找到约 49 条 “Phe-Gly” 相关结果 (用时 0.109 秒)
目录号 | 产品名称 | 中文名称 | 靶点 |
---|---|---|---|
M5684
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Guaifenesin | 愈创甘油醚 | Others |
Guaiacol glyceryl ether; Guaiphenesin; Glycerol guaiacolate | |||
Guaifenesin (愈创木酚甘油醚) 是化痰剂,可松弛肌肉。 | |||
M6021
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Vitamin E-TPGS (Tocofersolan) | 托可索伦;维生素E聚乙二醇琥珀酸酯 | Vitamin |
D-α-Tocopherol polyethylene glycol 1000 succinate; TPGS; Vitamin E-TPGS | |||
Vitamin E-TPGS(维生素E聚乙二醇琥珀酸酯,托可索伦)是维生素E的水溶性衍生物,既含有维生素E亲酯基团,又含有聚乙二醇亲水长链,因而具有较好的表面活性剂性质和水溶性,广泛应用于制剂的研究中,作为增溶剂、吸收促进剂、乳化剂、增塑剂以及水难溶性或脂溶性药物传递系统的载体,如固体分散体、眼部给药的载体、鼻腔内给药的载体等。 | |||
M10565
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Kisspeptin-10, human TFA | 亲吻促动素-10(人源)三氟乙酸盐 | Peptides |
KP-10; Tyr-Asn-Trp-Asn-Ser-Phe-Gly-Leu-Arg-Phe-NH2 | |||
Kisspeptin-10, human TFA 是一种有效的血管收缩剂和血管生成抑制剂,它通过其受体 GPR54 来抑制肿瘤转移作用。Kisspeptin-10/GPR54 信号通过 NFATc4 介导的 BMP2 表达来诱导成骨细胞分化。 | |||
M12591 | ChemBridge-6146494 | ChemBridge化合物-6146494 | Screening Compounds and Building Blocks |
N-[3-(3-bromophenyl)-2-(2-furoylamino)acryloyl]glycine (6146494) | |||
ChemBridge特有类药化合物/先导化合物-6146494,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M12625 | ChemBridge-6220207 | ChemBridge化合物-6220207 | Screening Compounds and Building Blocks |
N~1~-(2-bromophenyl)-N~2~-(4-ethoxyphenyl)-N~2~-(methylsulfonyl)glycinamide (6220207) | |||
ChemBridge特有类药化合物/先导化合物-6220207,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M12671 | ChemBridge-6402712 | ChemBridge化合物-6402712 | Screening Compounds and Building Blocks |
N~1~-cyclopropyl-N~2~-(4-ethoxyphenyl)-N~2~-[(4-methylphenyl)sulfonyl]glycinamide (6402712) | |||
ChemBridge特有类药化合物/先导化合物-6402712,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M12768 | ChemBridge-6723028 | ChemBridge化合物-6723028 | Screening Compounds and Building Blocks |
ethyl 2-{[N-(2,3-dimethylphenyl)-N-(phenylsulfonyl)glycyl]amino}benzoate (6723028) | |||
ChemBridge特有类药化合物/先导化合物-6723028,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M12771 | ChemBridge-6739985 | ChemBridge化合物-6739985 | Screening Compounds and Building Blocks |
methyl 2-({N-(2-methoxyphenyl)-N-[(4-methylphenyl)sulfonyl]glycyl}amino)benzoate (6739985) | |||
ChemBridge特有类药化合物/先导化合物-6739985,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M12782 | ChemBridge-6809058 | ChemBridge化合物-6809058 | Screening Compounds and Building Blocks |
N-[4-(methylsulfonyl)-2-nitrophenyl]glycine (6809058) | |||
ChemBridge特有类药化合物/先导化合物-6809058,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M12905 | ChemBridge-7361080 | ChemBridge化合物-7361080 | Screening Compounds and Building Blocks |
N-cyclohexyl-N-[(4-fluorophenyl)sulfonyl]glycine (7361080) | |||
ChemBridge特有类药化合物/先导化合物-7361080,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M12939 | ChemBridge-7579232 | ChemBridge化合物-7579232 | Screening Compounds and Building Blocks |
N~1~-(4-fluorophenyl)-N~2~-(4-methoxyphenyl)glycinamide (7579232) | |||
