找到约 1 条 “K-(D-1-Nal)-FwLL-NH2 TFA ” 相关结果 (用时 0.195 秒)
目录号 | 产品名称 | 中文名称 | 靶点 |
---|---|---|---|
M31029 | K-(D-1-Nal)-FwLL-NH2 TFA | K-(D-1-Nal)-FwLL-NH2 TFA | Ghrelin Receptor/GHSR |
K-(D-1-Nal)-FwLL-NH2 TFA is a high affinity and potent ghrelin receptor inverse agonist (Ki values are 4.9 and 31 nM in COS7 and HEK293T cells, respectively). K-(D-1-Nal)-FwLL-NH2 blocks ghrelin receptor-mediated Gq- and G13-dependent signaling pathways. |