找到约 14 条 “PR-104” 相关结果 (用时 0.203 秒)
目录号 | 产品名称 | 中文名称 | 靶点 |
---|---|---|---|
M25447 | PR-104 | DNA交联剂 | DNA/RNA Synthesis |
PR-104是一种新型的缺氧激活的DNA交联剂,对人肿瘤异种移植物有明显的活性,可用于异种肿瘤模型的研究。 | |||
M3229
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PR-104A | PR-104A | DNA/RNA Synthesis |
PR-104A(SN 27858)是一种低氧激活的前体药物 (HAP),通过将一个硝基基团还原成相应的羟胺(PR-104H)或胺(PR-104M)来激活DNA烷基化作用,具有抗癌活性。 | |||
M3768
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Ixabepilone | 伊沙匹隆 | Microtubule |
Ixempra, BMS-247550, NSC 710428 | |||
Ixabepilone (BMS 247550)是epothilone B类似物,同时也是一种大环类化合物,具有稳定微管的作用。 | |||
M12384 | ChemBridge-5831049 | ChemBridge化合物-5831049 | Screening Compounds and Building Blocks |
N-[3-(diethylamino)propyl]-5-(4-methylphenyl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide (5831049) | |||
ChemBridge特有类药化合物/先导化合物-5831049,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M13230 | ChemBridge-10467389 | ChemBridge化合物-10467389 | Screening Compounds and Building Blocks |
3-(1-piperidinylcarbonyl)-1-propyl-N-[2-(3-pyridinyl)ethyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine (10467389) | |||
ChemBridge特有类药化合物/先导化合物-10467389,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M45843 | ChemBridge-6181043 | ChemBridge化合物-6181043 | Screening Compounds and Building Blocks |
2-[(4-chlorobenzyl)thio]-N-isopropylacetamide (6181043) | |||
ChemBridge特有类药化合物/先导化合物-6181043,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M46613 | ChemBridge-8831048 | ChemBridge化合物-8831048 | Screening Compounds and Building Blocks |
N-(4-isopropylphenyl)-N'-(2-methoxy-5-methylphenyl)thiourea (8831048) | |||
ChemBridge特有类药化合物/先导化合物-8831048,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M47254 | ChemBridge-10436536 | ChemBridge化合物-10436536 | Screening Compounds and Building Blocks |
4-methyl-1-[3-(4-morpholinylcarbonyl)-1-(3-phenylpropyl)-1,4,6,7-tetrahydro-5H-pyrazolo[4,3-c]pyridin-5-yl]-1-oxo-2-pentanone (10436536) | |||
ChemBridge特有类药化合物/先导化合物-10436536,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M47279 | ChemBridge-11310451 | ChemBridge化合物-11310451 | Screening Compounds and Building Blocks |
1-(cyclopentylcarbonyl)-N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-4-piperidinecarboxamide (11310451) | |||
ChemBridge特有类药化合物/先导化合物-11310451,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M47975 | ChemBridge-37961041 | ChemBridge化合物-37961041 | Screening Compounds and Building Blocks |
1-[(5R)-5-phenyl-D-prolyl]-1',4'-dihydro-3'H-spiro[piperidine-4,2'-quinoxalin]-3'-one dihydrochloride (37961041) | |||
ChemBridge特有类药化合物/先导化合物-37961041,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M48644 | ChemBridge-66010402 | ChemBridge化合物-66010402 | Screening Compounds and Building Blocks |
2-isopropyl-N-[(1-propyl-1H-pyrazol-4-yl)methyl]-1,3-thiazole-4-carboxamide (66010402) | |||
ChemBridge特有类药化合物/先导化合物-66010402,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M48834 | ChemBridge-74710446 | ChemBridge化合物-74710446 | Screening Compounds and Building Blocks |
{3-(3-methyl-2-buten-1-yl)-1-[3-(1,3,5-trimethyl-1H-pyrazol-4-yl)propanoyl]-3-piperidinyl}methanol (74710446) | |||
ChemBridge特有类药化合物/先导化合物-74710446,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M49238 | ChemBridge-94341049 | ChemBridge化合物-94341049 | Screening Compounds and Building Blocks |
N-methyl-N-[2-(4-morpholinyl)propyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine (94341049) | |||
ChemBridge特有类药化合物/先导化合物-94341049,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M43539 | Protein kinase inhibitor 4 | Protein kinase inhibitor 4 | Trk |
Protein kinase inhibitor 4 是一种蛋白激酶抑制剂,可抑制 TRK-A 和 ROS1 (IC50 分别为 3.0 nM 和 104 nM)。 |