ChemBridge特有类药化合物/先导化合物-7579232,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M13002 | ChemBridge-7791502 | ChemBridge化合物-7791502 | Screening Compounds and Building Blocks |
N~2~-(5-chloro-2-methoxyphenyl)-N~2~-(methylsulfonyl)-N~1~-[4-(1-pyrrolidinylsulfonyl)phenyl]glycinamide (7791502) | |||
ChemBridge特有类药化合物/先导化合物-7791502,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M13013 | ChemBridge-7818994 | ChemBridge化合物-7818994 | Screening Compounds and Building Blocks |
N~2~-(5-chloro-2-methylphenyl)-N~1~-(2,6-difluorophenyl)-N~2~-(methylsulfonyl)glycinamide (7818994) | |||
ChemBridge特有类药化合物/先导化合物-7818994,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M15091
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2-(2-Phenylacetamido)acetic acid | 2-(2-Phenylacetamido)acetic acid | Metabolite/Endogenous Metabolite |
Phenaceturic Acid; Phenacetylglycine | |||
2-(2-Phenylacetamido)acetic acid 是一种内源性代谢产物。 | |||
M20485 | Phenylglyoxal hydrate | Phenylglyoxal hydrate | Dehydrogenase |
1-Phenylethanedione hydrate | |||
Phenylglyoxal is a potent inhibitor of mitochondrial aldehyde dehydrogenase. It reacts with arginine residues in purified Hageman factor (HF, Factor XII) and causes inhibition of its coagulant properties. | |||
M30430 | N-[3-(2-Furyl)acryloyl]-Phe-Gly-Gly | N-[3-(2-Furyl)acryloyl]-Phe-Gly-Gly | ACE |
FAPGG | |||
N-[3-(2-Furyl)acryloyl]-Phe-Gly-Gly (FAPGG) 是一种合成的用于血管紧张素转换酶 (ACE) 测定的显色底物。 | |||
M38897 | (-)-Phenylglycinol | (-)-Phenylglycinol | Others |
(-)-Phenylglycinol 是一种生化试剂,可作为生物材料或有机化合物,用于生命科学相关研究。 | |||
M39103 | 2-Phenylglycine | 2-Phenylglycine | Metabolite/Endogenous Metabolite |
2-Phenylglycine (DL-α-Phenylglycine) 是在 W2 至 W4 泌乳期间母乳中的代谢产物。 | |||
M39278 | (S)-(+)-2-Phenylglycine methyl ester hydrochloride | (S)-(+)-2-苯甘氨酸甲酯 盐酸盐 | Amino Acid Derivatives |
(S)-(+)-2-Phenylglycine methyl ester hydrochloride 是一种甘氨酸衍生物。 | |||
M39354 | N-(4-Cyanophenyl)glycine | N-(4-Cyanophenyl)glycine | Amino Acid Derivatives |
N-(4-Cyanophenyl)glycine 是一种甘氨酸衍生物。 | |||
M39370 | 2-Chlorophenylglycine | 2-Chlorophenylglycine | Amino Acid Derivatives |
2-Chlorophenylglycine 是一种甘氨酸衍生物。 | |||
M39580 | (S)-(+)-2-Phenylglycinol | (S)-(+)-2-Phenylglycinol | Others |
(S)-(+)-2-Phenylglycinol 是一种生化试剂,可作为生物材料或有机化合物,用于生命科学相关研究。 | |||
M39728 | D-4-Hydroxyphenylglycine | D-4-Hydroxyphenylglycine | Others |
D-4-Hydroxyphenylglycine (D-(-)-4-Hydroxyphenylglycine) 是生产半合成 β-内酰胺类抗生素的最重要原料之一,例如阿莫西林 和头孢羟氨苄。 | |||
M42369 | 3-Methoxy-4-hydroxyphenylglycol | 3-Methoxy-4-hydroxyphenylglycol | Metabolite/Endogenous Metabolite |
3-Methoxy-4-hydroxyphenylglycol (HMPG) 是大脑中去甲肾上腺素降解的代谢产物。 | |||
M42890 | Ethyl phenylglyoxylate | Ethyl phenylglyoxylate | Others |
Ethyl phenylglyoxylate (Ethyl benzoylformate; Phenylglyoxylic acid ethyl ester)是苯乙醛酸的乙酯,用作合成试剂。 | |||
M44059 | Cyclo(Phe-Gly) | 环(苯丙氨酸-甘氨酸)二肽 | Others |
环(苯丙氨酸-甘氨酸)二肽 | |||
M45637 | ChemBridge-5634520 | ChemBridge化合物-5634520 | Screening Compounds and Building Blocks |
methyl N-(4-methylphenyl)-N-(methylsulfonyl)glycinate (5634520) | |||
