找到约 23 条 “5-LOX-IN-2” 相关结果 (用时 0.109 秒)
目录号 | 产品名称 | 中文名称 | 靶点 |
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M5370
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5,5-Dimethyloxazolidine-2,4-dione | 5,5-Dimethyloxazolidine-2,4-dione | Metabolite/Endogenous Metabolite |
Dimethadione, Dimethyloxazolidinedione, Dimethadion | |||
Dimethadione是一种抗痉挛剂,是三甲双酮的活性代谢产物。 | |||
M6038
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Trimethadione | 三甲双酮 | Calcium Channel |
3,5,5,-Trimethyloxazolidine-2,4-dione | |||
Trimethadione是一一种恶唑烷二酮,抗惊厥化合物。 | |||
M13177 | ChemBridge-9010672 | ChemBridge化合物-9010672 | Screening Compounds and Building Blocks |
1-[2-(2,3-dihydro-1H-inden-5-yloxy)ethyl]piperidine hydrochloride (9010672) | |||
ChemBridge特有类药化合物/先导化合物-9010672,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M42005 | COX-2/15-LOX-IN-2 | COX-2/15-LOX-IN-2 | Lipoxygenase |
COX-2/15-LOX-IN-2 是有效的双 COX-2 和 15-LOX 抑制剂,其 IC50 值分别为 0.065 μM 和 1.86 μM。 | |||
M42481 | 5-LOX-IN-2 | 5-LOX-IN-2 | Lipoxygenase |
5-LOX-IN-2 是 一种 5-脂氧合酶抑制剂 (5-LOX ),IC50 为 0.33 μM,以剂量依赖的方式抑制 5-LOX。 | |||
M46017 | ChemBridge-6943202 | ChemBridge化合物-6943202 | Screening Compounds and Building Blocks |
1-(2,3-dihydro-1H-inden-5-yloxy)-3-[4-(4-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride (6943202) | |||
ChemBridge特有类药化合物/先导化合物-6943202,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M46019 | ChemBridge-6943807 | ChemBridge化合物-6943807 | Screening Compounds and Building Blocks |
1-(1,3-benzodioxol-5-yloxy)-3-[cyclohexyl(methyl)amino]-2-propanol hydrochloride (6943807) | |||
ChemBridge特有类药化合物/先导化合物-6943807,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M46734 | ChemBridge-8926036 | ChemBridge化合物-8926036 | Screening Compounds and Building Blocks |
2-[3-(2,3-dihydro-1H-inden-5-yloxy)-4-methoxyphenyl]-9-methyl-7-(trifluoromethyl)-2,3-dihydropyrido[3',2':4,5]thieno[3,2-d]pyrimidin-4(1H)-one (8926036) | |||
ChemBridge特有类药化合物/先导化合物-8926036,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M47655 | ChemBridge-25415991 | ChemBridge化合物-25415991 | Screening Compounds and Building Blocks |
2-[(1,3-benzodioxol-5-yloxy)methyl]-N-[1-(1H-indol-5-yl)ethyl]-1,3-oxazole-4-carboxamide (25415991) | |||
ChemBridge特有类药化合物/先导化合物-25415991,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M47927 | ChemBridge-35982747 | ChemBridge化合物-35982747 | Screening Compounds and Building Blocks |
N-[4-(1H-tetrazol-5-yloxy)phenyl]quinoline-5-carboxamide (35982747) | |||
ChemBridge特有类药化合物/先导化合物-35982747,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M48109 | ChemBridge-44146133 | ChemBridge化合物-44146133 | Screening Compounds and Building Blocks |
4-(5-{[4-(pyridin-3-yloxy)piperidin-1-yl]carbonyl}pyridin-2-yl)morpholine (44146133) | |||
ChemBridge特有类药化合物/先导化合物-44146133,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M48197 | ChemBridge-47387227 | ChemBridge化合物-47387227 | Screening Compounds and Building Blocks |
