找到约 24 条 “AM404” 相关结果 (用时 0.111 秒)
目录号 | 产品名称 | 中文名称 | 靶点 |
---|---|---|---|
M11426 | AM404 | AM404 | Cannabinoid |
N-(4-HYDROXYPHENYL)-ARACHIDONYLAMIDE | |||
AM404 是一种内源性大麻素再摄取抑制剂,可阻断 anandamide 转运,IC50 值在低微摩尔范围。去氧肾上腺素使大鼠离体肝动脉收缩,AM404 可使其放松,pEC50 值为 7.4 (对应的 EC50 值为 0.04 µM)。具有神经保护作用。 | |||
M12007 | ChemBridge-5340426 | ChemBridge化合物-5340426 | Screening Compounds and Building Blocks |
5-nitro-N-(4-nitrophenyl)spiro[benzimidazole-2,1'-cyclohexan]-4-amine (5340426) | |||
ChemBridge特有类药化合物/先导化合物-5340426,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M12066 | ChemBridge-5404078 | ChemBridge化合物-5404078 | Screening Compounds and Building Blocks |
3-[(4-chlorophenyl)amino]-3-(4-ethoxyphenyl)-1-phenyl-1-propanone (5404078) | |||
ChemBridge特有类药化合物/先导化合物-5404078,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M12632 | ChemBridge-6234042 | ChemBridge化合物-6234042 | Screening Compounds and Building Blocks |
N-(4-iodophenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine (6234042) | |||
ChemBridge特有类药化合物/先导化合物-6234042,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M12779 | ChemBridge-6781404 | ChemBridge化合物-6781404 | Screening Compounds and Building Blocks |
4-butoxy-N-(2-fluorophenyl)benzamide (6781404) | |||
ChemBridge特有类药化合物/先导化合物-6781404,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M12910 | ChemBridge-7404415 | ChemBridge化合物-7404415 | Screening Compounds and Building Blocks |
2-bromo-N-{[(2-sec-butylphenyl)amino]carbonothioyl}benzamide (7404415) | |||
ChemBridge特有类药化合物/先导化合物-7404415,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M25079 | Zeluvalimab | Zeluvalimab | PD-1/PD-L1 |
AMG-404 | |||
Zeluvalimab (AMG-404) 是一种靶向 PD-1 受体的单克隆抗体,可用于癌症的研究。 | |||
M45693 | ChemBridge-5754048 | ChemBridge化合物-5754048 | Screening Compounds and Building Blocks |
4-(acetylamino)-N-(1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)benzamide (5754048) | |||
ChemBridge特有类药化合物/先导化合物-5754048,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M46137 | ChemBridge-7404199 | ChemBridge化合物-7404199 | Screening Compounds and Building Blocks |
N-(5-isopropyl-1,3,4-thiadiazol-2-yl)-2-(4-methylphenyl)acetamide (7404199) | |||
ChemBridge特有类药化合物/先导化合物-7404199,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M47741 | ChemBridge-28624042 | ChemBridge化合物-28624042 | Screening Compounds and Building Blocks |
N-[(5-fluoro-1H-benzimidazol-2-yl)methyl]-5-isoxazol-5-yl-2-methylthiophene-3-sulfonamide (28624042) | |||
ChemBridge特有类药化合物/先导化合物-28624042,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M48036 | ChemBridge-40438375 | ChemBridge化合物-40438375 | Screening Compounds and Building Blocks |
4-methoxy-N-methyl-3-(1-methyl-1H-pyrazol-4-yl)benzamide (40438375) | |||
ChemBridge特有类药化合物/先导化合物-40438375,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M48037 | ChemBridge-40473376 | ChemBridge化合物-40473376 | Screening Compounds and Building Blocks |
6-methyl-N-[2-(1H-1,2,4-triazol-5-ylthio)ethyl]quinoline-8-sulfonamide (40473376) | |||
ChemBridge特有类药化合物/先导化合物-40473376,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M48088 | ChemBridge-43334047 | ChemBridge化合物-43334047 | Screening Compounds and Building Blocks |
