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 找到约 26 条 “TH-257” 相关结果 (用时 0.164 秒)

目录号 产品名称 中文名称 靶点
M8745 ITH12575 ITH12575 Others
ITH12575 is apotent and selective inhibitor of mitochondrial Na+/Ca2+ exchanger mNCX with neuroprotective activity.
M9499 TH-257 TH-257 LIM Kinase
TH257
TH-257是一种有效的选择性变构LIMK 1/2抑制剂,对LIMK1和LIMK2的IC50值分别为84 nM和39 nM。
M12443 ChemBridge-5925714 ChemBridge化合物-5925714 Screening Compounds and Building Blocks
N-[3-(hydrazinocarbonyl)-2-naphthyl]benzenesulfonamide (5925714)
ChemBridge特有类药化合物/先导化合物-5925714,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M46088 ChemBridge-7225782 ChemBridge化合物-7225782 Screening Compounds and Building Blocks
N-[4-(diethylamino)phenyl]-2-phenylbutanamide (7225782)
ChemBridge特有类药化合物/先导化合物-7225782,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M46420 ChemBridge-7925726 ChemBridge化合物-7925726 Screening Compounds and Building Blocks
N-(5-methyl-3-isoxazolyl)-2-(5-nitro-1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)acetamide (7925726)
ChemBridge特有类药化合物/先导化合物-7925726,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M46457 ChemBridge-7952576 ChemBridge化合物-7952576 Screening Compounds and Building Blocks
N-(5-methyl-3-isoxazolyl)-4-(2-oxo-1-pyrrolidinyl)benzenesulfonamide (7952576)
ChemBridge特有类药化合物/先导化合物-7952576,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M46732 ChemBridge-8925722 ChemBridge化合物-8925722 Screening Compounds and Building Blocks
5-methyl-N-(4-{[(2-methylphenyl)amino]sulfonyl}phenyl)-1,3-diphenyl-1H-pyrazole-4-carboxamide (8925722)
ChemBridge特有类药化合物/先导化合物-8925722,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M47052 ChemBridge-9225712 ChemBridge化合物-9225712 Screening Compounds and Building Blocks
2-methyl-9-phenyl-7-(1H-1,2,4-triazol-5-yl)pyrido[4,3-d][1,2,4]triazolo[1,5-a]pyrimidin-8(7H)-one (9225712)
ChemBridge特有类药化合物/先导化合物-9225712,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M47166 ChemBridge-9302570 ChemBridge化合物-9302570 Screening Compounds and Building Blocks
N-(4-methoxybenzyl)-5-(2-methoxyphenyl)-3-isoxazolecarboxamide (9302570)
ChemBridge特有类药化合物/先导化合物-9302570,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M47452 ChemBridge-17525765 ChemBridge化合物-17525765 Screening Compounds and Building Blocks
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(isopropylthio)acetyl]piperidine (17525765)
ChemBridge特有类药化合物/先导化合物-17525765,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M47576 ChemBridge-22062574 ChemBridge化合物-22062574 Screening Compounds and Building Blocks
N-methyl-N-[1-[1-(4-methyl-2-oxopentanoyl)-4-piperidinyl]-2-(2-methylphenyl)ethyl]-2-(1H-pyrazol-1-yl)acetamide (22062574)
ChemBridge特有类药化合物/先导化合物-22062574,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M47665 ChemBridge-25740113 ChemBridge化合物-25740113 Screening Compounds and Building Blocks
(3aR*,9bR*)-2-(5-ethyl-2,6-dimethylpyrimidin-4-yl)-7-methoxy-1,2,3,9b-tetrahydrochromeno[3,4-c]pyrrole-3a(4H)-carboxylic acid (25740113)
ChemBridge特有类药化合物/先导化合物-25740113,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M48163 ChemBridge-46257037 ChemBridge化合物-46257037 Screening Compounds and Building Blocks
6-(4-methyl-3-oxopiperazin-1-yl)-N-[(3-propylisoxazol-5-yl)methyl]nicotinamide (46257037)
ChemBridge特有类药化合物/先导化合物-46257037,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M48223 ChemBridge-48496257 ChemBridge化合物-48496257 Screening Compounds and Building Blocks
