找到约 34 条 “H-151” 相关结果 (用时 0.127 秒)
目录号 | 产品名称 | 中文名称 | 靶点 |
---|---|---|---|
M7278 | SCH 221510 | SCH 221510 | Others |
SCH 221510 is a potent and selective NOP agonist. | |||
M10126
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H-151 | H-151 | STING |
H151 | |||
H-151 是一种有效的,选择性的共价STING拮抗剂,可降低TBK1磷酸化并抑制人STING的棕榈酰化。 | |||
M11730 | ChemBridge-5151562 | ChemBridge化合物-5151562 | Screening Compounds and Building Blocks |
3-[3-(4'-bromo-4-biphenylyl)-1-phenyl-3-(phenylhydrazono)propyl]-4-hydroxy-2H-chromen-2-one (5151562) | |||
ChemBridge特有类药化合物/先导化合物-5151562,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M11737 | ChemBridge-5153248 | ChemBridge化合物-5153248 | Screening Compounds and Building Blocks |
4-bromo-N'-cyclohexylidenebenzohydrazide (5153248) | |||
ChemBridge特有类药化合物/先导化合物-5153248,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M11985 | ChemBridge-5315106 | ChemBridge化合物-5315106 | Screening Compounds and Building Blocks |
N'-(2,4-dichlorobenzylidene)-3,4-dihydroxybenzohydrazide (5315106) | |||
ChemBridge特有类药化合物/先导化合物-5315106,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M12424 | ChemBridge-5878151 | ChemBridge化合物-5878151 | Screening Compounds and Building Blocks |
1-[5-(3,4-dichlorophenyl)-2-furyl]-5-(2-furyl)-1,4-pentadien-3-one (5878151) | |||
ChemBridge特有类药化合物/先导化合物-5878151,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M12764 | ChemBridge-6714151 | ChemBridge化合物-6714151 | Screening Compounds and Building Blocks |
1-(3-chloro-4-methylbenzoyl)-4-(4-nitrophenyl)piperazine (6714151) | |||
ChemBridge特有类药化合物/先导化合物-6714151,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M13210 | ChemBridge-9151521 | ChemBridge化合物-9151521 | Screening Compounds and Building Blocks |
2-[(2-hydroxyphenyl)amino]-6-propyl-4(3H)-pyrimidinone (9151521) | |||
ChemBridge特有类药化合物/先导化合物-9151521,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M27592 | Icapamespib | Icapamespib | HSP |
PU-HZ151 | |||
Icapamespib (PU-HZ151) 是一种有效的 HSP90 抑制剂,EC50 值为5 nM. Icapamespib 可以透过血脑屏障。 | |||
M40528 | HM15136 | HM15136 | Glucagon Receptor |
HM15136是一种新型长效胰高血糖素类似物,同时也是胰高血糖素受体 (GCGR)的激动剂,可用于先天性高胰岛素血症的相关研究。 | |||
M45326
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ChemBridge-15135227 | ChemBridge化合物-15135227 | Screening Compounds and Building Blocks |
7-phenyl-2-(3-pyridin-3-yl-1,2,4-oxadiazol-5-yl)-5,6,7,8-tetrahydroimidazo[4,5-c]azepin-4(1H)-one | |||
ChemBridge特有类药化合物/先导化合物-15135227,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M45599 | ChemBridge-5539151 | ChemBridge化合物-5539151 | Screening Compounds and Building Blocks |
N-[2-(4-morpholinyl)ethyl]-1-phenylmethanesulfonamide (5539151) | |||
ChemBridge特有类药化合物/先导化合物-5539151,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M45826 | ChemBridge-6131513 | ChemBridge化合物-6131513 | Screening Compounds and Building Blocks |
methyl 2-amino-4-(2,4-dimethoxyphenyl)-3-thiophenecarboxylate (6131513) | |||
ChemBridge特有类药化合物/先导化合物-6131513,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M45856 | ChemBridge-6211513 | ChemBridge化合物-6211513 | Screening Compounds and Building Blocks |
2-(benzylthio)-N-(3-chlorophenyl)propanamide (6211513) | |||
ChemBridge特有类药化合物/先导化合物-6211513,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M46192 | ChemBridge-7645151 | ChemBridge化合物-7645151 | Screening Compounds and Building Blocks |
N-(4-{[(5-methyl-3-isoxazolyl)amino]sulfonyl}phenyl)-2-[(4-methyl-2-oxo-2H-chromen-7-yl)oxy]acetamide (7645151) | |||
ChemBridge特有类药化合物/先导化合物-7645151,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M46319 | ChemBridge-7815143 | ChemBridge化合物-7815143 | Screening Compounds and Building Blocks |
ethyl 4-({[(4-methoxy-2-methylphenyl)amino]carbonothioyl}amino)benzoate (7815143) | |||
ChemBridge特有类药化合物/先导化合物-7815143,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M46392 | ChemBridge-7911151 | ChemBridge化合物-7911151 | Screening Compounds and Building Blocks |
N-1,3-benzodioxol-5-yl-2-{[4-(2-furylmethyl)-5-(3-pyridinyl)-4H-1,2,4-triazol-3-yl]thio}acetamide (7911151) | |||
ChemBridge特有类药化合物/先导化合物-7911151,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M46686 | ChemBridge-8901517 | ChemBridge化合物-8901517 | Screening Compounds and Building Blocks |
2-iodo-N-[4-oxo-2-(8-quinolinyl)-1,4-dihydro-3(2H)-quinazolinyl]benzamide (8901517) | |||
