找到约 7 条 “Kynurenic acid” 相关结果 (用时 0.105 秒)

目录号 产品名称 中文名称 靶点
M6354 7-Chlorokynurenic acid 7-Chlorokynurenic acid Others
7-氯核仁酸是l -谷氨酸吸收的强有力的竞争性抑制剂。
M6355 7-Chlorokynurenic acid sodium salt 7-Chlorokynurenic acid sodium salt GluR
7-氯核仁酸钠盐是l -谷氨酸吸收的一种强有力的竞争性抑制剂。7-氯核仁酸钠盐。
M7873 Kynurenic acid Kynurenic acid Others
Quinurenic acid
Kynurenic acid 是一种内源性色氨酸代谢物,同时也是靶点 NMDA,glutamate,α7 nAChR的广谱性拮抗剂,以及GPR35/CXCR8 的激动剂。
M28153 5,7-Dichlorokynurenic acid 5,7-二氯犬尿喹啉酸 GluR
5,7-DCKA
5,7-Dichlorokynurenic acid (5,7-DCKA) 是一种选择性的 NMDA 受体甘氨酸位点竞争性拮抗剂,KB 值为 65 nM。5,7-Dichlorokynurenic acid 是犬尿酸的衍生物,可减少大鼠皮质细胞培养物中 NMDA 诱导的神经元损伤。
M56493 5,7-Dichlorokynurenic acid sodium 5,7-Dichlorokynurenic acid sodium GluR
5,7-Dichlorokynurenic acid (sodium) 是 5,7-Dichlorokynurenic acid 的钠盐形式。5,7-Dichlorokynurenic acid 是一种选择性的 NMDA 受体甘氨酸位点竞争性拮抗剂,KB 值为 65 nM。
M8246 GPR35 Agonist, Compound 10 GPR35 Agonist, Compound 10 Others
GPR35 agonist Compound 10 is a GPR35 agonist the binds with higher affinity than other known agonists, such as kynurenic acid and zaprinast.
M8381 JM6 JM6 Others
JM6 is a prodrug inhibitor of kynurenine 3-monooxygenase (KMO) that increases kynurenic acid levels and reduces extracellular glutamate in the brain.








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