找到约 26 条 “TH-257” 相关结果 (用时 0.112 秒)
目录号 | 产品名称 | 中文名称 | 靶点 |
---|---|---|---|
M8745 | ITH12575 | ITH12575 | Others |
ITH12575 is apotent and selective inhibitor of mitochondrial Na+/Ca2+ exchanger mNCX with neuroprotective activity. | |||
M9499
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TH-257 | TH-257 | LIM Kinase |
TH257 | |||
TH-257是一种有效的选择性变构LIMK 1/2抑制剂,对LIMK1和LIMK2的IC50值分别为84 nM和39 nM。 | |||
M12443 | ChemBridge-5925714 | ChemBridge化合物-5925714 | Screening Compounds and Building Blocks |
N-[3-(hydrazinocarbonyl)-2-naphthyl]benzenesulfonamide (5925714) | |||
ChemBridge特有类药化合物/先导化合物-5925714,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M46088 | ChemBridge-7225782 | ChemBridge化合物-7225782 | Screening Compounds and Building Blocks |
N-[4-(diethylamino)phenyl]-2-phenylbutanamide (7225782) | |||
ChemBridge特有类药化合物/先导化合物-7225782,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M46420 | ChemBridge-7925726 | ChemBridge化合物-7925726 | Screening Compounds and Building Blocks |
N-(5-methyl-3-isoxazolyl)-2-(5-nitro-1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)acetamide (7925726) | |||
ChemBridge特有类药化合物/先导化合物-7925726,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M46457 | ChemBridge-7952576 | ChemBridge化合物-7952576 | Screening Compounds and Building Blocks |
N-(5-methyl-3-isoxazolyl)-4-(2-oxo-1-pyrrolidinyl)benzenesulfonamide (7952576) | |||
ChemBridge特有类药化合物/先导化合物-7952576,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M46732 | ChemBridge-8925722 | ChemBridge化合物-8925722 | Screening Compounds and Building Blocks |
5-methyl-N-(4-{[(2-methylphenyl)amino]sulfonyl}phenyl)-1,3-diphenyl-1H-pyrazole-4-carboxamide (8925722) | |||
ChemBridge特有类药化合物/先导化合物-8925722,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M47052 | ChemBridge-9225712 | ChemBridge化合物-9225712 | Screening Compounds and Building Blocks |
2-methyl-9-phenyl-7-(1H-1,2,4-triazol-5-yl)pyrido[4,3-d][1,2,4]triazolo[1,5-a]pyrimidin-8(7H)-one (9225712) | |||
ChemBridge特有类药化合物/先导化合物-9225712,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M47166 | ChemBridge-9302570 | ChemBridge化合物-9302570 | Screening Compounds and Building Blocks |
N-(4-methoxybenzyl)-5-(2-methoxyphenyl)-3-isoxazolecarboxamide (9302570) | |||
ChemBridge特有类药化合物/先导化合物-9302570,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M47452 | ChemBridge-17525765 | ChemBridge化合物-17525765 | Screening Compounds and Building Blocks |
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(isopropylthio)acetyl]piperidine (17525765) | |||
ChemBridge特有类药化合物/先导化合物-17525765,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M47576 | ChemBridge-22062574 | ChemBridge化合物-22062574 | Screening Compounds and Building Blocks |
N-methyl-N-[1-[1-(4-methyl-2-oxopentanoyl)-4-piperidinyl]-2-(2-methylphenyl)ethyl]-2-(1H-pyrazol-1-yl)acetamide (22062574) | |||
ChemBridge特有类药化合物/先导化合物-22062574,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M47665 | ChemBridge-25740113 | ChemBridge化合物-25740113 | Screening Compounds and Building Blocks |
(3aR*,9bR*)-2-(5-ethyl-2,6-dimethylpyrimidin-4-yl)-7-methoxy-1,2,3,9b-tetrahydrochromeno[3,4-c]pyrrole-3a(4H)-carboxylic acid (25740113) | |||
ChemBridge特有类药化合物/先导化合物-25740113,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M48163 | ChemBridge-46257037 | ChemBridge化合物-46257037 | Screening Compounds and Building Blocks |
6-(4-methyl-3-oxopiperazin-1-yl)-N-[(3-propylisoxazol-5-yl)methyl]nicotinamide (46257037) | |||
ChemBridge特有类药化合物/先导化合物-46257037,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M48223 | ChemBridge-48496257 | ChemBridge化合物-48496257 | Screening Compounds and Building Blocks |