N-[(3-hydroxycyclobutyl)(6-methoxypyridin-3-yl)methyl]-6-methylimidazo[1,2-a]pyridine-2-carboxamide (48496257)
ChemBridge特有类药化合物/先导化合物-48496257,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M48420 ChemBridge-56257359 ChemBridge化合物-56257359 Screening Compounds and Building Blocks
[1-(3-chloro-4-{[1-(methylsulfonyl)-4-piperidinyl]oxy}benzoyl)-4-piperidinyl]methanol (56257359)
ChemBridge特有类药化合物/先导化合物-56257359,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M48472 ChemBridge-58825731 ChemBridge化合物-58825731 Screening Compounds and Building Blocks
N-[(S*)-(cis-3-hydroxycyclobutyl)(1-methyl-1H-pyrazol-4-yl)methyl]-2-(8-methylimidazo[1,2-a]pyridin-3-yl)acetamide (58825731)
ChemBridge特有类药化合物/先导化合物-58825731,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M48531 ChemBridge-61257229 ChemBridge化合物-61257229 Screening Compounds and Building Blocks
rac-(1S,3S,7aR)-3-phenyl-N-[2-(1H-tetrazol-5-yl)ethyl]hexahydro-1H-pyrrolizine-1-carboxamide (61257229)
ChemBridge特有类药化合物/先导化合物-61257229,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M48677 ChemBridge-67325780 ChemBridge化合物-67325780 Screening Compounds and Building Blocks
(3aS*,6aR*)-5-benzoyl-3-[2-(4-methoxyphenyl)ethyl]hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one (67325780)
ChemBridge特有类药化合物/先导化合物-67325780,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M48701 ChemBridge-68725758 ChemBridge化合物-68725758 Screening Compounds and Building Blocks
2-(1,2,4,5-tetrahydro-3H-3-benzazepin-3-ylmethyl)benzonitrile (68725758)
ChemBridge特有类药化合物/先导化合物-68725758,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M48729 ChemBridge-70192579 ChemBridge化合物-70192579 Screening Compounds and Building Blocks
N-methyl-6-(2-phenylpropyl)-4-(1-pyrrolidinylcarbonyl)-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-amine (70192579)
ChemBridge特有类药化合物/先导化合物-70192579,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M49193 ChemBridge-92574394 ChemBridge化合物-92574394 Screening Compounds and Building Blocks
2,3-dimethyl-6-{[3-(3-methyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]carbonyl}quinoxaline (92574394)
ChemBridge特有类药化合物/先导化合物-92574394,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M49981 ChemBridge-82525720 ChemBridge化合物-82525720 Screening Compounds and Building Blocks
3-methyl-N-[4-methyl-3-(propionylamino)phenyl]-4-morpholin-4-ylbenzamide (82525720)
ChemBridge特有类药化合物/先导化合物-82525720,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M49987 ChemBridge-72598257 ChemBridge化合物-72598257 Screening Compounds and Building Blocks
3-hydroxy-3-({[2-(methylamino)ethyl]amino}methyl)-1-(2-phenylethyl)piperidin-2-one (72598257)
ChemBridge特有类药化合物/先导化合物-72598257,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M49988 ChemBridge-62570111 ChemBridge化合物-62570111 Screening Compounds and Building Blocks
6-({[(6-methylimidazo[1,2-a]pyridin-2-yl)methyl]amino}methyl)-1,4-oxazepan-6-ol dihydrochloride (62570111)
ChemBridge特有类药化合物/先导化合物-62570111,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。
M4909 GSK2801 GSK2801 Epigenetic Reader Domain
GSK2801 is a selective bromodomains BAZ2A/B inhibitor with KD of 257 nM and 136 nM, respectively.
M15079 Recombinant Human NT-3 (E.coli) 重组人NT-3蛋白 (E.coli) Recombinant Proteins
Neurotrophin-3; NT-3; HDNF; Nerve Growth Factor 2
利用大肠杆菌表达系统制备了重组人神经营养因子-3,并表达了编码Tyr139-Thr257的目的基因。Accession #: P20783。









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