找到约 5 条 “Phosphatase-IN-1” 相关结果 (用时 0.301 秒)
目录号 | 产品名称 | 中文名称 | 靶点 |
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M9403
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TPI-1 | TPI-1 | Phosphatase |
Tyrosine Phosphatase Inhibitor 1 | |||
TPI-1是一种SHP-1的抑制剂,它抑制重组SHP-1的IC50值为40 nM。 | |||
M42551 | Phosphatase-IN-1 | Phosphatase-IN-1 | Phosphatase |
Phosphatase-IN-1 是一种 propranolol 衍生物,是一种磷脂酸磷酸酶 (Pah) 抑制剂。 | |||
M20719
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Raphin1 acetate | Raphin1 acetate | Phosphatase |
Raphin1 acetate is an orally bioavailable, selective inhibitor of the regulatory phosphatase PPP1R15B (R15B). Raphin1 acetate binds strongly to the R15B-PP1c holophosphatase with Kd of 0.033 μM. | |||
M20734 | (E/Z)-BCI | (E/Z)-BCI | Phosphatase |
BCI, NSC 150117 | |||
(E/Z)-BCI (BCI, NSC 150117) is an inhibitor of dual specific phosphatase 1/6 (DUSP1/DUSP6) and mitogen-activated protein kinase with EC50 of 13.3 μM and 8.0 μM for DUSP6 and DUSP1 in cells, respectively. (E)-BCI induces apoptosis via generation of reactive oxygen species (ROS) and activation of intrinsic mitochondrial pathway in H1299 lung cancer cells. | |||
M56742 | PPM1A-IN-1 | PPM1A-IN-1 | Phosphatase |
PPM1A-IN-1 是 PP2C Ser/Thr 磷酸酶 protein phosphatase Mg2+/Mn2+-dependent 1A 的抑制剂。PPM1A-IN-1 对 Mycobacterium tuberculosis 发挥抑菌活性。 |