哌啶基吡唑 Estrogen Receptor
MPP
Methyl-piperidino-pyrazole(MPP)是一种特异性雌激素受体 α拮抗剂。
M11565 ChemBridge-4004729 ChemBridge化合物-4004729 Screening Compounds and Building Blocks
3-phenyl-1H-pyrazole-4-carboxylic acid (4004729)
ChemBridge特有类药化合物/先导化合物-4004729,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M11567 ChemBridge-4012182 ChemBridge化合物-4012182 Screening Compounds and Building Blocks
3-(3-fluorophenyl)-1H-pyrazole-4-carboxylic acid (4012182)
ChemBridge特有类药化合物/先导化合物-4012182,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M11606 ChemBridge-5107414 ChemBridge化合物-5107414 Screening Compounds and Building Blocks
5-ethoxy-1-(4-nitrophenyl)-3-phenyl-4,5-dihydro-1H-pyrazole (5107414)
ChemBridge特有类药化合物/先导化合物-5107414,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M11776 ChemBridge-5175423 ChemBridge化合物-5175423 Screening Compounds and Building Blocks
5-amino-1-phenyl-1H-pyrazole-4-carboxylic acid (5175423)
ChemBridge特有类药化合物/先导化合物-5175423,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M11851 ChemBridge-5223191 ChemBridge化合物-5223191 Screening Compounds and Building Blocks
1-methyl-N-{2-methyl-4-[(2-methylphenyl)diazenyl]phenyl}-1H-pyrazole-5-carboxamide (5223191)
ChemBridge特有类药化合物/先导化合物-5223191,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M11968 ChemBridge-5304192 ChemBridge化合物-5304192 Screening Compounds and Building Blocks
5-methyl-4-{[(4-nitrophenyl)amino]methylene}-2-phenyl-2,4-dihydro-3H-pyrazole-3-thione (5304192)
ChemBridge特有类药化合物/先导化合物-5304192,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M11984 ChemBridge-5314457 ChemBridge化合物-5314457 Screening Compounds and Building Blocks
3-phenyl-1H-pyrazole-5-carbohydrazide (5314457)
ChemBridge特有类药化合物/先导化合物-5314457,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M12243 ChemBridge-5662148 ChemBridge化合物-5662148 Screening Compounds and Building Blocks
5-amino-3-{2-[2-[(4-chlorobenzyl)oxy]-4-(diethylamino)phenyl]-1-cyanovinyl}-1-phenyl-1H-pyrazole-4-carbonitrile (5662148)
ChemBridge特有类药化合物/先导化合物-5662148,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M12254 ChemBridge-5669313 ChemBridge化合物-5669313 Screening Compounds and Building Blocks
5-amino-3-[2-(5-bromo-2-isopropoxyphenyl)-1-cyanovinyl]-1-phenyl-1H-pyrazole-4-carbonitrile (5669313)
ChemBridge特有类药化合物/先导化合物-5669313,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M12352 ChemBridge-5784220 ChemBridge化合物-5784220 Screening Compounds and Building Blocks
N'-[(2-hydroxy-1-naphthyl)methylene]-3-(2-naphthyl)-1H-pyrazole-5-carbohydrazide (5784220)
ChemBridge特有类药化合物/先导化合物-5784220,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M12367 ChemBridge-5793851 ChemBridge化合物-5793851 Screening Compounds and Building Blocks
6-amino-4-(2-hydroxy-5-nitrophenyl)-3-methyl-1,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile (5793851)
ChemBridge特有类药化合物/先导化合物-5793851,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M12462 ChemBridge-5947495 ChemBridge化合物-5947495 Screening Compounds and Building Blocks
N-(5-chloro-2-methoxyphenyl)-3-methyl-1-phenyl-1H-thieno[2,3-c]pyrazole-5-carboxamide (5947495)
ChemBridge特有类药化合物/先导化合物-5947495,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M12695 ChemBridge-6513926 ChemBridge化合物-6513926 Screening Compounds and Building Blocks
3-(4-methoxyphenyl)-N,1-diphenyl-1H-pyrazole-4-carboxamide (6513926)
ChemBridge特有类药化合物/先导化合物-6513926,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M12964 ChemBridge-7685300 ChemBridge化合物-7685300 Screening Compounds and Building Blocks
6-amino-1-(3-bromo-2-chloro-4-hydroxy-5-methoxyphenyl)-3-methyl-4-phenyl-1,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile (7685300)
ChemBridge特有类药化合物/先导化合物-7685300,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M13009 ChemBridge-7805127 ChemBridge化合物-7805127 Screening Compounds and Building Blocks
4-({[(5-chloro-2-methoxyphenyl)amino]carbonothioyl}amino)-1-ethyl-1H-pyrazole-3-carboxamide (7805127)
ChemBridge特有类药化合物/先导化合物-7805127,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M13079 ChemBridge-7932356 ChemBridge化合物-7932356 Screening Compounds and Building Blocks
