找到约 31 条 “CG” 相关结果 （用时 0.044 秒）
| 目录号 | 产品名称 | 中文名称 | 靶点 |
|---|---|---|---|
| M6568 | CCG 2046 | CCG 2046 | Others |
| ccg2046是g蛋白信号转导调控因子4 (RGS4)的抑制剂。 | |||
| M6569 | CCG 63802 | CCG 63802 | Others |
| ccg63802是g蛋白信号调节蛋白4 (RGS4)的抑制剂。 | |||
| M6581 | CGH 2466 dihydrochloride | CGH 2466 dihydrochloride | Others |
| CGH 2466二盐酸盐是腺苷A1、A2B和A3受体拮抗剂(IC50值分别为19、21和80 nM)。也抑制p38 MAPK (IC50 = 187 - 400 nM)和4D型磷酸二酯酶(IC50 = 22 nM)。在体内和体外都有有效的抗炎作用。对哮喘和慢性阻塞性肺疾病(COPD)的研究可能有用。 | |||
| M6582 | CGP 12177 hydrochloride | CGP 12177 hydrochloride | Others |
| 盐酸CGP 12177是β3肾上腺素受体的部分激动剂。β1-和β2-肾上腺素受体拮抗剂(β1， β2和β3受体的Ki值分别为0.9,4和88 nM)。 | |||
| M6583 | CGP 36216 hydrochloride | CGP 36216 hydrochloride | Others |
| 盐酸CGP 36216是一种选择性的GABAB拮抗剂。显示突触前受体的活性;在GABAB突触后受体上无效。 | |||
| M6584 | CGP 39551 | CGP 39551 | Others |
| CGP 39551是一种强效、选择性和竞争性的NMDA拮抗剂。 | |||
| M6586 | CGP 53353 | CGP 53353 | Others |
| CGP 53353是PKCβII的选择性抑制剂。 | |||
| M6587 | CGP 54626 hydrochloride | CGP 54626 hydrochloride | Others |
| CGP 54626盐酸盐是一种有效的、选择性的GABAB受体拮抗剂(IC50 = 4 nM)。 | |||
| M6588 | CGP 55845 hydrochloride | CGP 55845 hydrochloride | Others |
| CGP 55845盐酸盐是一种有效的，选择性的GABAB受体拮抗剂(IC50 = 5 nM)，防止激动剂结合(pKi = 8.35)和抑制GABA和谷氨酸释放(pEC50值分别为8.08和7.85)。抑制GABAB对巴氯芬的反应(异丙肾上腺素试验中IC50 = 130 nM)，并在体外增强对葡萄糖的低血糖反应。 | |||
M6589
|
CGP 60474 | CGP 60474 | CDK |
| CGP60474 是一种高效的抗内毒素活性化合物，是一种有效的细胞周期蛋白依赖激酶 (CDK) 抑制剂 (CDK1/B、CDK2/E、CDK2/a、CDK4/D、CDK5/p25、CDK7/H 和 CDK9/T 的 IC50 值分别为 26、3、4、216、10、200 和 13 nM)。CGP60474 是一种选择性和 ATP 竞争性 PKC 抑制剂。 | |||
| M6590 | CGS 12066B dimaleate | CGS 12066B dimaleate | Others |
| CGS 12066B双马来酸酯是5-HT1B完全激动剂，比5-HT1A选择性高10倍，比5-HT2C选择性高1000倍。中央主动跟踪系统管理。 | |||
| M6591 | CGS 19755 | CGS 19755 | Others |
| CGS 19755是一种强有力的、有竞争力的NMDA拮抗剂。 | |||
| M6658 | DCG IV | DCG IV | Others |
| DCG IV is a very potent, selective group II mGlu agonist. Also NMDA agonist. | |||
| M7215
|
Rp-8-pCPT-cGMPS sodium | Rp-8-pCPT-cGMPS sodium | PKG |
| Rp-8-pCPT-cGMPS sodium is a pKG inhibitor. | |||
| M7687 | CGS-12066 maleate salt | CGS-12066 maleate salt | Others |
| 5-HT1B serotonin receptor agonist. | |||
| M7695 | CGS-9343B | CGS-9343B | Others |
| CGS-9343B is a selective calmodulin antagonist with minimal protein kinase C or antidopaminergic activity. | |||
| M7699
|
CGS-15943 | CGS-15943 | Adenosine Receptor |
| Highly potent, non-selective adenosine receptor antagonist. | |||
| M7702
|
CGP-20712A methanesulfonate salt | CGP-20712A methanesulfonate salt | Adrenergic Receptor |
| CGP 20712 A | |||
| CGP-20712A methanesulfonate salt 是一种高效性的，选择性的 β1 肾上腺素受体拮抗剂，IC50为 0.7 nM。CGP 20712A 具有抗高血压活性，可逆转 RKT 诱导的胃松弛。 | |||
