找到约 5 条 “Huwentoxin I” 相关结果 （用时 0.445 秒）
| 目录号 | 产品名称 | 中文名称 | 靶点 |
|---|---|---|---|
M10458
|
Huwentoxin IV TFA | Huwentoxin IV TFA | Sodium Channel |
| Huwentoxin-IV | |||
| Huwentoxin IV TFA 是一种有效的，选择性的钠通道阻滞剂，它抑制神经元 Nav1.7，Nav1.2，Nav1.3 和 Nav1.4的IC50 值分别为 26、150、338 和 400 nM。 | |||
| M52722 | Huwentoxin-IV | Huwentoxin-IV | Sodium Channel |
| Huwentoxin-IV 是一种有效的、选择性钠通道阻滞剂，可抑制神经元 Nav1.7，Nav1.2，Nav1.3 和 Nav1.4，IC50 值分别为 26、150、338 和 400 nM。 | |||
| M52799 | Huwentoxin I | Huwentoxin I | Calcium Channel |
| Huwentoxin I (HWTX-I) 是一种肽毒素，可抑制电压门控钠通道和 N 型钙通道。 | |||
| M52802 | Huwentoxin XVI | Huwentoxin XVI | Calcium Channel |
| Huwentoxin XVI，一种来自鸟蛛 Ornithoctonus huwena 的止痛剂，一种高度可逆和选择性的哺乳动物 N 型钙通道 (N-type calcium channel) (IC50 约为 60 nM) 拮抗剂。 | |||
| M58140 | HwTx-IV | HwTx-IV | Sodium Channel |
| Huwentoxin-IV | |||
| Huwentoxin-IV (HwTx-IV) is a 35-residue neurotoxin peptide with potential application as a novel analgesic. Huwentoxin-IV, a component of tarantula venom, potently blocks sodium channels and is an attractive scaffold for engineering a Nav1.7-selective molecule. | |||
