找到约 12 条 “84-16-2” 相关结果 (用时 0.11 秒)
目录号 | 产品名称 | 中文名称 | 靶点 |
---|---|---|---|
M3333 | Hexestrol | 己烷雌酚 | Estrogen Receptor |
Bibenzyl | |||
Hexestrol是一种非甾体合成雌激素,其与ERα和ERβ结合,EC50分别为0.07 nM和0.175 nM,Ki 值均为 0.06 nM。Hexestrol 可用于研究雌激素缺乏引起的疾病。 | |||
M7326 | SR 142948 | SR 142948 | Others |
SR 142948 is a highly potent NT receptor antagonist. | |||
M8205 | SR 142948A | SR 142948A | Others |
SR 142948A is a non-peptide Neurotensin receptor antagonist. | |||
M8414 | MJN110 | MJN110 | MAGL |
MJN110 is a potent selective inhibitor of MAGL, the enzyme predominantly responsible for the degradation of the endocannabinoid 2-arachidonoylglycerol (2-AG) with >10,000 selectivity over FAAH. | |||
M8506 | ML351 | ML351 | Lipoxygenase |
ML351 is a cell penetrant, selective and highly potent human lipoxygenase-12/15 (15-Lipoxygenase-1, 12/15-LOX) inhibitor that exhibits protective effects against oxidative glutamate toxicity in mouse neuronal HT22 cells. | |||
M18584 | Eleutheroside B1 | 刺五加苷B1 | Others |
Eleutheroside B1 刺五加苷B1 | |||
M20965 | FDL169 | FDL169 | CFTR |
FDL169 is a CFTR corrector that is designed to fix and restore the function of the defective CFTR protein. | |||
M25256 | Lexatumumab | Lexatumumab | Apoptosis |
HGS-ETR 2 ETR2-ST01 Anti-Human ERBB3 Recombinant Antibody | |||
Lexatumumab (HGS-ETR 2) 是一种人源激动 TRAIL 受体 2 (TRAIL-R2, DR5, APO-2) IgG4κ 型单克隆抗体。Lexatumumab 在恶性间皮瘤中诱导细胞凋亡 (apoptosis)。Lexatumumab 可用于恶性胸膜间皮瘤 (MPM) 研究。 | |||
M49795 | ALC-0159 | ALC-0159 | Liposome |
ALC-0159是一种聚乙二醇的脂质结合物,可用作疫苗的赋形剂。 | |||
M54418 | FC131 TFA | FC131 TFA | CXCR |
FC131 TFA 是一种 CXCR4 拮抗剂,抑制 [125I]-SDF-1 与 CXCR4 结合,IC50 值为 4.5 nM。 | |||
M3282 | GW842166X | GW842166X | Cannabinoid |
GW842166X是一种有效的,高选择性cannabinoid receptor CB2受体激动剂,EC50为63 nM,对CB1受体没有显著的活性。 | |||
M25278 | Pegdinetanib | Pegdinetanib | VEGFR/PDGFR |
BMS-844203; CT-322 | |||
Pegdinetanib (BMS-844203; CT-322) 是一种选择性 VEGFR-2 (VEGFR) 抑制剂,对人和鼠 VEGFR-2 的 Kd 分别为 11 nM 和 250 nM,IC50 分别为 16 nM 和 240 nM。Pegdinetanib 不与 VEGFR-1 或 VEGFR-3 结合。Pegdinetanib 具有抗肿瘤活性。 |
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