找到约 5 条 “155-84-0” 相关结果 (用时 0.727 秒)
目录号 | 产品名称 | 中文名称 | 靶点 |
---|---|---|---|
M3127
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VUF 10166 | VUF 10166 | 5-HT Receptor |
VUF 10166是一种新型有效的,竞争性5-HT3A受体拮抗剂,Ki为0.04 nM,对5-HT3AB受体的亲和力显著下降。 | |||
M14356 | N-Acetyl-L-arginine | N-Acetyl-L-arginine | Metabolite/Endogenous Metabolite |
Ac-Arg-OH | |||
N-Acetyl-L-arginine (Ac-Arg-OH) 是一种被发现存在于血液渗析性肾不足儿童患者血清中的,胍基诺化合物。 | |||
M19867
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Gatifloxacin hydrochloride | Gatifloxacin hydrochloride | Topoisomerase |
AM-1155 hydrochloride; CG5501 hydrochloride; BMS-206584 hydrochloride; PD135432 hydrochloride | |||
Gatifloxacin (AM-1155, CG5501, BMS-206584, PD135432) hydrochloride is a potent fluoroquinolone antibiotic with broad-spectrum antibacterial activity. Gatifloxacin hydrochloride inhibits bacterial type II topoisomerases with IC50 of 13.8 μg/ml and 0.109 μg/ml for S. aureus topoisomerase IV and E. coli DNA gyrase, respectively. | |||
M28883 | Gatifloxacin sesquihydrate | Gatifloxacin sesquihydrate | Antibiotic |
AM-1155 sesquihydrate; BMS-206584 sesquihydrate; PD135432 sesquihydrate | |||
Gatifloxacin sesquihydrate (AM-1155 sesquihydrate) 是一种有效的氟喹诺酮类抗生素 (antibiotic),具有广谱抗菌活性。Gatifloxacin sesquihydrate (AM-1155 sesquihydrate) 可抑制细菌 II 型拓扑异构酶 (type II topoisomerases) (IC50=13.8 μg/ml; 金黄色葡萄球菌拓扑异构酶 IV) 和大肠杆菌 DNA 解旋酶 (IC50=0.109 μg/ml)。 | |||
M29902 | Gatifloxacin mesylate | 甲磺酸加替沙星 | Antibiotic |
AM-1155 mesylate; BMS-206584 mesylate; PD135432 mesylate | |||
Gatifloxacin mesylate (AM-1155 mesylate) 是一种有效的氟喹诺酮类抗生素 (antibiotic),具有广谱抗菌活性。Gatifloxacin mesylate (AM-1155 mesylate) 可抑制细菌 II 型拓扑异构酶 (type II topoisomerases) (IC50=13.8 μg/ml; 金黄色葡萄球菌拓扑异构酶 IV) 和大肠杆菌 DNA 解旋酶 (IC50=0.109 μg/ml)。 |