ChemBridge特有类药化合物/先导化合物-8901517,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M46835 | ChemBridge-9072151 | ChemBridge化合物-9072151 | Screening Compounds and Building Blocks |
8-sec-butyl-1,7-dimethyl-3-(3-methylbutyl)-1H-imidazo[2,1-f]purine-2,4(3H,8H)-dione (9072151) | |||
ChemBridge特有类药化合物/先导化合物-9072151,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M46983 | ChemBridge-9151602 | ChemBridge化合物-9151602 | Screening Compounds and Building Blocks |
N-{2-[(2-chlorophenyl)amino]-2-oxoethyl}-2-furamide (9151602) | |||
ChemBridge特有类药化合物/先导化合物-9151602,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M46984 | ChemBridge-9151901 | ChemBridge化合物-9151901 | Screening Compounds and Building Blocks |
3-[4-methyl-5-(1-piperidinylcarbonyl)-1,3-thiazol-2-yl]pyridine (9151901) | |||
ChemBridge特有类药化合物/先导化合物-9151901,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M47037 | ChemBridge-9215162 | ChemBridge化合物-9215162 | Screening Compounds and Building Blocks |
4-[(4-fluorophenoxy)acetyl]-3,4-dihydro-2(1H)-quinoxalinone (9215162) | |||
ChemBridge特有类药化合物/先导化合物-9215162,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M47283 | ChemBridge-11515325 | ChemBridge化合物-11515325 | Screening Compounds and Building Blocks |
N-[(1-cyclopentylpiperidin-4-yl)methyl]-3-(methoxymethyl)piperidine-1-sulfonamide (11515325) | |||
ChemBridge特有类药化合物/先导化合物-11515325,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M47393 | ChemBridge-15110689 | ChemBridge化合物-15110689 | Screening Compounds and Building Blocks |
2-{[(1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl)amino]methyl}-4(3H)-quinazolinone (15110689) | |||
ChemBridge特有类药化合物/先导化合物-15110689,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M47394 | ChemBridge-15119077 | ChemBridge化合物-15119077 | Screening Compounds and Building Blocks |
N-{4-[1-(imidazo[1,2-a]pyridin-3-ylmethyl)-1H-1,2,3-triazol-4-yl]phenyl}acetamide (15119077) | |||
ChemBridge特有类药化合物/先导化合物-15119077,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M47395 | ChemBridge-15123722 | ChemBridge化合物-15123722 | Screening Compounds and Building Blocks |
4-[(3-ethyl-5-isoxazolyl)carbonyl]-5-methyl-1-(4-methylphenyl)-2-piperazinone (15123722) | |||
ChemBridge特有类药化合物/先导化合物-15123722,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M47397 | ChemBridge-15135771 | ChemBridge化合物-15135771 | Screening Compounds and Building Blocks |
1-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-4-piperidinamine dihydrochloride (15135771) | |||
ChemBridge特有类药化合物/先导化合物-15135771,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M47398 | ChemBridge-15168253 | ChemBridge化合物-15168253 | Screening Compounds and Building Blocks |
1-[(5-phenyl-1H-pyrazol-3-yl)carbonyl]-4-(tetrahydrofuran-3-ylmethyl)-1,4-diazepane (15168253) | |||
ChemBridge特有类药化合物/先导化合物-15168253,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M47399 | ChemBridge-15181021 | ChemBridge化合物-15181021 | Screening Compounds and Building Blocks |
2-(5-amino-1H-1,2,4-triazol-3-yl)-N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)acetamide (15181021) | |||
ChemBridge特有类药化合物/先导化合物-15181021,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M47776 | ChemBridge-30151353 | ChemBridge化合物-30151353 | Screening Compounds and Building Blocks |
5-methoxy-3-methyl-N-(7-methyl[1,2,4]triazolo[4,3-a]pyrimidin-3-yl)-1H-indole-2-carboxamide (30151353) | |||
ChemBridge特有类药化合物/先导化合物-30151353,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M2669
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Entacapone | 恩他卡朋 | FTO |
OR-611 | |||
Entacapone是一种 FTO demethylation的抑制剂,IC50为3.5 μM,Entacapone还抑制儿茶酚-O-甲基转移酶(COMT)活性,IC50为151 nM。 | |||
M8767 | MIND4-17 | MIND4-17 | Others |
MIND4-17 is a potent NRF2 (nuclear factor erythroid 2-related factor 2) activator that covalently modifies a critical stress-sensor cysteine (C151) in the BTB domain of the E3 ligase substrate adaptor protein Kelch-like ECH-associated protein 1 (KEAP1). | |||
M30504 | Pentachloropseudilin | Pentachloropseudilin | Myosin |
Antibiotic A 15104 Y; PClP | |||
Pentachloropseudilin (Antibiotic A 15104 Y; PClP) 是一种可逆的、变构有效的肌球蛋白 (Myo1s) 抑制剂,对 Myo1s 的 IC50 范围为 1 至 5 μM,对于 2 类和 5 类肌球蛋白,IC50 范围 > 90 μM。Pentachloropseudilin 是转化生长因子-β (TGF-β) 刺激的信号传导的有效抑制剂,对 TGF-β 的 IC50 值为 0.1-0.2 μM。 | |||
M41311 | RTA 744 | RTA 744 | Apoptosis |
RTA 744 (WP 744) 是一种阿霉素 (Doxorubicin,HY-15142A) 类似物。 |