5-amino-3-{2-[3-(4-chlorophenyl)-1H-pyrazol-4-yl]-1-cyanovinyl}-1-(2-hydroxyethyl)-1H-pyrazole-4-carbonitrile (7932356)
ChemBridge特有类药化合物/先导化合物-7932356,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M13101 ChemBridge-7953989 ChemBridge化合物-7953989 Screening Compounds and Building Blocks
1-(2,4-dichlorobenzyl)-1H-pyrazole-3,5-dicarboxylic acid (7953989)
ChemBridge特有类药化合物/先导化合物-7953989,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M13149 ChemBridge-7998757 ChemBridge化合物-7998757 Screening Compounds and Building Blocks
1-(4-bromobenzyl)-1H-pyrazole-3,5-dicarboxylic acid (7998757)
ChemBridge特有类药化合物/先导化合物-7998757,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M13166 ChemBridge-9000194 ChemBridge化合物-9000194 Screening Compounds and Building Blocks
1-(2-chlorobenzyl)-1H-pyrazole-3,5-dicarboxylic acid (9000194)
ChemBridge特有类药化合物/先导化合物-9000194,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M13172 ChemBridge-9002906 ChemBridge化合物-9002906 Screening Compounds and Building Blocks
1-(4-fluorobenzyl)-1H-pyrazole-3,5-dicarboxylic acid (9002906)
ChemBridge特有类药化合物/先导化合物-9002906,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M13271 ChemBridge-34521546 ChemBridge化合物-34521546 Screening Compounds and Building Blocks
N-{[1-(2,3-dihydro-1H-inden-2-yl)-3-piperidinyl]methyl}-N-(2-methoxyethyl)-1,4,5,6-tetrahydrocyclopenta[c]pyrazole-3-carboxamide (34521546)
ChemBridge特有类药化合物/先导化合物-34521546,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M18001 1H-Pyrazole-1-carboxamidine hydrochloride 1H-吡唑-1-甲脒盐酸盐 Others
1H-Pyrazole-1-carboximidamide hydrochloride 是一种生化试剂,可作为生物材料或有机化合物,用于生命科学相关研究。
M20460 3-Methylpyrazole 3-Methylpyrazole Dehydrogenase
3-MP
3-Methylpyrazole (3-MP) is a weak or non-inhibitor of alcohol dehydrogenase.
M20476 Fipronil Fipronil Anti-infection
Fluocyanobenpyrazole, Termidor
Fipronil is a recalcitrant phenylpyrazole-based pesticide used for flea/tick treatment and termite control that is distributed in urban aquatic environments via stormwater and contributes to stream toxicity.
M20487 AS057278 AS057278 Others
3-Methylpyrazole-5-carboxylic acid
AS057278 (3-Methylpyrazole-5-carboxylic acid, MPC) is an inhibitor of D-amino acid oxidase (DAAO).
M38865 N,N'-Di-Boc-1H-pyrazole-1-carboximidamide N,N'-Di-Boc-1H-pyrazole-1-carboximidamide Others
N,N'-Di-Boc-1H-pyrazole-1-carboximidamide 是一种生化试剂,可作为生物材料或有机化合物,用于生命科学相关研究。
M45409 ChemBridge-4004174 ChemBridge化合物-4004174 Screening Compounds and Building Blocks
3-isobutyl-1-methyl-1H-pyrazole-5-carboxylic acid (4004174)
ChemBridge特有类药化合物/先导化合物-4004174,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M14634 MPP dihydrochloride MPP dihydrochloride Estrogen Receptor
MPP Dihydrochloride(Methylpiperidino Pyrazole Dihydrochloride)是一种强效且选择性的雌激素受体(ER)调节剂。MPP Dihydrochloride可降低雌激素受体α(ERα)的磷酸化水平,但不影响Akt的磷酸化。MPP Dihydrochloride可用于抗肿瘤研究,它在RL95-2子宫内膜癌细胞中表现出显著的抗增殖活性,IC50值为20.01 μM。此外,MPP Dihydrochloride还能够逆转β-雌二醇的正向效应。
M55926 Phthalazinone pyrazole  Phthalazinone pyrazole  Aurora Kinase
Phthalazinone pyrazole 是一种有效的、选择性的、具有口服活性的 Aurora-A 激酶抑制剂,其 IC50 值为 0.031 μM。Phthalazinone pyrazole 可以阻止有丝分裂并随后通过增殖细胞的凋亡抑制肿瘤生长。
M57405 1,3-dimethyl-1H-pyrazole-4-sulfonamide 1,3-dimethyl-1H-pyrazole-4-sulfonamide Others
1,3-dimethyl-1H-pyrazole-4-sulfonamide
M57581 5-AMINO-1-(4-BROMO-PHENYL)-1H-PYRAZOLE-4-CARBOXYLIC ACID 5-AMINO-1-(4-BROMO-PHENYL)-1H-PYRAZOLE-4-CARBOXYLIC ACID Others
5-AMINO-1-(4-BROMO-PHENYL)-1H-PYRAZOLE-4-CARBOXYLIC ACID
M57801 1,4,5,6-Tetrahydro-1-phenyl-3-cyclopentapyrazoleacetic acid 1,4,5,6-Tetrahydro-1-phenyl-3-cyclopentapyrazoleacetic acid Others
1,4,5,6-Tetrahydro-1-phenyl-3-cyclopentapyrazoleacetic acid
M57944 tert-butyl 3-oxo-2,3-dihydro-1H-pyrazole-1-carboxylate tert-butyl 3-oxo-2,3-dihydro-1H-pyrazole-1-carboxylate Others
tert-butyl 3-oxo-2,3-dihydro-1H-pyrazole-1-carboxylate
M58316 Pyrazole 吡唑 Metabolite/Endogenous Metabolite
1H-pyrazole
Pyrazole 是一种内源性代谢产物。具有抗菌、抗病毒、抗肿瘤、抗炎等多种活性。








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