找到约 31 条 “PYR-41” 相关结果 (用时 0.213 秒)
目录号 | 产品名称 | 中文名称 | 靶点 |
---|---|---|---|
M2969
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PYR-41 | PYR-41 | E1/E2/E3 Enzyme |
PYR-41是一种可渗透细胞的吡唑酮化合物,不可逆地抑制泛素激活酶E1的活性,对E2无活性。 | |||
M9180
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Pyridostatin Trifluoroacetate Salt | Pyridostatin Trifluoroacetate Salt | DNA/RNA Synthesis |
Pyridostatin TFA salt; PDS; CAS# 1085412-37-8(free base) | |||
Pyridostatin Trifluoroacetate Salt是一种G-quadruplexe稳定剂,无细胞试验中Kd为490 nM。Pyridostatin Trifluoroacetate Salt可以促进DNA双链断裂(DSB)的形成。 | |||
M11560 | ChemBridge-4004241 | ChemBridge化合物-4004241 | Screening Compounds and Building Blocks |
3-pyridin-2-ylpropanoic acid (4004241) | |||
ChemBridge特有类药化合物/先导化合物-4004241,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M11606 | ChemBridge-5107414 | ChemBridge化合物-5107414 | Screening Compounds and Building Blocks |
5-ethoxy-1-(4-nitrophenyl)-3-phenyl-4,5-dihydro-1H-pyrazole (5107414) | |||
ChemBridge特有类药化合物/先导化合物-5107414,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M11697 | ChemBridge-5141565 | ChemBridge化合物-5141565 | Screening Compounds and Building Blocks |
4-amino-1-[6-(hydroxymethyl)-2-oxidotetrahydrofuro[3,4-d][1,3,2]dioxathiol-4-yl]-2(1H)-pyrimidinone hydrochloride (5141565) | |||
ChemBridge特有类药化合物/先导化合物-5141565,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M11834 | ChemBridge-5215341 | ChemBridge化合物-5215341 | Screening Compounds and Building Blocks |
1,1'-(1,2-phenylene)bis(1H-pyrrole-2,5-dione) (5215341) | |||
ChemBridge特有类药化合物/先导化合物-5215341,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M11899 | ChemBridge-5241292 | ChemBridge化合物-5241292 | Screening Compounds and Building Blocks |
2-(benzylthio)-5-(diphenylmethyl)-6-hydroxy-4(1H)-pyrimidinone (5241292) | |||
ChemBridge特有类药化合物/先导化合物-5241292,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M11968 | ChemBridge-5304192 | ChemBridge化合物-5304192 | Screening Compounds and Building Blocks |
5-methyl-4-{[(4-nitrophenyl)amino]methylene}-2-phenyl-2,4-dihydro-3H-pyrazole-3-thione (5304192) | |||
ChemBridge特有类药化合物/先导化合物-5304192,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M11975 | ChemBridge-5310341 | ChemBridge化合物-5310341 | Screening Compounds and Building Blocks |
4-[(5-chloro-2-pyridinyl)amino]-4-oxobutanoic acid (5310341) | |||
ChemBridge特有类药化合物/先导化合物-5310341,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M12193 | ChemBridge-5631437 | ChemBridge化合物-5631437 | Screening Compounds and Building Blocks |
ethyl 4-{4-[(5-nitro-2-furyl)methylene]-3,5-dioxo-1-pyrazolidinyl}benzoate (5631437) | |||
ChemBridge特有类药化合物/先导化合物-5631437,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M12265 | ChemBridge-5674122 | ChemBridge化合物-5674122 | Screening Compounds and Building Blocks |
2-benzyl-3-(4-chlorophenyl)-5-(4-nitrophenyl)pyrazolo[1,5-a]pyrimidin-7(4H)-one (5674122) | |||
ChemBridge特有类药化合物/先导化合物-5674122,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M12470 | ChemBridge-5965041 | ChemBridge化合物-5965041 | Screening Compounds and Building Blocks |
5-(2,5-dimethyl-1H-pyrrol-1-yl)-2-hydroxybenzoic acid (5965041) | |||
ChemBridge特有类药化合物/先导化合物-5965041,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M12538 | ChemBridge-6048841 | ChemBridge化合物-6048841 | Screening Compounds and Building Blocks |
cyclopentyl 1,6-dimethyl-4-(6-nitro-1,3-benzodioxol-5-yl)-2-oxo-1,2,3,4-tetrahydro-5-pyrimidinecarboxylate (6048841) | |||
ChemBridge特有类药化合物/先导化合物-6048841,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M12563 | ChemBridge-6092141 | ChemBridge化合物-6092141 | Screening Compounds and Building Blocks |
2-thioxo-5-[(1,2,5-trimethyl-1H-pyrrol-3-yl)methylene]-1,3-thiazolidin-4-one (6092141) | |||
ChemBridge特有类药化合物/先导化合物-6092141,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M12586 | ChemBridge-6141194 | ChemBridge化合物-6141194 | Screening Compounds and Building Blocks |
3,3'-({4-methoxy-3-[(2-pyridinylthio)methyl]phenyl}methylene)bis(4-hydroxy-2H-chromen-2-one) (6141194) | |||
ChemBridge特有类药化合物/先导化合物-6141194,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M12614 | ChemBridge-6194143 | ChemBridge化合物-6194143 | Screening Compounds and Building Blocks |
N-(5-chloro-2-pyridinyl)-4-propoxybenzamide (6194143) | |||
