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 找到约 4 条 “PHD-IN-1” 相关结果 (用时 0.159 秒)

目录号 产品名称 中文名称 靶点
M42436 PHD2-IN-1 PHD2-IN-1 HIF
PHD2-IN-1 是一种强效的、具有口服活性的 HIF-脯氨酰羟化酶2 (PHD2) 抑制剂,IC50 为 22.53 nM,可用于贫血病研究。
M42439 PHD-IN-1 PHD-IN-1 HIF
PHD-IN-1 是一种有效的 PHD2 抑制剂,IC50 值 ≤5 nM。
M8467 OF-1 OF-1 Others
OF-1 is a chemical probe for the bromodomains of the BRPF (BRomodomain and PHD Finger containing) family of scaffolding proteins (BRPF1, BRPF2, BRPF3) that assemble histone acetyltransferase (HAT) complexes of the MYST family members MOZ and MORF.
M20749 TP0463518 TP0463518 HIF
TP0463518 is a potent hypoxia-inducible factor prolyl hydroxylases (PHDs) inhibitor with Ki of 5.3 nM for human PHD2. TP0463518 inhibits human PHD1, human PHD3 and monkey PHD2 with IC50 of 18 nM, 63 nM and 22 nM, respectively.









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