| M7717 | CGP 52608 | CGP 52608 | Others |
| CGP 52608 is a specific activator of retinoic acid receptor-related orphan receptor α (RORA). | |||
| M7998 | PET-cGMP | PET-cGMP | Others |
| cGMP-dependent protein kinase (PKG I and PKG II) activator. | |||
| M8214 | CGP 37849 | CGP 37849 | Others |
| CGP 37849 induces phencyclidine-like behavioral syndrome in amygdala-kindled rats that includes ataxia, locomotion and stereotypies. | |||
| M8287 | CGP77675 | CGP77675 | Others |
| CGP77675 is a potent Src kinase inhibitor. | |||
| M8314 | CGS 9895 | CGS 9895 | Others |
| CGS 9895 is a GABA antagonist that acts via the benzodiazepine binding site of ag containing GABA receptors. | |||
| M8360 | CGP36742 | CGP36742 | Others |
| CGP36742 was the first orally active GABAB-selective antagonist. | |||
| M8585 | Rp-8-Br-cGMPS sodium salt | Rp-8-Br-cGMPS sodium salt | Others |
| Rp-8-bromo-cGMPS is a cell permeable cGMP analog that blocks cGMP-dependent protein kinase (cGK, G-kinase, Protein Kinase G, PKG). | |||
| M8923
|
CCG215022 | CCG215022 | PKA |
| CCG215022 是一种G蛋白偶联受体激酶 (GRK) 抑制剂，作用于 GRK2，GRK5 和 GRK1，IC50 分别为 0.15±0.07 μM，0.38±0.06 μM 和 3.9±1 μM。 | |||
| M11840 | ChemBridge-5217444 | ChemBridge化合物-5217444 | Screening Compounds and Building Blocks |
| 6-(1,3-dioxo-1H-benzo[de]isoquinolin-2(3H)-yl)-N-hydroxyhexanamide (5217444) | |||
| ChemBridge特有类药化合物/先导化合物-5217444，由AbMole（奥默生物）独家提供。具体售价货期请咨询AbMole（奥默生物）。运费额外计算。 | |||
| M12841 | ChemBridge-7003154 | ChemBridge化合物-7003154 | Screening Compounds and Building Blocks |
| methyl N-[(4-chlorophenyl)sulfonyl]-4-nitrobenzenesulfinimidoate (7003154) | |||
| ChemBridge特有类药化合物/先导化合物-7003154，由AbMole（奥默生物）独家提供。具体售价货期请咨询AbMole（奥默生物）。运费额外计算。 | |||
| M18653 | EGCG Octaacetate | 乙酰化EGCG | Others |
| EGCG Octaacetate 乙酰化EGCG | |||
| M21338
|
Recombinant Human FGF1/ECGF Protein (154AA, E.coli) | 重组人FGF1/ECGF 蛋白 (154AA, E.coli) | Cytokines and Growth Factors |
| ECGS; HBGF-1; FGF-a; FGF-acidic | |||
| FGF acid, also known as ECGF, FGF-1 and HBGF-1, is a non-glycosylated heparin-binding growth factor expressed in brain, kidney, retina, smooth muscle cells, bone stroma, osteoblasts, astrocytes and endothelial cells. | |||
| M49940
|
Recombinant Rat IL-2 (HEK293, C-6His) | 重组大鼠IL-2 (HEK293, C-6His) | Cytokines and Growth Factors |
| Interleukin-2 | |||
| Interleukin-2 (IL-2) is a O-glycosylated four α-helix bundle cytokine that has potent stimulatory activity for antigenactivated T cells. IL-2 stimulates growth and differentiation of B-cells, NK cells, lymphokine-activated killer cells, monocytes, macrophages and oligodendrocytes. | |||
