找到约 4 条 “Carvedilol” 相关结果 (用时 0.103 秒)
目录号 | 产品名称 | 中文名称 | 靶点 |
---|---|---|---|
M3482
![]() |
Carvedilol | 卡维地洛 | Adrenergic Receptor |
BM 14190 | |||
Carvedilol(卡维地洛)是一种第三代非选择性β/α1受体阻滞剂。在动物实验中,Carvedilol通过阻断β1、β2和α1受体,发挥降压和心血管保护作用。Carvedilol还能清除自由基并抑制脂质过氧化,IC50值为5 μM。并且,Carvedilol还是一种自噬诱导剂,可以抑制NLRP3炎性小体。 | |||
M1580
![]() |
4-Hydroxy phenyl carvedilol | 4-Hydroxy phenyl carvedilol | Metabolite/Endogenous Metabolite |
4-Hydroxyphenyl Carvedilol; 4-Hydroxycarvedilol | |||
4-Hydroxyphenyl Carvedilol是Carvedilol的代谢物。 | |||
M20525 | Carvedilol Phosphate | Carvedilol Phosphate | Others |
Carvedilol Phosphate is the phosphate salt form of carvedilol, a racemic mixture and adrenergic blocking agent with antihypertensive activity and devoid of intrinsic sympathomimetic activity. | |||
M20531 | Carvedilol EP IMpurity E | Carvedilol EP IMpurity E | Others |
Used as pharmaceutical intermediates-Intermediates |