找到约 36 条 “PY-60” 相关结果 (用时 0.136 秒)

目录号 产品名称 中文名称 靶点
M5366 4-Aminoantipyrine 4-Aminoantipyrine COX
Ampyrone, NSC 60242
4-Aminoantipyrine(Ampyrone)是aminopyrine的代谢产物,具有镇痛、消炎退热的效果。Ampyrone刺激肝微粒体,用来测定胞外液。
M11870 ChemBridge-5231609 ChemBridge化合物-5231609 Screening Compounds and Building Blocks
2-[(3-cyano-5-ethyl-4,6-dimethyl-2-pyridinyl)thio]acetamide (5231609)
ChemBridge特有类药化合物/先导化合物-5231609,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M11904 ChemBridge-5244606 ChemBridge化合物-5244606 Screening Compounds and Building Blocks
(4-bromophenyl)(4-pyridinyl)methanone (5244606)
ChemBridge特有类药化合物/先导化合物-5244606,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M11931 ChemBridge-5260504 ChemBridge化合物-5260504 Screening Compounds and Building Blocks
1-(4-biphenylylmethyl)-4-(2-pyridinyl)piperazine (5260504)
ChemBridge特有类药化合物/先导化合物-5260504,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M12178 ChemBridge-5603529 ChemBridge化合物-5603529 Screening Compounds and Building Blocks
4-methoxybenzyl 6-methyl-2-oxo-4-phenyl-1,2,3,4-tetrahydro-5-pyrimidinecarboxylate (5603529)
ChemBridge特有类药化合物/先导化合物-5603529,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M12248 ChemBridge-5666005 ChemBridge化合物-5666005 Screening Compounds and Building Blocks
ethyl 5-(1,3-benzodioxol-5-yl)-2-(4-hydroxybenzylidene)-7-methyl-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate (5666005)
ChemBridge特有类药化合物/先导化合物-5666005,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M12335 ChemBridge-5761460 ChemBridge化合物-5761460 Screening Compounds and Building Blocks
methyl 4-{2,5-dioxo-3-[4-(2-pyrimidinyl)-1-piperazinyl]-1-pyrrolidinyl}benzoate (5761460)
ChemBridge特有类药化合物/先导化合物-5761460,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M12351 ChemBridge-5782601 ChemBridge化合物-5782601 Screening Compounds and Building Blocks
1-cyclohexyl-2-(2,6-difluorobenzyl)octahydropyrrolo[1,2-a]pyrazine (5782601)
ChemBridge特有类药化合物/先导化合物-5782601,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M12426 ChemBridge-5906014 ChemBridge化合物-5906014 Screening Compounds and Building Blocks
3-[5-(4-methylphenyl)-1,2,4-oxadiazol-3-yl]pyridine (5906014)
ChemBridge特有类药化合物/先导化合物-5906014,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M12456 ChemBridge-5935603 ChemBridge化合物-5935603 Screening Compounds and Building Blocks
N'-[4-(2,7-dimethylimidazo[1,2-a]pyridin-3-yl)-1,3-thiazol-2-yl]-N,N-dimethyl-1,4-benzenediamine hydrobromide (5935603)
ChemBridge特有类药化合物/先导化合物-5935603,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M12504 ChemBridge-6007262 ChemBridge化合物-6007262 Screening Compounds and Building Blocks
2-[(2,5-dimethyl-1-phenyl-1H-pyrrol-3-yl)methylene][1,3]thiazolo[3,2-a]benzimidazol-3(2H)-one (6007262)
ChemBridge特有类药化合物/先导化合物-6007262,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M12507 ChemBridge-6017246 ChemBridge化合物-6017246 Screening Compounds and Building Blocks
3-{5-[(2-amino-3,7-dicyano-4,6-dimethyl-5H-cyclopenta[b]pyridin-5-ylidene)methyl]-2-furyl}benzoic acid (6017246)