ChemBridge特有类药化合物/先导化合物-6194143,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M13007 | ChemBridge-7799415 | ChemBridge化合物-7799415 | Screening Compounds and Building Blocks |
2-[5-(2-naphthyl)-1,2,4-oxadiazol-3-yl]pyridine (7799415) | |||
ChemBridge特有类药化合物/先导化合物-7799415,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M13092 | ChemBridge-7941261 | ChemBridge化合物-7941261 | Screening Compounds and Building Blocks |
4-{[(4-methylphenyl)thio]methyl}-N-(3-pyridinylmethyl)benzamide (7941261) | |||
ChemBridge特有类药化合物/先导化合物-7941261,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M13143 | ChemBridge-7994941 | ChemBridge化合物-7994941 | Screening Compounds and Building Blocks |
5-amino-7-isopropyl-2-phenyl-4,7-dihydro[1,3]oxazolo[5,4-b]pyridine-6-carbonitrile (7994941) | |||
ChemBridge特有类药化合物/先导化合物-7994941,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M13144 | ChemBridge-7995441 | ChemBridge化合物-7995441 | Screening Compounds and Building Blocks |
4,5-dichloro-2-(2-methylphenyl)-3(2H)-pyridazinone (7995441) | |||
ChemBridge特有类药化合物/先导化合物-7995441,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M13189 | ChemBridge-9041014 | ChemBridge化合物-9041014 | Screening Compounds and Building Blocks |
N-(3,4-dimethoxyphenyl)-6-phenylpyrimidin-4-amine (9041014) | |||
ChemBridge特有类药化合物/先导化合物-9041014,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M13270 | ChemBridge-34185989 | ChemBridge化合物-34185989 | Screening Compounds and Building Blocks |
methyl 5-[(1,5-dimethyl-4-hexen-1-yl)amino]-3-[(methoxyacetyl)amino]-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate (34185989) | |||
ChemBridge特有类药化合物/先导化合物-34185989,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M13277 | ChemBridge-39124139 | ChemBridge化合物-39124139 | Screening Compounds and Building Blocks |
N-{2-[methyl(methylsulfonyl)amino]ethyl}-5-phenyl-1H-pyrrole-2-carboxamide (39124139) | |||
ChemBridge特有类药化合物/先导化合物-39124139,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M13279 | ChemBridge-41107369 | ChemBridge化合物-41107369 | Screening Compounds and Building Blocks |
4-[(3-cyclobutyl-1,4,6,7-tetrahydro-5H-pyrazolo[4,3-c]pyridin-5-yl)carbonyl]-3a,4,5,9b-tetrahydro-3H-cyclopenta[c]quinoline (41107369) | |||
ChemBridge特有类药化合物/先导化合物-41107369,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M13316 | ChemBridge-81412635 | ChemBridge化合物-81412635 | Screening Compounds and Building Blocks |
methyl 2-[(diethylamino)sulfonyl]-6-[(1,3-dimethyl-1H-pyrazol-5-yl)carbonyl]-4,5,6,7-tetrahydrothieno[2,3-c]pyridine-3-carboxylate (81412635) | |||
ChemBridge特有类药化合物/先导化合物-81412635,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M13334 | ChemBridge-99441193 | ChemBridge化合物-99441193 | Screening Compounds and Building Blocks |
N-{[1-(1H-imidazol-4-ylmethyl)pyrrolidin-3-yl]methyl}-8-methylimidazo[1,2-a]pyridine-2-carboxamide (99441193) | |||
ChemBridge特有类药化合物/先导化合物-99441193,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M40504
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ChemBridge-23475241 | ChemBridge化合物-23475241 | Screening Compounds and Building Blocks |
1-ethyl-N-(4-methoxybenzyl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridine-3-carboxamide(23475241) | |||
ChemBridge热销化合物 23475241 | |||
M45409 | ChemBridge-4004174 | ChemBridge化合物-4004174 | Screening Compounds and Building Blocks |
3-isobutyl-1-methyl-1H-pyrazole-5-carboxylic acid (4004174) | |||
ChemBridge特有类药化合物/先导化合物-4004174,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M45504 | ChemBridge-5224144 | ChemBridge化合物-5224144 | Screening Compounds and Building Blocks |
3-(4-{[1,3-dioxo-2-(2-pyridinyl)-2,3-dihydro-1H-isoindol-5-yl]oxy}phenoxy)benzoic acid (5224144) | |||
ChemBridge特有类药化合物/先导化合物-5224144,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M45517 | ChemBridge-5241078 | ChemBridge化合物-5241078 | Screening Compounds and Building Blocks |
1-benzyl-5-({[2-hydroxy-1-(hydroxymethyl)-1-methylethyl]amino}methylene)-2,4,6(1H,3H,5H)-pyrimidinetrione (5241078) | |||
ChemBridge特有类药化合物/先导化合物-5241078,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M40154 | 5,7,3',4'-Tetrahydroxy-3-methoxy-8,5'-diprenylflavone | 5,7,3',4'-Tetrahydroxy-3-methoxy-8,5'-diprenylflavone | Others |
5,7,3',4'-Tetrahydroxy-3-methoxy-8,5'-diprenylflavone 是一种天然产物,可从 B. papyrifera 中提取。5,7,3',4'-Tetrahydroxy-3-methoxy-8,5'-diprenylflavone 对 ER 阳性乳腺癌细胞具有有效的抗增殖作用,对 MCF-7 细胞 IC50 为 4.41 μM。 |