找到约 4 条 “Carvedilol” 相关结果 (用时 0.103 秒)

目录号 产品名称 中文名称 靶点
M3482 Carvedilol 卡维地洛 Adrenergic Receptor
BM 14190
Carvedilol(卡维地洛)是一种第三代非选择性β/α1受体阻滞剂。在动物实验中,Carvedilol通过阻断β1、β2和α1受体,发挥降压和心血管保护作用。Carvedilol还能清除自由基并抑制脂质过氧化,IC50值为5 μM。并且,Carvedilol还是一种自噬诱导剂,可以抑制NLRP3炎性小体。
M1580 4-Hydroxy phenyl carvedilol 4-Hydroxy phenyl carvedilol Metabolite/Endogenous Metabolite
4-Hydroxyphenyl Carvedilol; 4-Hydroxycarvedilol
4-Hydroxyphenyl Carvedilol是Carvedilol的代谢物。
M20525 Carvedilol Phosphate Carvedilol Phosphate Others
Carvedilol Phosphate is the phosphate salt form of carvedilol, a racemic mixture and adrenergic blocking agent with antihypertensive activity and devoid of intrinsic sympathomimetic activity.
M20531 Carvedilol EP IMpurity E Carvedilol EP IMpurity E Others
Used as pharmaceutical intermediates-Intermediates








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