ChemBridge特有类药化合物/先导化合物-6017246,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M12512 ChemBridge-6026920 ChemBridge化合物-6026920 Screening Compounds and Building Blocks
3-(benzyloxy)-N-(4-chloro-3-[1,3]oxazolo[4,5-b]pyridin-2-ylphenyl)benzamide (6026920)
ChemBridge特有类药化合物/先导化合物-6026920,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M12513 ChemBridge-6027864 ChemBridge化合物-6027864 Screening Compounds and Building Blocks
2-(4-chloro-3,5-dimethylphenoxy)-N-(4-methyl-2-pyridinyl)acetamide (6027864)
ChemBridge特有类药化合物/先导化合物-6027864,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M12515 ChemBridge-6035242 ChemBridge化合物-6035242 Screening Compounds and Building Blocks
2-amino-6-{[2-(3,4-dihydroxyphenyl)-2-oxoethyl]thio}-4-(4-hydroxyphenyl)-3,5-pyridinedicarbonitrile (6035242)
ChemBridge特有类药化合物/先导化合物-6035242,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M12522 ChemBridge-6043266 ChemBridge化合物-6043266 Screening Compounds and Building Blocks
3-(3-methyl-4-{[5-(4-nitrophenyl)-2-furyl]methylene}-5-oxo-4,5-dihydro-1H-pyrazol-1-yl)benzoic acid (6043266)
ChemBridge特有类药化合物/先导化合物-6043266,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M12536 ChemBridge-6047396 ChemBridge化合物-6047396 Screening Compounds and Building Blocks
3-(5-bromo-2-pyridinyl)-2-(3-pyridinyl)-4(3H)-quinazolinone (6047396)
ChemBridge特有类药化合物/先导化合物-6047396,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M12537 ChemBridge-6048069 ChemBridge化合物-6048069 Screening Compounds and Building Blocks
15-carboxy-13-isopropylatis-13-ene-17,18-dioic acid (6048069)
ChemBridge特有类药化合物/先导化合物-6048069,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M12538 ChemBridge-6048841 ChemBridge化合物-6048841 Screening Compounds and Building Blocks
cyclopentyl 1,6-dimethyl-4-(6-nitro-1,3-benzodioxol-5-yl)-2-oxo-1,2,3,4-tetrahydro-5-pyrimidinecarboxylate (6048841)
ChemBridge特有类药化合物/先导化合物-6048841,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M12541 ChemBridge-6057025 ChemBridge化合物-6057025 Screening Compounds and Building Blocks
1-(4-bromo-3-methylphenyl)-5-[3-(2-furyl)-2-propen-1-ylidene]-2,4,6(1H,3H,5H)-pyrimidinetrione (6057025)
ChemBridge特有类药化合物/先导化合物-6057025,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M12544 ChemBridge-6062214 ChemBridge化合物-6062214 Screening Compounds and Building Blocks
1-(4-bromo-3-methylphenyl)-5-[(5-nitro-2-furyl)methylene]-2,4,6(1H,3H,5H)-pyrimidinetrione (6062214)
ChemBridge特有类药化合物/先导化合物-6062214,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M12545 ChemBridge-6062767 ChemBridge化合物-6062767 Screening Compounds and Building Blocks
1-(4-ethylphenyl)-5-[(5-iodo-2-furyl)methylene]-2-thioxodihydro-4,6(1H,5H)-pyrimidinedione (6062767)
ChemBridge特有类药化合物/先导化合物-6062767,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M12548 ChemBridge-6072466 ChemBridge化合物-6072466 Screening Compounds and Building Blocks
(3-{[1-(4-methylphenyl)-2,4,6-trioxotetrahydro-5(2H)-pyrimidinylidene]methyl}-1H-indol-1-yl)acetic acid (6072466)
