找到约 2 条 “GSK 5959” 相关结果 （用时 0.179 秒）
| 目录号 | 产品名称 | 中文名称 | 靶点 |
|---|---|---|---|
M5239
|
Batefenterol | 巴特芬托尔 | Adrenergic Receptor |
| GSK961081; TD-5959 | |||
| Batefenterol (GSK961081; TD-5959) 是一种新的muscarinic受体拮抗剂和β2-肾上腺素受体激动剂; 对hM2，hM3和β2-肾上腺素受体有高亲和力，Ki值分别为1.4, 1.3和3.7nM。 | |||
| M20549 | GSK 5959 | GSK 5959 | Epigenetic Reader Domain |
| GSK5959 is a potent and selective BRPF1 bromodomain inhibitor with an IC50 of 80 nM and exhibits >100-fold selectivity for BRPF1 over a panel of 35 other bromodomains, including BRPF2/3 and BET family bromodomains. | |||