N-[(3-hydroxycyclobutyl)(6-methoxypyridin-3-yl)methyl]-6-methylimidazo[1,2-a]pyridine-2-carboxamide (48496257) | |||
ChemBridge特有类药化合物/先导化合物-48496257,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M48420 | ChemBridge-56257359 | ChemBridge化合物-56257359 | Screening Compounds and Building Blocks |
[1-(3-chloro-4-{[1-(methylsulfonyl)-4-piperidinyl]oxy}benzoyl)-4-piperidinyl]methanol (56257359) | |||
ChemBridge特有类药化合物/先导化合物-56257359,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M48472 | ChemBridge-58825731 | ChemBridge化合物-58825731 | Screening Compounds and Building Blocks |
N-[(S*)-(cis-3-hydroxycyclobutyl)(1-methyl-1H-pyrazol-4-yl)methyl]-2-(8-methylimidazo[1,2-a]pyridin-3-yl)acetamide (58825731) | |||
ChemBridge特有类药化合物/先导化合物-58825731,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M48531 | ChemBridge-61257229 | ChemBridge化合物-61257229 | Screening Compounds and Building Blocks |
rac-(1S,3S,7aR)-3-phenyl-N-[2-(1H-tetrazol-5-yl)ethyl]hexahydro-1H-pyrrolizine-1-carboxamide (61257229) | |||
ChemBridge特有类药化合物/先导化合物-61257229,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M48677 | ChemBridge-67325780 | ChemBridge化合物-67325780 | Screening Compounds and Building Blocks |
(3aS*,6aR*)-5-benzoyl-3-[2-(4-methoxyphenyl)ethyl]hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one (67325780) | |||
ChemBridge特有类药化合物/先导化合物-67325780,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M48701 | ChemBridge-68725758 | ChemBridge化合物-68725758 | Screening Compounds and Building Blocks |
2-(1,2,4,5-tetrahydro-3H-3-benzazepin-3-ylmethyl)benzonitrile (68725758) | |||
ChemBridge特有类药化合物/先导化合物-68725758,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M48729 | ChemBridge-70192579 | ChemBridge化合物-70192579 | Screening Compounds and Building Blocks |
N-methyl-6-(2-phenylpropyl)-4-(1-pyrrolidinylcarbonyl)-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-amine (70192579) | |||
ChemBridge特有类药化合物/先导化合物-70192579,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M49193 | ChemBridge-92574394 | ChemBridge化合物-92574394 | Screening Compounds and Building Blocks |
2,3-dimethyl-6-{[3-(3-methyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]carbonyl}quinoxaline (92574394) | |||
ChemBridge特有类药化合物/先导化合物-92574394,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M49981 | ChemBridge-82525720 | ChemBridge化合物-82525720 | Screening Compounds and Building Blocks |
3-methyl-N-[4-methyl-3-(propionylamino)phenyl]-4-morpholin-4-ylbenzamide (82525720) | |||
ChemBridge特有类药化合物/先导化合物-82525720,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M49987 | ChemBridge-72598257 | ChemBridge化合物-72598257 | Screening Compounds and Building Blocks |
3-hydroxy-3-({[2-(methylamino)ethyl]amino}methyl)-1-(2-phenylethyl)piperidin-2-one (72598257) | |||
ChemBridge特有类药化合物/先导化合物-72598257,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M49988 | ChemBridge-62570111 | ChemBridge化合物-62570111 | Screening Compounds and Building Blocks |
6-({[(6-methylimidazo[1,2-a]pyridin-2-yl)methyl]amino}methyl)-1,4-oxazepan-6-ol dihydrochloride (62570111) | |||
ChemBridge特有类药化合物/先导化合物-62570111,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M4909
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GSK2801 | GSK2801 | Epigenetic Reader Domain |
GSK2801 is a selective bromodomains BAZ2A/B inhibitor with KD of 257 nM and 136 nM, respectively. | |||
M15079
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Recombinant Human NT-3 (E.coli) | 重组人NT-3蛋白 (E.coli) | Cytokines and Growth Factors |
Neurotrophin-3; NT-3; HDNF; Nerve Growth Factor 2 | |||
利用大肠杆菌表达系统制备了重组人神经营养因子-3,并表达了编码Tyr139-Thr257的目的基因。Accession #: P20783。 |