找到约 3 条 “GLUT inhibitor-1” 相关结果 （用时 0.103 秒）
| 目录号 | 产品名称 | 中文名称 | 靶点 |
|---|---|---|---|
M54563
|
GLUT inhibitor-1 | GLUT inhibitor-1 | GLUT |
| GLUT inhibitor-1是一种有效且具有口服活性的葡萄糖转运蛋白（GLUT）抑制剂，能靶向 GLUT1 和 GLUT3，其IC50值分别为 242 nM 和 179 nM。GLUT inhibitor-1可用于癌症和自身免疫性疾病的相关研究。 | |||
| M56801 | Glutaminyl Cyclase Inhibitor 1 | Glutaminyl Cyclase Inhibitor 1 | Amyloid |
| Glutaminyl Cyclase Inhibitor 1是谷氨酰胺酰基环化酶 (glutaminyl cyclase) 抑制剂，IC50 值为0.5 μM。 | |||
| M20864 | L-2-Hydroxyglutaric acid disodium | L-2-Hydroxyglutaric acid disodium | Histone demethylase |
| (S)-2-Hydroxyglutaric acid disodium, L-2-Hydroxyglutarate disodium, LGA, L-2HG | |||
| L-2-Hydroxyglutaric acid disodium ((S)-2-Hydroxyglutaric acid disodium, L-2-Hydroxyglutarate disodium, LGA, L-2HG) is an epigenetic modifier and a putative oncometabolite in kidney cancer that inhibits histone demethylases and hence promotes histone methylation. L-2-Hydroxyglutaric acid disodium is also an inhibitor of mitochondrial creatine kinase (Mi-CK) with Km and Ki of 2.52 mM and 11.13 mM, respectively. | |||
