找到约 3 条 “ALK inhibitor 1” 相关结果 (用时 0.119 秒)
目录号 | 产品名称 | 中文名称 | 靶点 |
---|---|---|---|
M14877
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ALK inhibitor 1 | ALK inhibitor 1 | ALK |
ALK inhibitor 1 (compound 17) 是一种有效的,嘧啶类 ALK 抑制剂。ALK inhibitor 1 是有效的睾丸特异性丝氨酸/苏氨酸激酶 2 (TSSK2; IC50=31 nM) 和粘着斑激酶 (FAK; IC50=2 nM) 抑制剂。 | |||
M28499 | ALK kinase inhibitor-1 | ALK kinase inhibitor-1 | ALK |
ALK kinase inhibitor-1 是一种间变性淋巴瘤激酶 ALK 抑制剂。 | |||
M20633 | TP0427736 HCl | TP0427736 HCl | Src-bcr-Abl |
TP0427736 is a potent inhibitor of ALK5 kinase activity with an IC50 of 2.72 nM and this effect is 300-fold higher than the inhibitory effect on ALK3 (IC50 = 836 nM for ALK3). It also inhibits Smad2/3 phosphorylation in A549 cells induced by TGF-β1 with an IC50 value of 8.68 nM. |