找到约 3 条 “Huwentoxin-IV” 相关结果 (用时 0.128 秒)
目录号 | 产品名称 | 中文名称 | 靶点 |
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M10458
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Huwentoxin IV TFA | Huwentoxin IV TFA | Sodium Channel |
Huwentoxin-IV | |||
Huwentoxin IV TFA 是一种有效的,选择性的钠通道阻滞剂,它抑制神经元 Nav1.7,Nav1.2,Nav1.3 和 Nav1.4的IC50 值分别为 26、150、338 和 400 nM。 | |||
M52722 | Huwentoxin-IV | Huwentoxin-IV | Sodium Channel |
Huwentoxin-IV 是一种有效的、选择性钠通道阻滞剂,可抑制神经元 Nav1.7,Nav1.2,Nav1.3 和 Nav1.4,IC50 值分别为 26、150、338 和 400 nM。 | |||
M58140 | HwTx-IV | HwTx-IV | Sodium Channel |
Huwentoxin-IV | |||
Huwentoxin-IV (HwTx-IV) is a 35-residue neurotoxin peptide with potential application as a novel analgesic. Huwentoxin-IV, a component of tarantula venom, potently blocks sodium channels and is an attractive scaffold for engineering a Nav1.7-selective molecule. |