找到约 7 条 “Kynurenic acid” 相关结果 (用时 0.105 秒)
目录号 | 产品名称 | 中文名称 | 靶点 |
---|---|---|---|
M6354 | 7-Chlorokynurenic acid | 7-Chlorokynurenic acid | Others |
7-氯核仁酸是l -谷氨酸吸收的强有力的竞争性抑制剂。 | |||
M6355
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7-Chlorokynurenic acid sodium salt | 7-Chlorokynurenic acid sodium salt | GluR |
7-氯核仁酸钠盐是l -谷氨酸吸收的一种强有力的竞争性抑制剂。7-氯核仁酸钠盐。 | |||
M7873
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Kynurenic acid | Kynurenic acid | Others |
Quinurenic acid | |||
Kynurenic acid 是一种内源性色氨酸代谢物,同时也是靶点 NMDA,glutamate,α7 nAChR的广谱性拮抗剂,以及GPR35/CXCR8 的激动剂。 | |||
M28153 | 5,7-Dichlorokynurenic acid | 5,7-二氯犬尿喹啉酸 | GluR |
5,7-DCKA | |||
5,7-Dichlorokynurenic acid (5,7-DCKA) 是一种选择性的 NMDA 受体甘氨酸位点竞争性拮抗剂,KB 值为 65 nM。5,7-Dichlorokynurenic acid 是犬尿酸的衍生物,可减少大鼠皮质细胞培养物中 NMDA 诱导的神经元损伤。 | |||
M56493 | 5,7-Dichlorokynurenic acid sodium | 5,7-Dichlorokynurenic acid sodium | GluR |
5,7-Dichlorokynurenic acid (sodium) 是 5,7-Dichlorokynurenic acid 的钠盐形式。5,7-Dichlorokynurenic acid 是一种选择性的 NMDA 受体甘氨酸位点竞争性拮抗剂,KB 值为 65 nM。 | |||
M8246 | GPR35 Agonist, Compound 10 | GPR35 Agonist, Compound 10 | Others |
GPR35 agonist Compound 10 is a GPR35 agonist the binds with higher affinity than other known agonists, such as kynurenic acid and zaprinast. | |||
M8381 | JM6 | JM6 | Others |
JM6 is a prodrug inhibitor of kynurenine 3-monooxygenase (KMO) that increases kynurenic acid levels and reduces extracellular glutamate in the brain. |