找到约 10 条 “Omeprazole” 相关结果 (用时 0.115 秒)
目录号 | 产品名称 | 中文名称 | 靶点 |
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M1834
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Omeprazole | 奥美拉唑 | Proton Pump |
H 16868; Omeprazol | |||
Omeprazole (H 16868) 是一种首创的(first-in-class)质子泵 (proton pump) 抑制剂 (PPI)。Omeprazole 竞争性抑制 CYP2C19 活性,Ki 为 2 到 6 μM。Omeprazole 还抑制革兰氏阳性菌和革兰氏阴性菌生长。 | |||
M3448
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Esomeprazole Sodium | 埃索美拉唑钠 | Proton Pump |
(S)-Omeprazole sodium | |||
Esomeprazole Sodium (埃索美拉唑钠)是Esomeprazole的一种钠盐,是有效的质子泵(Proton Pump)抑制剂,IC50为0.076 mg/kg。 | |||
M3575
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Esomeprazole Magnesium | 埃索美拉唑镁 | Proton Pump |
Esomeprazole magnesium ((S)-Omeprazole magnesium) 是一种有效的具有口服活性 H+, K+-ATPase 抑制剂,可用于上消化道疾病和胃食管反流疾病的研究。还可通过抑制 V-H+-ATPases 来抑制外泌体的释放。 | |||
M1583
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Omeprazole sulfone | 奥美拉唑砜 | Metabolite/Endogenous Metabolite |
Omeprazole sulfone; Omeprazole sulphone | |||
Omeprazole sulfone是Omeprazole的代谢物。 | |||
M6194
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Esomeprazole Magnesium trihydrate | 埃索美拉唑镁 | Autophagy |
(S)-Omeprazole magnesium trihydrate | |||
Esomeprazole镁盐三水合物是质子泵抑制剂,能通过抑制胃壁细胞中的H+/K+ ATPase来降低酸分泌。 | |||
M20514
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Omeprazole Sodium | Omeprazole Sodium | Proton Pump |
Omeprazole Sodium is the sodium salt form of omeprazole, which is a proton pump inhibitor and suppresses gastric acid secretion. | |||
M20570
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Ufiprazole | Ufiprazole | Others |
Omeprazole sulfide | |||
Ufiprazole (Omeprazole sulfide) is an intermediate used in the production of the gastric proton pump inhibitors omeprazole and esomeprazole. | |||
M22268 | Esomeprazole potassium salt | Esomeprazole potassium salt | Others |
Esomeprazole potassium salt | |||
M22284 | Esomeprazole magnesium salt | Esomeprazole magnesium salt | Others |
Esomeprazole magnesium salt | |||
M55502
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Esomeprazole-d3 sodium | 埃索美拉唑-D3钠盐 | Proton Pump |
埃索美拉唑-D3钠盐 Esomeprazole-d3 sodium |