找到约 4 条 “Glucagon Receptor Antagonist I” 相关结果 (用时 0.404 秒)
目录号 | 产品名称 | 中文名称 | 靶点 |
---|---|---|---|
M57829 | Glucagon Receptor Antagonist I | Glucagon Receptor Antagonist I | Others |
Glucagon Receptor Antagonist I | |||
M21377 | PF-06372222 | PF-06372222 | Others |
PF-06372222 is a small-molecule negative allosteric modulator of the glucagon receptor (GCGR). PF-06372222 is also an antagonist for glucagon-like peptide-1 receptor GLP-1R, which inhibits glucagon secretion and glucose-dependent insulin secretion. | |||
M13966
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Adomeglivant | 阿度格列凡 | Glucagon Receptor |
LY2409021 | |||
Adomeglivant (LY2409021) 是一种有效的选择性胰高血糖素受体 (GluR) 变构拮抗剂。Adomeglivant 广泛应用于 2 型糖尿病的研究。 | |||
M13971
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MK 0893 | MK 0893 | Glucagon Receptor |
MK 0893 是一种有效,选择性的胰高血糖素受体拮抗剂,IC50 值为 6.6 nM。 |