1-(3-methoxybenzyl)-5-{[4-(3-pyridinyloxy)-1-piperidinyl]carbonyl}-2-piperidinone (47387227) | |||
ChemBridge特有类药化合物/先导化合物-47387227,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M48576 | ChemBridge-62949254 | ChemBridge化合物-62949254 | Screening Compounds and Building Blocks |
N-[4-(1H-tetrazol-5-yloxy)phenyl]quinoline-8-carboxamide (62949254) | |||
ChemBridge特有类药化合物/先导化合物-62949254,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M48665 | ChemBridge-67052491 | ChemBridge化合物-67052491 | Screening Compounds and Building Blocks |
6-methyl-2-pyridin-3-yl-N-[4-(1H-tetrazol-5-yloxy)phenyl]quinoline-4-carboxamide (67052491) | |||
ChemBridge特有类药化合物/先导化合物-67052491,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M49021 | ChemBridge-84103708 | ChemBridge化合物-84103708 | Screening Compounds and Building Blocks |
N,N-dimethyl-N'-(5-{[4-(pyridin-3-yloxy)piperidin-1-yl]carbonyl}pyridin-2-yl)ethane-1,2-diamine (84103708) | |||
ChemBridge特有类药化合物/先导化合物-84103708,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M6394
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AC 45594 | AC 45594 | Anti-infection |
4-Heptyloxyphenol | |||
AC 45594(4-Heptyloxyphenol)是一种类固醇生成因子 1 (SF-1)的反向激动剂先导物,IC50值为 50-100 nM。4-Heptyloxyphenol (AC 45594) 对 P. gingivalis, S. artemidis, Str. sobrinus 有抗菌活性 (MIC: 0.10, 0.21, 0.14 mM)。 | |||
M7964
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Nordihydroguaiaretic acid | 去甲二氢愈创木酸 | Lipoxygenase |
NDGA | |||
Nordihydroguaiaretic acid (NDGA) 是一种 5-脂氧合酶 (5LOX) (IC50=8 μM) 和酪氨酸激酶抑制剂,具有抗氧化、清除自由基的活性。Nordihydroguaiaretic acid (NDGA) 是一种具有细胞毒性的 insulin-like growth factor-I receptor (IGF-1R)/HER2 的抑制剂,可诱导细胞凋亡。Nordihydroguaiaretic acid (NDGA) 是一种ABA合成抑制剂。 | |||
M8506
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ML351 | ML351 | Lipoxygenase |
ML351 is a cell penetrant, selective and highly potent human lipoxygenase-12/15 (15-Lipoxygenase-1, 12/15-LOX) inhibitor that exhibits protective effects against oxidative glutamate toxicity in mouse neuronal HT22 cells. | |||
M42482 | h15-LOX-2 inhibitor 1 | h15-LOX-2 inhibitor 1 | Lipoxygenase |
h15-LOX-2 inhibitor 1 是一种人上皮细胞 15-lipoxygenase-2 (h15-LOX-2) 抑制剂,其 IC50 值为 0.34 μM。 | |||
M42484 | COX-2/15-LOX-IN-3 | COX-2/15-LOX-IN-3 | Lipoxygenase |
COX-2/15-LOX-IN-3 是 COX-2/15-LOX 的双抑制剂,IC50s 分别为 0.075 μM 和 1.97 μM。 | |||
M42485 | COX-2/15-LOX-IN-4 | COX-2/15-LOX-IN-4 | Lipoxygenase |
COX-2/15-LOX-IN-4 是 COX-2/15-LOX 的双抑制剂,IC50s 分别为 0.075 μM 和 1.97 μM。 | |||
M45337 | ALOX15-IN-2 | ALOX15-IN-2 | Lipoxygenase |
ALOX15-IN-2是一种有效的兔和人 ALOX15 亚油酸加氧酶 (linoleate oxygenase) 活性抑制剂,对 ALOX15 直系同源物亚油酸 (LA) 和花生四烯酸 (AA) 的 IC50 分别为 1.55 和 2.79 μM。 | |||
M56711 | 5-LOX-IN-1 | 5-LOX-IN-1 | Lipoxygenase |
5-LOX-IN-1 是 5-Lipoxygenase (5-LOX) 的抑制剂,IC50 值为 2.3 μM。5-LOX-IN-1 可用于癌症的研究。 |