找到约 10 条 “Paclitaxel C” 相关结果 (用时 0.105 秒)
目录号 | 产品名称 | 中文名称 | 靶点 |
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M5039
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10-Deacetyl-7-xylosyl paclitaxel | 10-Deacetyl-7-xylosyl paclitaxel | Microtubule |
10-Deacetyl-7-xylosyltaxol; 10-Deacetylpaclitaxel 7-Xyloside; 10-Deacetyltaxol 7-Xyloside | |||
10-去乙酰-7-木糖基紫杉醇是一种紫杉醇衍生物,具有改善的药理特性和更高的水溶性。 | |||
M39809 | Paclitaxel C | Paclitaxel C | Others |
Paclitaxel C 是一种可以在 taxus cutting 中分离得到的化合物。 | |||
M1970
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Paclitaxel | 紫杉醇 | Microtubule |
Taxol; NSC 125973 | |||
Paclitaxel是一种来源于植物红豆杉屈树皮的二萜类化合物,同时也是微管(Microtubule)聚合物稳定剂,能促进微管蛋白聚合抑制解聚,保持微管蛋白稳定,抑制细胞有丝分裂,作用于人内皮细胞,IC50为0.1 pM。 | |||
M8493
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NSC756093 | NSC756093 | Others |
NSC756093, a podophyllotoxin analog, is a potent and specific inhibitor of GBP1:PIM1 interaction that inhibits proliferation of paclitaxel resistant cancer cells. | |||
M8641 | LP117 | LP117 | Others |
LP117 is a pirinixic acid derivative that interferes with ATP-binding cassette (ABC) transporter ABCB1-mediated substrates transport, including vincristine, vinorelbine, paclitaxel, and actinomycin D, but not doxorubicin, rhodamine 123, or JC-1. | |||
M18304 | 7-Epi-10-deacetyl-taxol | 7-表-10-去乙酰基紫杉醇 | Others |
7-Epi 10-desacetyl paclitaxel (7-epi-10-deacetyltaxol) 是一种紫杉醇衍生物,对 HeLa 细胞具有细胞毒性,其 IC50 值为 85 μM。 | |||
M20888 | Epothilone A | Epothilone A | Microtubule |
Epothilone A is a paclitaxel-like microtubule-stabilizing agent with EC0.01 of 2 μM. | |||
M25241
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Bavituximab | Bavituximab | Others |
Anti-Human Phosphatidylserine Recombinant Antibody | |||
Bavituximab (Anti-Human Phosphatidylserine Recombinant Antibody) 是一种磷脂酰丝氨酸 (PS) 靶向的单克隆抗体,能够作用肿瘤血管系统和重新激活抗肿瘤免疫来抑制肿瘤生长。Bavituximab 联合Paclitaxel 和 Carboplatin ,对非小细胞肺癌的抑制有加强效果。 | |||
M40134 | 7-Xylosyl-10-Deacetyltaxol C | 7-Xylosyl-10-Deacetyltaxol C | Others |
7-Xylosyl-10-Deacetyltaxol C (7-Xylosyl-10-Deacetylpaclitaxel C) 是一种来源于 T. cuspidate 的紫杉醇衍生物,具有抗肿瘤活性,可以抑制 S180 肉瘤的生长。 | |||
M40201 | 7-Xylosyl-10-Deacetyltaxol B | 7-Xylosyl-10-Deacetyltaxol B | Others |
7-Xylosyl-10-Deacetyltaxol B (7-xylosyl-10-Deacetylpaclitaxel B) 是一种来源于T. cuspidate 的紫杉醇衍生物,具有抗肿瘤活性,可以抑制 S180 肉瘤的生长。 |