ChemBridge特有类药化合物/先导化合物-6072466,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M12554 ChemBridge-6078578 ChemBridge化合物-6078578 Screening Compounds and Building Blocks
4-[(2-{[1-(4-methylphenyl)-2,4,6-trioxotetrahydro-5(2H)-pyrimidinylidene]methyl}phenoxy)methyl]benzoic acid (6078578)
ChemBridge特有类药化合物/先导化合物-6078578,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M12559 ChemBridge-6088649 ChemBridge化合物-6088649 Screening Compounds and Building Blocks
2-thioxo-5-[(1,2,5-trimethyl-1H-pyrrol-3-yl)methylene]dihydro-4,6(1H,5H)-pyrimidinedione (6088649)
ChemBridge特有类药化合物/先导化合物-6088649,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M12560 ChemBridge-6089114 ChemBridge化合物-6089114 Screening Compounds and Building Blocks
5-[(1,2,5-trimethyl-1H-pyrrol-3-yl)methylene]-2,4,6(1H,3H,5H)-pyrimidinetrione (6089114)
ChemBridge特有类药化合物/先导化合物-6089114,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M12563 ChemBridge-6092141 ChemBridge化合物-6092141 Screening Compounds and Building Blocks
2-thioxo-5-[(1,2,5-trimethyl-1H-pyrrol-3-yl)methylene]-1,3-thiazolidin-4-one (6092141)
ChemBridge特有类药化合物/先导化合物-6092141,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M12608 ChemBridge-6176046 ChemBridge化合物-6176046 Screening Compounds and Building Blocks
5-{[2,5-dimethyl-1-(3-pyridinyl)-1H-pyrrol-3-yl]methylene}-1,3-thiazolidine-2,4-dione (6176046)
ChemBridge特有类药化合物/先导化合物-6176046,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M12620 ChemBridge-6206065 ChemBridge化合物-6206065 Screening Compounds and Building Blocks
5-{[2,5-dimethyl-1-(3-pyridinyl)-1H-pyrrol-3-yl]methylene}-2,4-imidazolidinedione (6206065)
ChemBridge特有类药化合物/先导化合物-6206065,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M12622 ChemBridge-6211600 ChemBridge化合物-6211600 Screening Compounds and Building Blocks
5-[(1,2,5-trimethyl-1H-pyrrol-3-yl)methylene]-2,4-imidazolidinedione (6211600)
ChemBridge特有类药化合物/先导化合物-6211600,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M3243 Pyroxamide Pyroxamide HDAC
NSC-696085
Pyroxamide (NSC 696085)是一种有效的亲和纯化的HDAC1抑制剂,ID50 of 100 nM。
M5043 4-Chloro-7H-pyrrolo[2,3-d]pyrimidine 4-Chloro-7H-pyrrolo[2,3-d]pyrimidine Others
4-Chloro-7H-pyrrolo[2,3-d]pyrimidine是一种重要的医药中间体,在国内外广泛用于许多医药中间体的合成。包括CP690550、CGP76030等,同时也是许多市售药物的支架。此外,4-Chloro-7H-pyrrolo[2,3-d]pyrimidine也是Tofatinib原料药的中间体。
M7061 NTNCB hydrochloride NTNCB hydrochloride Neuropeptide Receptor
盐酸NTNCB是一种选择性的、非肽竞争性的NPY Y5拮抗剂。人重组Y5和Y1受体的Ki值分别为8.0和16032 nM。能拮抗NPY对forskolin刺激的cAMP的抑制作用。与克隆的人D2和α2C受体有一定的亲和力(Ki值分别为63和100 nM)。
M8438 Retro-2 cycl Retro-2 cycl Anti-infection
RN 1-001
Retro-2 cycl (RN 1-001) 是一种逆行运输抑制剂。Retro-2 cycl (RN 1-001) 抑制 JCPyV 和 HPV16 伪病毒,IC50 分别为 54 μM 和 160 μM。
M21083 PY-60 PY-60 YAP
PY-60 是一种靶向膜联蛋白A2 (ANXA2) 的 YAP 转录活性的特异的激活剂 (Kd=1.4 µM)。PY-60 直接与 ANXA2 结合并拮抗其抑制 YAP 活性的正常细胞功能。
M29770 Spiclomazine hydrochloride Spiclomazine hydrochloride Ras
APY-606; Clospirazine hydrochloride
Spiclomazine hydrochloride (APY-606) 是一种抗精神病药和抗肿瘤药。Spiclomazine hydrochloride 抑制 KRas。Spiclomazine hydrochloride 诱导癌细胞凋亡(apoptosis)。








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