找到约 19 条 “MIN-101” 相关结果 (用时 0.108 秒)
目录号 | 产品名称 | 中文名称 | 靶点 |
---|---|---|---|
M5928
![]() |
Riboflavin | 维生素B2 | Vitamin |
Vitamin B2; E101 | |||
Riboflavin 是一种易被吸收的微量营养素,对维持人和其他动物的健康起到了关键作用。 | |||
M7339
![]() |
Texas Red (Sulforhodamine 101) | 磺基罗丹明 101 | Fluorescent Dye |
Sulforhodamine 101; SR101 | |||
Texas Red (磺基罗丹明 101;Sulforhodamine 101) 是一种两性罗丹明红色荧光染料 (excitation/emission: 586/605 nm)。Texas Red 被广泛用于研究神经元形态,并作为星形胶质细胞的细胞类型选择性荧光标记物,在体内和切片制备中都有应用。 | |||
M8955
![]() |
MIN-101 | MIN-101 | 5-HT Receptor |
Roluperidone; CYR-101 | |||
MIN-101 (Roluperidone)是一种新型化合物,同时也是5-HT2A和sigma-2受体的拮抗剂,对5-HT2A和sigma-2受体的Ki值分别为 7.53 nM 和 8.19 nM。此外,MIN-101还能抑制α-肾上腺素能受体的活性。 | |||
M11583 | ChemBridge-5101031 | ChemBridge化合物-5101031 | Screening Compounds and Building Blocks |
N-(4-nitrophenyl)-N'-pentyl-6-(2,2,2-trifluoroethoxy)-1,3,5-triazine-2,4-diamine (5101031) | |||
ChemBridge特有类药化合物/先导化合物-5101031,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M11584 | ChemBridge-5101039 | ChemBridge化合物-5101039 | Screening Compounds and Building Blocks |
N-methyl-N'-(4-nitrophenyl)-6-(2,2,2-trifluoroethoxy)-1,3,5-triazine-2,4-diamine (5101039) | |||
ChemBridge特有类药化合物/先导化合物-5101039,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M12886 | ChemBridge-7221014 | ChemBridge化合物-7221014 | Screening Compounds and Building Blocks |
2-[(2-phenylbutanoyl)amino]-4,5,6,7,8,9-hexahydrocycloocta[b]thiophene-3-carboxamide (7221014) | |||
ChemBridge特有类药化合物/先导化合物-7221014,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M13189 | ChemBridge-9041014 | ChemBridge化合物-9041014 | Screening Compounds and Building Blocks |
N-(3,4-dimethoxyphenyl)-6-phenylpyrimidin-4-amine (9041014) | |||
ChemBridge特有类药化合物/先导化合物-9041014,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M40744
![]() |
Rhodamine 101 chloride | 氯化罗丹明 101 | Fluorescent Dye |
Rhodamine 101 chloride是一种荧光染料,激发和发射波长最大值分别为 565 nM 和 595 nM。 | |||
M45816 | ChemBridge-6101682 | ChemBridge化合物-6101682 | Screening Compounds and Building Blocks |
2-amino-7-(4-methylphenyl)-7,8-dihydro-5(6H)-quinazolinone (6101682) | |||
ChemBridge特有类药化合物/先导化合物-6101682,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M46043 | ChemBridge-7002101 | ChemBridge化合物-7002101 | Screening Compounds and Building Blocks |
N-{2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}-1-butanamine oxalate (7002101) | |||
ChemBridge特有类药化合物/先导化合物-7002101,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M47252 | ChemBridge-10198243 | ChemBridge化合物-10198243 | Screening Compounds and Building Blocks |
methyl 6-{[(2-methyl-7,8-dihydro-4H-pyrazolo[1,5-a][1,4]diazepin-5(6H)-yl)carbonyl]amino}-3,4-dihydroquinoline-1(2H)-carboxylate (10198243) | |||
ChemBridge特有类药化合物/先导化合物-10198243,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M47274 | ChemBridge-11015072 | ChemBridge化合物-11015072 | Screening Compounds and Building Blocks |
2-amino-N-[(5-isobutyl-1,2,4-oxadiazol-3-yl)methyl]-1,3-thiazole-4-carboxamide (11015072) | |||
ChemBridge特有类药化合物/先导化合物-11015072,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M47544 | ChemBridge-21018625 | ChemBridge化合物-21018625 | Screening Compounds and Building Blocks |
3-(4-aminopyridin-3-yl)-N-(3-azepan-1-ylpropyl)-N-methylbenzamide (21018625) | |||
ChemBridge特有类药化合物/先导化合物-21018625,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M48239 | ChemBridge-49101166 | ChemBridge化合物-49101166 | Screening Compounds and Building Blocks |
methyl 3-({[(3-methyl-1H-1,2,4-triazol-5-yl)acetyl]amino}methyl)-5-{[(2E)-3-phenyl-2-propenoyl]amino}benzoate (49101166) | |||
ChemBridge特有类药化合物/先导化合物-49101166,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M48504 | ChemBridge-60010133 | ChemBridge化合物-60010133 | Screening Compounds and Building Blocks |
3-[2-(3-fluorophenyl)ethyl]-7-{methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4(3H)-one (60010133) | |||
ChemBridge特有类药化合物/先导化合物-60010133,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M50045 | ChemBridge-81011449 | ChemBridge化合物-81011449 | Screening Compounds and Building Blocks |
1-amino-N-{2-[4-(2-furylmethyl)-2-morpholinyl]ethyl}cyclopentanecarboxamide dihydrochloride (81011449) | |||
ChemBridge特有类药化合物/先导化合物-81011449,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M50124 | ChemBridge-5210193 | ChemBridge化合物-5210193 | Screening Compounds and Building Blocks |
6-{[2-(acetylamino)-3-(1,3-benzodioxol-5-yl)acryloyl]amino}hexanoic acid (5210193) | |||
ChemBridge特有类药化合物/先导化合物-5210193,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M25441
![]() |
Recombinant Human Endothelin B Receptor Protein (HEK293, His Tag) | 重组人EDNRB蛋白 (HEK293, His Tag) | Cytokines and Growth Factors |
human EDNRB | |||
EDNRB is a new candidate tumor suppressor gene which is often down-regulated or even silenced by promoter hypermethylation in various human cancers. The recombinant human EDNRB consists 86 amino acids and predicts a molecular mass of 9.5 kDa. A DNA sequence encoding the human EDNRB (NP_000106.1) (Met1-Lys101) was expressed with a polyhistidine tag at the C-terminus. | |||
M30560 | JNJ10191584 | JNJ10191584 | Histamine Receptor |
VUF6002 | |||
JNJ10191584 (VUF6002) 是具有口服活性的、选择性的 histamine H4 受体 拮抗剂,Ki 值为 26 nM。JNJ10191584 对 H4 受体的选择性是 H3 受体的 540 倍,对 H3 受体的 Ki 值为 14.1 μM。JNJ10191584 抑制嗜酸性粒细胞和肥大细胞的趋化作用,IC50 值分别为 530 nM 和 138 nM。 |