1'-(4-amino-2-pyrimidinyl)-2-(dimethylamino)-5,6-dihydrospiro[cyclopenta[d]pyrimidine-7,3'-piperidin]-4(3H)-one (43334047) | |||
ChemBridge特有类药化合物/先导化合物-43334047,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M48240 | ChemBridge-49139404 | ChemBridge化合物-49139404 | Screening Compounds and Building Blocks |
N-[(5-isobutylisoxazol-3-yl)methyl]-1-(methylsulfonyl)prolinamide (49139404) | |||
ChemBridge特有类药化合物/先导化合物-49139404,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M48324 | ChemBridge-52340487 | ChemBridge化合物-52340487 | Screening Compounds and Building Blocks |
N-[2-methyl-2-(4-morpholinyl)propyl]-3-(4-{[(3-methylphenyl)acetyl]amino}-1H-pyrazol-1-yl)benzamide (52340487) | |||
ChemBridge特有类药化合物/先导化合物-52340487,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M48369 | ChemBridge-54048714 | ChemBridge化合物-54048714 | Screening Compounds and Building Blocks |
2-(4-fluorophenyl)-N-{[1-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)piperidin-4-yl]methyl}acetamide formate (54048714) | |||
ChemBridge特有类药化合物/先导化合物-54048714,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M48391 | ChemBridge-54940494 | ChemBridge化合物-54940494 | Screening Compounds and Building Blocks |
N-(1H-imidazol-2-ylmethyl)-5-(methylsulfonyl)-4-(3-piperidinyl)-2-pyrimidinamine dihydrochloride (54940494) | |||
ChemBridge特有类药化合物/先导化合物-54940494,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M48603 | ChemBridge-64049092 | ChemBridge化合物-64049092 | Screening Compounds and Building Blocks |
5-tert-butyl-4-[(7,9-dioxo-8-azaspiro[4.5]dec-8-yl)methyl]-2-furamide (64049092) | |||
ChemBridge特有类药化合物/先导化合物-64049092,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M49320 | ChemBridge-98440420 | ChemBridge化合物-98440420 | Screening Compounds and Building Blocks |
1-(hydroxymethyl)-N-[2-(1-methylpiperidin-3-yl)ethyl]cyclopropanecarboxamide (98440420) | |||
ChemBridge特有类药化合物/先导化合物-98440420,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M49959 | ChemBridge-85340456 | ChemBridge化合物-85340456 | Screening Compounds and Building Blocks |
N-[3-({[(2-oxopiperidin-3-yl)amino]carbonyl}amino)phenyl]cyclopentanecarboxamide (85340456) | |||
ChemBridge特有类药化合物/先导化合物-85340456,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M49997 | ChemBridge-17240452 | ChemBridge化合物-17240452 | Screening Compounds and Building Blocks |
N-(3-chloro-4-methylphenyl)-3-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]propanamide (17240452) | |||
ChemBridge特有类药化合物/先导化合物-17240452,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M50084 | ChemBridge-75404391 | ChemBridge化合物-75404391 | Screening Compounds and Building Blocks |
3-(2-aminoethoxy)-4-methyl-N-[2-(4-phenyl-2-pyrimidinyl)ethyl]benzamide acetate (75404391) | |||
ChemBridge特有类药化合物/先导化合物-75404391,由AbMole(奥默生物)独家提供。具体售价货期请咨询AbMole(奥默生物)。运费额外计算。 | |||
M58515
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CDDO-TFEA | CDDO-TFEA | Keap1-Nrf2 |
CDDO-Trifluoethyl amide; RTA 404; TP-500 | |||
CDDO-TFEA (RTA 404; TP-500) 是 CDDO 的三氟乙酰胺衍生物,可以穿过血脑屏障。CDDO 是一种 Nrf2 激活剂,可抑制增殖并诱导各种癌细胞分化和凋亡。CDDO-TFEA 可以增强各种神经退行性疾病模型中的 Nrf2 表达和信号传导。 | |||
M24942 | Vibecotamab | Vibecotamab | Others |
XmAb14045 | |||
Vibecotamab (XmAb14045) 是一种有效的针对 CD123 和 CD3 的双特异性抗体,可刺激T细胞介导的 CD123 表达细胞的靶向杀伤。Vibecotamab 具有抗肿瘤活性,可用于急性髓系白血病研究。 |