ChemBridge特有类药化合物/先导化合物-5634520,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M45776 | ChemBridge-6012256 | ChemBridge化合物-6012256 | Screening Compounds and Building Blocks |
N~1~-cyclopentyl-N~2~-(3,4-dimethoxyphenyl)-N~2~-[(4-methylphenyl)sulfonyl]glycinamide (6012256) | |||
ChemBridge特有类药化合物/先导化合物-6012256,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M45845 | ChemBridge-6187162 | ChemBridge化合物-6187162 | Screening Compounds and Building Blocks |
N~1~-cyclopentyl-N~2~-(3-methoxyphenyl)-N~2~-(phenylsulfonyl)glycinamide (6187162) | |||
ChemBridge特有类药化合物/先导化合物-6187162,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M45859 | ChemBridge-6226431 | ChemBridge化合物-6226431 | Screening Compounds and Building Blocks |
methyl N-(2-ethylphenyl)-N-(methylsulfonyl)glycinate (6226431) | |||
ChemBridge特有类药化合物/先导化合物-6226431,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M13354
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Angiopep-2 TFA | Angiopep-2 TFA | Peptides |
Angiopep-2 TFA 是脑肽载体。抗肿瘤化合物与 Angiopep-2 肽载体的结合可提高其在脑癌中的活性。 氨基酸序列号:Thr-Phe-Phe-Tyr-Gly-Gly-Ser-Arg-Gly-Lys-Arg-Asn-Asn-Phe-Lys-Thr-Glu-Glu-Tyr | |||
M13445
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Peripheral Myelin P0 Protein (180-199), mouse | Peripheral Myelin P0 Protein (180-199), mouse | Peptides |
Peripheral Myelin P0 Protein (180-199), mouse 是一种神经原性肽,是鼠类外周神经髓磷脂的纯化成分。 序列:Ser-Ser-Lys-Arg-Gly-Arg-Gln-Thr-Pro-Val-Leu-Tyr-Ala-Met-Leu-Asp-His-Ser-Arg-Ser | |||
M14157
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D-JNKI-1 | D-JNKI-1 | JNK |
AM-111; XG-102; Brimapitide | |||
D-JNKI-1 (AM-111) 是高效可渗透细胞的 JNK 抑制剂。序列: Asp-Gln-Ser-Arg-Pro-Val-Gln-Pro-Phe-Leu-Asn-Leu-Thr-Thr-Pro-Arg-Lys-Pro-Arg-Pro-Pro-Arg-Arg-Arg-Gln-Arg-Arg-Lys-Lys-Arg-Gly-NH2。 | |||
M15099
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Tat-beclin 1 | Tat-beclin 1 | Autophagy |
Tat-BECN1 | |||
Tat-beclin 1 是一种自噬蛋白区域 (beclin 1) 衍生的肽,是自噬 (autophagy) 的有效诱导剂,能够通过动员内源性Beclin 1刺激自噬。 序列:Tyr-Gly-Arg-Lys-Lys-Arg-Arg-Gln-Arg-Arg-Arg-Gly-Gly-Thr-Asn-Val-Phe-Asn-Ala-Thr-Phe-Glu-Ile-Trp-His-Asp-Gly-Glu-Phe-Gly-Thr | |||
M19934
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Penicillin V potassium salt | Penicillin V potassium salt | Antibiotic |
Phenoxymethylpenicillin potassium salt | |||
Phenoxymethylpenicillin, also known as penicillin V, is an antibiotic useful for the treatment of a number of bacterial infections. It acts by inhibiting the biosynthesis of cell-wall peptidoglycan. | |||
M19949
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Phloracetophenone | Phloracetophenone | Cytochrome P450 (e.g. CYP17) |
2,4,6-trihydroxyacetophenone | |||
Phloracetophenone, or 2,4,6-trihydroxyacetophenone (THA), the aglycone component of phloracetophenone glucoside, is a naturally occurring compound obtained from the rhizome of Curcuma comosa (Family Zingiberaceae). | |||
M20005
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TAT-DEF-Elk-1 TFA | TAT-DEF-Elk-1 TFA | Peptides |
TDE TFA | |||
