找到约 5 条 “Phosphatase-IN-1” 相关结果 (用时 0.301 秒)

目录号 产品名称 中文名称 靶点
M9403 TPI-1 TPI-1 Phosphatase
Tyrosine Phosphatase Inhibitor 1
TPI-1是一种SHP-1的抑制剂,它抑制重组SHP-1的IC50值为40 nM。
M42551 Phosphatase-IN-1 Phosphatase-IN-1 Phosphatase
Phosphatase-IN-1 是一种 propranolol 衍生物,是一种磷脂酸磷酸酶 (Pah) 抑制剂。
M20719 Raphin1 acetate Raphin1 acetate Phosphatase
Raphin1 acetate is an orally bioavailable, selective inhibitor of the regulatory phosphatase PPP1R15B (R15B). Raphin1 acetate binds strongly to the R15B-PP1c holophosphatase with Kd of 0.033 μM.
M20734 (E/Z)-BCI (E/Z)-BCI Phosphatase
BCI, NSC 150117
(E/Z)-BCI (BCI, NSC 150117) is an inhibitor of dual specific phosphatase 1/6 (DUSP1/DUSP6) and mitogen-activated protein kinase with EC50 of 13.3 μM and 8.0 μM for DUSP6 and DUSP1 in cells, respectively. (E)-BCI induces apoptosis via generation of reactive oxygen species (ROS) and activation of intrinsic mitochondrial pathway in H1299 lung cancer cells.
M56742 PPM1A-IN-1  PPM1A-IN-1  Phosphatase
PPM1A-IN-1 是 PP2C Ser/Thr 磷酸酶 protein phosphatase Mg2+/Mn2+-dependent 1A 的抑制剂。PPM1A-IN-1 对 Mycobacterium tuberculosis 发挥抑菌活性。








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