TAT-DEF-Elk-1 TFA (TDE TFA) 是一种 Elk-1 的可穿透细胞的肽抑制剂,通过模仿和特异性干扰 Elk-1 的 DEF 结构域来实现抑制。序列:Gly-Arg-Lys-Lys-Arg-Arg-Gln-Arg-Arg-Arg-Pro-Pro-Ser-Pro-Ala-Lys-Leu-Ser-Phe-Gln-Phe-Pro-Ser-Ser-Gly-Ser-Ala-Gln-Val-His-Ile。 | |||
M20820
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Gly-Phe β-naphthylamide | Gly-Phe β-naphthylamide | Others |
Gly-Phe beta-naphthylamide | |||
Gly-Phe β-naphthylamide (Gly-Phe beta-naphthylamide) is a substrate of cathepsin C that accumulates within the lysosome. Gly-Phe-β-naphthylamide can inhibit the cathepsin-dependent activation of caspase-8. | |||
M21001 | Glycerol phenylbutyrate | Glycerol phenylbutyrate | Others |
GT4P, HPN-100M, Ravicti | |||
Glycerol phenylbutyrate (GT4P, HPN-100M, Ravicti) is a nitrogen-binding agent and acts as a sigma-2 (σ2) receptor ligand with a pKi of 8.02. Glycerol phenylbutyrate is a prodrug in which phenylbutyrate (PBA) is released from the glycerol backbone by lipases in the gastrointestinal tract. | |||
M21324
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β-Casomorphin, bovine acetate | β-Casomorphin, bovine acetate | Opioid Receptor |
β-Casomorphin-7 (bovine); Bovine β-casomorphin-7 acetate | |||
β-casomorphin, bovine (β-Casomorphin-7 (bovine) ) acetate是阿片 (opioid) 活性的多肽,与阿片受体结合的 IC50 值为 14 μM。序列:Tyr-Pro-Phe-Pro-Gly-Pro-Ile。 | |||
M31356
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Iberiotoxin TFA | Iberiotoxin TFA | Potassium Channel |
Iberiotoxin TFA是一种选择性的,高亲和力的大电导钙激活的钾通道(BKCa)的阻断剂,Kd约为 1 nM。序列号:Glp-Phe-Thr-Asp-Val-Asp-Cys-Ser-Val-Ser-Lys-Glu-Cys-Trp-Ser-Val-Cys-Lys-Asp-Leu-Phe-GlyVal-Asp-Arg-Gly-Lys-Cys-Met-Gly-Lys-Lys-Cys-Arg-Cys-Tyr-Gln(Cys7&Cys28,Cys13&Cys33,Cys17&Cys35 bridge) | |||
M39037 | Phellamurin | Phellamurin | P-glycoprotein |
Phellamurin 是一种来自 Phellodendron amurense 叶的植物黄酮糖苷,可抑制肠道 P-糖蛋白 (P-glycoprotein)。Phellamurin 还抑制凤蝶的产卵。 | |||
M39457 | H-Phg(4-Cl)-OH | H-Phg(4-Cl)-OH | Amino Acid Derivatives |
H-Phg(4-Cl)-OH (L-4-Chlorophenylglycine) 是一种甘氨酸衍生物。 | |||
M39815 | Oxfenicine | Oxfenicine | Others |
Oxfenicine (L-p-Hydroxyphenylglycine) 是一种具有口服活性的肉碱棕榈酰转移酶-1 抑制剂。Oxfenicine 可抑制心脏中脂肪酸的氧化。 | |||
M40644
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PreScission Protease | PreScission Protease | Enzymes & Coenzymes |
HRV 3C Protease; HRV3C Protease | |||
PreScission Protease是一种大肠杆菌中重组表达的带GST标签的人鼻病毒14型的3C蛋白酶,能在低温条件下(4°C)特异性地识别八肽序列Leu-Glu-Val-Leu-Phe-Gln-Gly-Pro或核心五肽序列Leu-Phe-Gln-Gly-Pro,并在Gln和Gly氨基酸残基之间进行酶切,常用于去除融合蛋白的Glutathione S-transferase (GST)、His或者其它标签。 | |||
M49888 | 4-Hydroxy-3-methoxyphenylglycol sulfate potassium salt | 4-羟基-3-甲氧基苯基乙二醇-4-硫酸钾盐 | Others |
4-Hydroxy-3-methoxyphenylglycol sulfate potassium salt | |||
M50838 | Phe-Arg-Arg-Gly | Phe-Arg-Arg-Gly | Others |
Phe-Arg-Arg-Gly 是一种可用于活性分子偶联的多肽。 | |||
M51296 | Gly-Phe-Gly-Aldehyde semicarbazone | Gly-Phe-Gly-Aldehyde semicarbazone | Others |
Gly-Phe-Gly-Aldehyde semicarbazone 是一种多肽。 | |||
M51329 | Acetylarginyltryptophyl diphenylglycine | Acetylarginyltryptophyl diphenylglycine | Others |
Acetylarginyltryptophyl diphenylglycine 是一种具有抗衰老(anti-aging)作用的生物活性肽,已被报道用作化妆品成分。 |